Discovery of GNE-502 as an orally bioavailable and potent degrader for estrogen receptor positive breast cancer
Zbieg, Jason R., Liang, Jun, Li, Jun, Blake, Robert A., Chang, Jae, Friedman, Lori, Goodacre, Simon, Hartman, Steven J., Rei Ingalla, Ellen, Kiefer, James R., Kleinheinz, Tracy, Labadie, Sharada, Lai, Tommy, Liao, Jiangpeng, McLean, Nev, Metcalfe, Ciara, Mody, Vidhi, Nannini, Michelle, Ortwine, Daniel F., Ran, Yingqing, Ray, Nick, Roussel, Fabien, Sambrone, Amy, Sampath, Deepak, Vinogradova, Maia, Wai, John, Wang, Tao, Yeap, Kuen, Zhang, Birong, Zheng, Xiaoping, Zhong, Yu, Wang, Xiaojing
Published in Bioorganic & medicinal chemistry letters (15.10.2021)
Published in Bioorganic & medicinal chemistry letters (15.10.2021)
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