An integrated console for capsule-based, automated organic synthesis
Jiang, Tuo, Bordi, Samuele, McMillan, Angus E, Chen, Kuang-Yen, Saito, Fumito, Nichols, Paula L, Wanner, Benedikt M, Bode, Jeffrey W
Published in Chemical science (Cambridge) (28.05.2021)
Published in Chemical science (Cambridge) (28.05.2021)
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Reagent-Based Scaffold Diversity for DNA-Encoded Library Design: Solid Phase Synthesis of DNA-Tagged sp 3 -Rich Heterocycles by SnAP Chemistry
Škopić, Mateja Klika, Losch, Florian, McMillan, Angus E, Willeke, Niklas, Malenica, Mateo, Bering, Luis, Bode, Jeffrey, Brunschweiger, Andreas
Published in Organic letters (18.02.2022)
Published in Organic letters (18.02.2022)
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Stereoretentive Etherification of an α‑Aryl-β-amino Alcohol Using a Selective Aziridinium Ring Opening for the Synthesis of AZD7594
McMillan, Angus E, Steven, Alan, Ashworth, Ian W, Mullen, Alexander K, Chan, Lai C, Galan Espinosa, Maria Rita, Pilling, Michael J, Raw, Steven A, Jones, Martin F
Published in Journal of organic chemistry (19.04.2019)
Published in Journal of organic chemistry (19.04.2019)
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Route Design to Manufacture: Synthesis of the Heterocyclic Fragment of AZD5718 Using a Non-cryogenic Lithiation-Alkoxycarbonylation Reaction
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Published in Organic process research & development (16.04.2021)
Published in Organic process research & development (16.04.2021)
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Rapid route design of AZD7594
Carter, Holly L, Connor, Amand W, Hart, Richard, McCabe, James, McIntyre, Allyson C, McMillan, Angus E, Monks, Natalie R, Mullen, Alexander K, Ronson, Thomas O, Steven, Alan, Tomasi, Simone, Yates, Simon D
Published in Reaction chemistry & engineering (01.09.2019)
Published in Reaction chemistry & engineering (01.09.2019)
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Reagent-Based Scaffold Diversity for DNA-Encoded Library Design: Solid Phase Synthesis of DNA-Tagged sp(3)-Rich Heterocycles by SnAP Chemistry
Skopic, Mateja Klika, Losch, Florian, McMillan, Angus E., Willeke, Niklas, Malenica, Mateo, Bering, Luis, Bode, Jeffrey, Brunschweiger, Andreas
Published in Organic letters (18.02.2022)
Published in Organic letters (18.02.2022)
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Journal Article
Reagent-Based Scaffold Diversity for DNA-Encoded Library Design: Solid Phase Synthesis of DNA-Tagged sp3‑Rich Heterocycles by SnAP Chemistry
Škopić, Mateja Klika, Losch, Florian, McMillan, Angus E, Willeke, Niklas, Malenica, Mateo, Bering, Luis, Bode, Jeffrey, Brunschweiger, Andreas
Published in Organic letters (18.02.2022)
Published in Organic letters (18.02.2022)
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Structural diversification of the aminobicyclo[4.3.0]nonane skeleton using alkynylsilyl-derived allylic trichloroacetimidatesElectronic supplementary information (ESI) available: NOE data for compounds 16-25 and, 1H and 13C NMR spectra of all compounds. See DOI: 10.1039/c7ob00456g
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