Discovery of a Covalent FEM1B Recruiter for Targeted Protein Degradation Applications
Henning, Nathaniel J, Manford, Andrew G, Spradlin, Jessica N, Brittain, Scott M, Zhang, Erika, McKenna, Jeffrey M, Tallarico, John A, Schirle, Markus, Rape, Michael, Nomura, Daniel K
Published in Journal of the American Chemical Society (19.01.2022)
Published in Journal of the American Chemical Society (19.01.2022)
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Harnessing the anti-cancer natural product nimbolide for targeted protein degradation
Spradlin, Jessica N, Hu, Xirui, Ward, Carl C, Brittain, Scott M, Jones, Michael D, Ou, Lisha, To, Milton, Proudfoot, Andrew, Ornelas, Elizabeth, Woldegiorgis, Mikias, Olzmann, James A, Bussiere, Dirksen E, Thomas, Jason R, Tallarico, John A, McKenna, Jeffrey M, Schirle, Markus, Maimone, Thomas J, Nomura, Daniel K
Published in Nature chemical biology (01.07.2019)
Published in Nature chemical biology (01.07.2019)
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PARP-1 Activation Requires Local Unfolding of an Autoinhibitory Domain
Dawicki-McKenna, Jennine M., Langelier, Marie-France, DeNizio, Jamie E., Riccio, Amanda A., Cao, Connie D., Karch, Kelly R., McCauley, Michael, Steffen, Jamin D., Black, Ben E., Pascal, John M.
Published in Molecular cell (03.12.2015)
Published in Molecular cell (03.12.2015)
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Engagement of MHC class I by the inhibitory receptor LILRB1 suppresses macrophages and is a target of cancer immunotherapy
Barkal, Amira A, Weiskopf, Kipp, Kao, Kevin S, Gordon, Sydney R, Rosental, Benyamin, Yiu, Ying Y, George, Benson M, Markovic, Maxim, Ring, Nan G, Tsai, Jonathan M, McKenna, Kelly M, Ho, Po Yi, Cheng, Robin Z, Chen, James Y, Barkal, Layla J, Ring, Aaron M, Weissman, Irving L, Maute, Roy L
Published in Nature immunology (01.01.2018)
Published in Nature immunology (01.01.2018)
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A new conceptual framework for the transformation of groundwater dissolved organic matter
McDonough, Liza K, Andersen, Martin S, Behnke, Megan I, Rutlidge, Helen, Oudone, Phetdala, Meredith, Karina, O'Carroll, Denis M, Santos, Isaac R, Marjo, Christopher E, Spencer, Robert G M, McKenna, Amy M, Baker, Andy
Published in Nature communications (20.04.2022)
Published in Nature communications (20.04.2022)
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Covalent Ligand Screening Uncovers a RNF4 E3 Ligase Recruiter for Targeted Protein Degradation Applications
Ward, Carl C, Kleinman, Jordan I, Brittain, Scott M, Lee, Patrick S, Chung, Clive Yik Sham, Kim, Kenneth, Petri, Yana, Thomas, Jason R, Tallarico, John A, McKenna, Jeffrey M, Schirle, Markus, Nomura, Daniel K
Published in ACS chemical biology (15.11.2019)
Published in ACS chemical biology (15.11.2019)
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Bardoxolone conjugation enables targeted protein degradation of BRD4
Tong, Bingqi, Luo, Mai, Xie, Yi, Spradlin, Jessica N, Tallarico, John A, McKenna, Jeffrey M, Schirle, Markus, Maimone, Thomas J, Nomura, Daniel K
Published in Scientific reports (23.09.2020)
Published in Scientific reports (23.09.2020)
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Discovery of a Functional Covalent Ligand Targeting an Intrinsically Disordered Cysteine within MYC
Boike, Lydia, Cioffi, Alexander G., Majewski, Felix C., Co, Jennifer, Henning, Nathaniel J., Jones, Michael D., Liu, Gang, McKenna, Jeffrey M., Tallarico, John A., Schirle, Markus, Nomura, Daniel K.
Published in Cell chemical biology (21.01.2021)
Published in Cell chemical biology (21.01.2021)
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Macrophages eat cancer cells using their own calreticulin as a guide: Roles of TLR and Btk
Feng, Mingye, Chen, James Y., Weissman-Tsukamoto, Rachel, Volkmer, Jens-Peter, Ho, Po Yi, McKenna, Kelly M., Cheshier, Samuel, Zhang, Michael, Guo, Nan, Gip, Phung, Mitra, Siddhartha S., Weissman, Irving L.
Published in Proceedings of the National Academy of Sciences - PNAS (17.02.2015)
Published in Proceedings of the National Academy of Sciences - PNAS (17.02.2015)
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1.1-billion-year-old porphyrins establish a marine ecosystem dominated by bacterial primary producers
Gueneli, N., McKenna, A. M., Ohkouchi, N., Boreham, C. J., Beghin, J., Javaux, E. J., Brocks, J. J.
Published in Proceedings of the National Academy of Sciences - PNAS (24.07.2018)
Published in Proceedings of the National Academy of Sciences - PNAS (24.07.2018)
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Contractile properties and sarcoplasmic reticulum calcium content in type I and type II skeletal muscle fibres in active aged humans
Lamboley, C. R., Wyckelsma, V. L., Dutka, T. L., McKenna, M. J., Murphy, R. M., Lamb, G. D.
Published in The Journal of physiology (01.06.2015)
Published in The Journal of physiology (01.06.2015)
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Bioactivity of Humic Acids Extracted From Shale Ore: Molecular Characterization and Structure-Activity Relationship With Tomato Plant Yield Under Nutritional Stress
Monda, Hiarhi, McKenna, Amy M., Fountain, Ryan, Lamar, Richard T.
Published in Frontiers in plant science (26.05.2021)
Published in Frontiers in plant science (26.05.2021)
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Assessing the Risk of Ships Striking Large Whales in Marine Spatial Planning
REDFERN, J. V., MCKENNA, M. F., MOORE, T. J., CALAMBOKIDIS, J., DEANGELIS, M. L., BECKER, E. A., BARLOW, J., FORNEY, K. A., FIEDLER, P. C., CHIVERS, S. J.
Published in Conservation biology (01.04.2013)
Published in Conservation biology (01.04.2013)
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Encouraging Healthier Food and Beverage Purchasing and Consumption: A Review of Interventions within Grocery Retail Settings
Wolgast, Henry, Halverson, McKenna M, Kennedy, Nicole, Gallard, Isabel, Karpyn, Allison
Published in International journal of environmental research and public health (01.12.2022)
Published in International journal of environmental research and public health (01.12.2022)
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Unravelling High-Molecular-Weight DBP Toxicity Drivers in Chlorinated and Chloraminated Drinking Water: Effect-Directed Analysis of Molecular Weight Fractions
Dong, Huiyu, Cuthbertson, Amy A, Plewa, Michael J, Weisbrod, Chad R, McKenna, Amy M, Richardson, Susan D
Published in Environmental science & technology (28.11.2023)
Published in Environmental science & technology (28.11.2023)
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