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Structure of human neutrophil elastase in complex with a peptide chloromethyl ketone inhibitor at 1.84-A resolution
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Crystallographic analysis of a complex between human immunodeficiency virus type 1 protease and acetyl-pepstatin at 2.0-A resolution
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Three-dimensional structure of aspartyl protease from human immunodeficiency virus HIV-1
Navia, M A, Fitzgerald, P M, McKeever, B M, Leu, C T, Heimbach, J C, Herber, W K, Sigal, I S, Darke, P L, Springer, J P
Published in Nature (London) (16.02.1989)
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Crystallization of human neutrophil elastase
Williams, H R, Lin, T Y, Navia, M A, Springer, J P, McKeever, B M, Hoogsteen, K, Dorn, C P
Published in The Journal of biological chemistry (15.12.1987)
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Positions of His‐64 and a bound water in human carbonic anhydrase II upon binding three structurally related inhibitors
Smith, Graham M., Alexander, Richard S, Christianson, David W., Mckeever, Brian M., Ponticello, Gerald S., Springer, James P., Randall, William C., Baldwin, John J., Habecker, Charles N.
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Thienothiopyran-2-sulfonamides: novel topically active carbonic anhydrase inhibitors for the treatment of glaucoma
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New isomeric classes of topically active ocular hypotensive carbonic anhydrase inhibitors: 5-substituted thieno[2,3-b]thiophene-2-sulfonamides and 5-substituted thieno[3,2-b]thiophene-2-sulfonamides
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Shi, Guo Q, Dropinski, James F, McKeever, Brian M, Xu, Shihua, Becker, Joseph W, Berger, Joel P, MacNaul, Karen L, Elbrecht, Alex, Zhou, Gaochao, Doebber, Thomas W, Wang, Peiran, Chao, Yu-Sheng, Forrest, Mike, Heck, James V, Moller, David E, Jones, A. Brian
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Protein Crystal Growth in Microgravity
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Published in Science (American Association for the Advancement of Science) (03.11.1989)
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Synthesis and antiviral activity of a series of HIV-1 protease inhibitors with functionality tethered to the P sub(1) or P sub(1)' phenyl substituents: X-ray crystal structure assisted design
Thompson, W J, Fitzgerald, PMD, Holloway, M K, Emini, E A, Darke, P L, McKeever, B M, Schleif, WA, Quintero, J C, Zugay, JA
Published in Journal of medicinal chemistry (01.01.1992)
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Published in Journal of medicinal chemistry (01.01.1992)
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