International Union of Pharmacology. LXV. The pharmacology and classification of the nuclear receptor superfamily: glucocorticoid, mineralocorticoid, progesterone, and androgen receptors
Lu, Nick Z, Wardell, Suzanne E, Burnstein, Kerry L, Defranco, Donald, Fuller, Peter J, Giguere, Vincent, Hochberg, Richard B, McKay, Lorraine, Renoir, Jack-Michel, Weigel, Nancy L, Wilson, Elizabeth M, McDonnell, Donald P, Cidlowski, John A
Published in Pharmacological reviews (01.12.2006)
Published in Pharmacological reviews (01.12.2006)
Get full text
Journal Article
Pharmacokinetic/Pharmacodynamic Models for Corticosteroid Receptor Down-Regulation and Glutamine Synthetase Induction in Rat Skeletal Muscle by a Receptor/Gene-Mediated Mechanism
Sun, Y N, McKay, L I, DuBois, D C, Jusko, W J, Almon, R R
Published in The Journal of pharmacology and experimental therapeutics (01.02.1999)
Get full text
Published in The Journal of pharmacology and experimental therapeutics (01.02.1999)
Journal Article
Dimethyl-diphenyl-propanamide Derivatives As Nonsteroidal Dissociated Glucocorticoid Receptor Agonists
Yang, Bingwei V, Weinstein, David S, Doweyko, Lidia M, Gong, Hua, Vaccaro, Wayne, Huynh, Tram, Xiao, Hai-yun, Doweyko, Arthur M, Mckay, Lorraine, Holloway, Deborah A, Somerville, John E, Habte, Sium, Cunningham, Mark, McMahon, Michele, Townsend, Robert, Shuster, David, Dodd, John H, Nadler, Steven G, Barrish, Joel C
Published in Journal of medicinal chemistry (09.12.2010)
Published in Journal of medicinal chemistry (09.12.2010)
Get full text
Journal Article
Discovery of potent and selective nonsteroidal indazolyl amide glucocorticoid receptor agonists
Sheppeck, James E., Gilmore, John L., Xiao, Hai-Yun, Dhar, T.G. Murali, Nirschl, David, Doweyko, Arthur M., Sack, Jack S., Corbett, Martin J., Malley, Mary F., Gougoutas, Jack Z., Mckay, Lorraine, Cunningham, Mark D., Habte, Sium F., Dodd, John H., Nadler, Steven G., Somerville, John E., Barrish, Joel C.
Published in Bioorganic & medicinal chemistry letters (01.10.2013)
Published in Bioorganic & medicinal chemistry letters (01.10.2013)
Get full text
Journal Article
Synthesis and structure–activity relationships of novel indazolyl glucocorticoid receptor partial agonists
Gilmore, John L., Sheppeck, James E., Wang, Jim, Dhar, T.G. Murali, Cavallaro, Cullen, Doweyko, Arthur M., Mckay, Lorraine, Cunningham, Mark D., Habte, Sium F., Nadler, Steven G., Dodd, John H., Somerville, John E., Barrish, Joel C.
Published in Bioorganic & medicinal chemistry letters (01.10.2013)
Published in Bioorganic & medicinal chemistry letters (01.10.2013)
Get full text
Journal Article
Discovery of novel dihydro-9,10-ethano-anthracene carboxamides as glucocorticoid receptor modulators
Yang, Bingwei V., Vaccaro, Wayne, Doweyko, Arthur M., Doweyko, Lidia M., Huynh, Tram, Tortolani, David, Nadler, Steven G., McKay, Lorraine, Somerville, John, Holloway, Deborah A., Habte, Sium, Weinstein, David S., Barrish, Joel C.
Published in Bioorganic & medicinal chemistry letters (15.04.2009)
Published in Bioorganic & medicinal chemistry letters (15.04.2009)
Get full text
Journal Article
Corticosteroid effects in skeletal muscle: Gene induction/receptor autoregulation
McKay, Lorraine I., DuBois, Debra C., Sun, Yu-Nien, Almon, Richard R., Jusko, William J.
Published in Muscle & nerve (01.10.1997)
Published in Muscle & nerve (01.10.1997)
Get full text
Journal Article
Differential dynamics of receptor down-regulation and tyrosine aminotransferase induction following glucocorticoid treatment
DuBois, Debra C., Xu, Zhi-Xin, McKay, Lorraine, Almon, Richard R., Pyszcznski, Nancy, Jusko, William J.
Published in The Journal of steroid biochemistry and molecular biology (01.09.1995)
Published in The Journal of steroid biochemistry and molecular biology (01.09.1995)
Get full text
Journal Article