Pd-Catalyzed N-Arylation of Heteroarylamines
Yin, Jingjun, Zhao, Matthew M, Huffman, Mark A, McNamara, James M
Published in Organic letters (03.10.2002)
Published in Organic letters (03.10.2002)
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Efficient Synthesis of NK1 Receptor Antagonist Aprepitant Using a Crystallization-Induced Diastereoselective Transformation
Brands, Karel M. J, Payack, Joseph F, Rosen, Jonathan D, Nelson, Todd D, Candelario, Alexander, Huffman, Mark A, Zhao, Matthew M, Li, Jing, Craig, Bridgette, Song, Zhiguo J, Tschaen, David M, Hansen, Karl, Devine, Paul N, Pye, Philip J, Rossen, Kai, Dormer, Peter G, Reamer, Robert A, Welch, Christopher J, Mathre, David J, Tsou, Nancy N, McNamara, James M, Reider, Paul J
Published in Journal of the American Chemical Society (26.02.2003)
Published in Journal of the American Chemical Society (26.02.2003)
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Stereoselective Synthesis of a Potent Thrombin Inhibitor by a Novel P2−P3 Lactone Ring Opening
Nelson, Todd D, LeBlond, Carl R, Frantz, Doug E, Matty, Louis, Mitten, Jeffrey V, Weaver, Damian G, Moore, Jeffrey C, Kim, Jaehon M, Boyd, Russell, Kim, Pei-Yi, Gbewonyo, Kodzo, Brower, Mark, Sturr, Michael, McLaughlin, Kathleen, McMasters, Daniel R, Kress, Michael H, McNamara, James M, Dolling, Ulf H
Published in Journal of organic chemistry (28.05.2004)
Published in Journal of organic chemistry (28.05.2004)
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Practical Asymmetric Synthesis of Aprepitant, a Potent Human NK-1 Receptor Antagonist, via a Stereoselective Lewis Acid-Catalyzed Trans Acetalization Reaction
Zhao, Matthew M, McNamara, James M, Ho, Guo-Jie, Emerson, Khateeta M, Song, Zhiguo J, Tschaen, David M, Brands, Karel M. J, Dolling, Ulf-H, Grabowski, Edward J. J, Reider, Paul J, Cottrell, Ian F, Ashwood, Michael S, Bishop, Brian C
Published in Journal of organic chemistry (20.09.2002)
Published in Journal of organic chemistry (20.09.2002)
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Practical routes to the triarylsulfonyl chloride intermediate of a β3 adrenergic receptor agonist
Ikemoto, Norihiro, Liu, Jinchu, Brands, Karel M.J, McNamara, James M, Reider, Paul J
Published in Tetrahedron (01.02.2003)
Published in Tetrahedron (01.02.2003)
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Journal Article
Synthesis of a Tetrahydropyran NK1 Receptor Antagonist via Asymmetric Conjugate Addition
Huffman, Mark A, Smitrovich, Jacqueline H, Rosen, Jonathan D, Boice, Geneviève N, Qu, Chuanxing, Nelson, Todd D, McNamara, James M
Published in Journal of organic chemistry (27.05.2005)
Published in Journal of organic chemistry (27.05.2005)
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Journal Article
A very concise synthesis of a potent N-(1,3-thiazol-2-yl)pyridin-2-amine KDR kinase inhibitor
Zhao, Matthew, Yin, Jingjun, Huffman, Mark A., McNamara, James M.
Published in Tetrahedron (06.02.2006)
Published in Tetrahedron (06.02.2006)
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Journal Article
Synthesis of a NO-Releasing Prodrug of Rofecoxib
Engelhardt, F. Conrad, Shi, Yao-Jun, Cowden, Cameron J, Conlon, David A, Pipik, Brenda, Zhou, George, McNamara, James M, Dolling, Ulf-H
Published in Journal of organic chemistry (20.01.2006)
Published in Journal of organic chemistry (20.01.2006)
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Efficient Synthesis of a Highly Selective NPY-5 Receptor Antagonist: A Drug Candidate for the Treatment of Obesity
Itoh, Takahiro, Kato, Shinji, Nonoyama, Nobuaki, Wada, Toshihiro, Maeda, Kenji, Mase, Toshiaki, Zhao, Matthew M, Song, Jake Z, Tschaen, David M, McNamara, James M
Published in Organic process research & development (21.07.2006)
Published in Organic process research & development (21.07.2006)
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Journal Article
Process Development and Large-Scale Synthesis of a PDE4 Inhibitor
Conlon, David A, Drahus-Paone, Antoinette, Ho, Guo-Jie, Pipik, Brenda, Helmy, Roy, McNamara, James M, Shi, Yao-Jun, Williams, J. Michael, Macdonald, Dwight, Deschênes, Denis, Gallant, Michel, Mastracchio, Anthony, Roy, Bruno, Scheigetz, John
Published in Organic process research & development (01.01.2006)
Published in Organic process research & development (01.01.2006)
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Journal Article
One-Pot Preparation of 7-Hydroxyquinoline
Cameron, Mark, Hoerrner, R. Scott, McNamara, James M, Figus, Margaret, Thomas, Scott
Published in Organic process research & development (01.01.2006)
Published in Organic process research & development (01.01.2006)
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Journal Article
A regioselective synthesis of 2,4-dialkyl resorcinols
Ceglia, Scott S., Kress, Michael H., Nelson, Todd D., McNamara, James M.
Published in Tetrahedron letters (07.03.2005)
Published in Tetrahedron letters (07.03.2005)
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A convenient synthesis of 3-aryl-δ-lactones
Rosen, Jonathan D, Nelson, Todd D, Huffman, Mark A, McNamara, James M
Published in Tetrahedron letters (06.01.2003)
Published in Tetrahedron letters (06.01.2003)
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Journal Article
Practical chemoenzymatic synthesis of a 3-pyridylethanolamino β3 adrenergic receptor agonist
Chung, John Y.L, Ho, Guo-Jie, Chartrain, Michel, Roberge, Chris, Zhao, Dalian, Leazer, John, Farr, Roger, Robbins, Michael, Emerson, Kateeta, Mathre, David J, McNamara, James M, Hughes, David L, Grabowski, Edward J.J, Reider, Paul J
Published in Tetrahedron letters (10.09.1999)
Published in Tetrahedron letters (10.09.1999)
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A Highly Efficient Synthesis of Fibrinogen Receptor Antagonist L-734,217 via a Novel Chemoselective Silyl-Mediated Conjugate Addition of δ-Lactams to 4-Vinylpyridine
Chung, John Y. L, Hughes, David L, Zhao, Dalian, Song, Zhiguo, Mathre, David J, Ho, Guo-Jie, McNamara, James M, Douglas, Alan W, Reamer, R. A, Tsay, Fuh-Rong, Varsolona, Richard, McCauley, James, Grabowski, Edward J. J, Reider, Paul J
Published in Journal of organic chemistry (12.01.1996)
Published in Journal of organic chemistry (12.01.1996)
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