Highly Selective Inhibition of Tyrosine Kinase 2 (TYK2) for the Treatment of Autoimmune Diseases: Discovery of the Allosteric Inhibitor BMS-986165
Wrobleski, Stephen T, Moslin, Ryan, Lin, Shuqun, Zhang, Yanlei, Spergel, Steven, Kempson, James, Tokarski, John S, Strnad, Joann, Zupa-Fernandez, Adriana, Cheng, Lihong, Shuster, David, Gillooly, Kathleen, Yang, Xiaoxia, Heimrich, Elizabeth, McIntyre, Kim W, Chaudhry, Charu, Khan, Javed, Ruzanov, Max, Tredup, Jeffrey, Mulligan, Dawn, Xie, Dianlin, Sun, Huadong, Huang, Christine, D’Arienzo, Celia, Aranibar, Nelly, Chiney, Manoj, Chimalakonda, Anjaneya, Pitts, William J, Lombardo, Louis, Carter, Percy H, Burke, James R, Weinstein, David S
Published in Journal of medicinal chemistry (24.10.2019)
Published in Journal of medicinal chemistry (24.10.2019)
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Journal Article
Analyzing RNA posttranscriptional modifications to decipher the epitranscriptomic code
Deng, L., Kumar, J., Rose, R., McIntyre, W., Fabris, Daniele
Published in Mass spectrometry reviews (01.01.2024)
Published in Mass spectrometry reviews (01.01.2024)
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Journal Article
Randomized Controlled Trial of Individualized Dialysate Cooling for Cardiac Protection in Hemodialysis Patients
Odudu, Aghogho, Eldehni, Mohamed Tarek, McCann, Gerry P, McIntyre, Christopher W
Published in Clinical journal of the American Society of Nephrology (07.08.2015)
Published in Clinical journal of the American Society of Nephrology (07.08.2015)
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Journal Article
Antiseizure effects of the cannabinoids in the amygdala‐kindling model
Fallah, Merrick S., Dlugosz, Lukasz, Scott, Brian W., Thompson, Miles D., Burnham, W. McIntyre
Published in Epilepsia (Copenhagen) (01.09.2021)
Published in Epilepsia (Copenhagen) (01.09.2021)
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Journal Article
Intradialytic Cardiac Magnetic Resonance Imaging to Assess Cardiovascular Responses in a Short-Term Trial of Hemodiafiltration and Hemodialysis
Buchanan, Charlotte, Mohammed, Azharuddin, Cox, Eleanor, Köhler, Katrin, Canaud, Bernard, Taal, Maarten W, Selby, Nicholas M, Francis, Susan, McIntyre, Chris W
Published in Journal of the American Society of Nephrology (01.04.2017)
Published in Journal of the American Society of Nephrology (01.04.2017)
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Journal Article
The clinical utility and cost impact of cystatin C measurement in the diagnosis and management of chronic kidney disease: A primary care cohort study
Shardlow, Adam, McIntyre, Natasha J, Fraser, Simon D S, Roderick, Paul, Raftery, James, Fluck, Richard J, McIntyre, Christopher W, Taal, Maarten W
Published in PLoS medicine (10.10.2017)
Published in PLoS medicine (10.10.2017)
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Journal Article
Hemodialysis-Induced Repetitive Myocardial Injury Results in Global and Segmental Reduction in Systolic Cardiac Function
Burton, James O, Jefferies, Helen J, Selby, Nicholas M, McIntyre, Christopher W
Published in Clinical journal of the American Society of Nephrology (01.12.2009)
Published in Clinical journal of the American Society of Nephrology (01.12.2009)
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Journal Article
Autoimmune pathways in mice and humans are blocked by pharmacological stabilization of the TYK2 pseudokinase domain
Burke, James R, Cheng, Lihong, Gillooly, Kathleen M, Strnad, Joann, Zupa-Fernandez, Adriana, Catlett, Ian M, Zhang, Yifan, Heimrich, Elizabeth M, McIntyre, Kim W, Cunningham, Mark D, Carman, Julie A, Zhou, Xiadi, Banas, Dana, Chaudhry, Charu, Li, Sha, D'Arienzo, Celia, Chimalakonda, Anjaneya, Yang, XiaoXia, Xie, Jenny H, Pang, Jian, Zhao, Qihong, Rose, Shawn M, Huang, Jinwen, Moslin, Ryan M, Wrobleski, Stephen T, Weinstein, David S, Salter-Cid, Luisa M
Published in Science translational medicine (24.07.2019)
Published in Science translational medicine (24.07.2019)
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Journal Article
Frequent Hemodialysis Schedules Are Associated with Reduced Levels of Dialysis-induced Cardiac Injury (Myocardial Stunning)
Jefferies, Helen J, Virk, Bhupinder, Schiller, Brigitte, Moran, John, McIntyre, Christopher W
Published in Clinical journal of the American Society of Nephrology (01.06.2011)
Published in Clinical journal of the American Society of Nephrology (01.06.2011)
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Journal Article
Impact of Compliance with a Care Bundle on Acute Kidney Injury Outcomes: A Prospective Observational Study
Kolhe, Nitin V, Staples, David, Reilly, Timothy, Merrison, Daniel, Mcintyre, Christopher W, Fluck, Richard J, Selby, Nicholas M, Taal, Maarten W
Published in PloS one (10.07.2015)
Published in PloS one (10.07.2015)
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Journal Article
Bruton's tyrosine kinase inhibitor BMS-986142 in experimental models of rheumatoid arthritis enhances efficacy of agents representing clinical standard-of-care
Gillooly, Kathleen M, Pulicicchio, Claudine, Pattoli, Mark A, Cheng, Lihong, Skala, Stacey, Heimrich, Elizabeth M, McIntyre, Kim W, Taylor, Tracy L, Kukral, Daniel W, Dudhgaonkar, Shailesh, Nagar, Jignesh, Banas, Dana, Watterson, Scott H, Tino, Joseph A, Fura, Aberra, Burke, James R
Published in PloS one (24.07.2017)
Published in PloS one (24.07.2017)
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Journal Article
Use of Electronic Results Reporting to Diagnose and Monitor AKI in Hospitalized Patients
Selby, Nicholas M, Crowley, Lisa, Fluck, Richard J, McIntyre, Christopher W, Monaghan, John, Lawson, Nigel, Kolhe, Nitin V
Published in Clinical journal of the American Society of Nephrology (01.04.2012)
Published in Clinical journal of the American Society of Nephrology (01.04.2012)
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Journal Article
Hemodialysis-Related Acute Brain Injury Demonstrated by Application of Intradialytic Magnetic Resonance Imaging and Spectroscopy
Anazodo, Udunna C, Wong, Dickson Y, Théberge, Jean, Dacey, Madeleine, Gomes, Janice, Penny, Jarrin D, van Ginkel, Michael, Poirier, Stefan E, McIntyre, Christopher W
Published in Journal of the American Society of Nephrology (01.06.2023)
Published in Journal of the American Society of Nephrology (01.06.2023)
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