Preparation of Amino-Substituted Indenes and 1,4-Dihydronaphthalenes Using a One-Pot Multireaction Approach: Total Synthesis of Oxybenzo[c]phenanthridine Alkaloids
Calder, Ewen D. D, McGonagle, Fiona I, Harkiss, Alexander H, McGonagle, Grant A, Sutherland, Andrew
Published in Journal of organic chemistry (15.08.2014)
Published in Journal of organic chemistry (15.08.2014)
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Journal Article
Selective CDK6 degradation mediated by cereblon, VHL, and novel IAP-recruiting PROTACs
Anderson, Niall A., Cryan, Jenni, Ahmed, Adil, Dai, Han, McGonagle, Grant A., Rozier, Christine, Benowitz, Andrew B.
Published in Bioorganic & medicinal chemistry letters (01.05.2020)
Published in Bioorganic & medicinal chemistry letters (01.05.2020)
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Journal Article
Targeting IRAK4 for Degradation with PROTACs
Nunes, Joao, McGonagle, Grant A, Eden, Jessica, Kiritharan, Girieshanie, Touzet, Megane, Lewell, Xiao, Emery, John, Eidam, Hilary, Harling, John D, Anderson, Niall A
Published in ACS medicinal chemistry letters (11.07.2019)
Published in ACS medicinal chemistry letters (11.07.2019)
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Discovery of GSK251: A Highly Potent, Highly Selective, Orally Bioavailable Inhibitor of PI3Kδ with a Novel Binding Mode
Down, Kenneth, Amour, Augustin, Anderson, Niall A, Barton, Nick, Campos, Sebastien, Cannons, Edward P, Clissold, Cole, Convery, Maire A, Coward, John J, Doyle, Kevin, Duempelfeld, Birgit, Edwards, Christopher D, Goldsmith, Michael D, Krause, Jana, Mallett, David N, McGonagle, Grant A, Patel, Vipulkumar K, Rowedder, James, Rowland, Paul, Sharpe, Andrew, Sriskantharajah, Srividya, Thomas, Daniel A, Thomson, Douglas W, Uddin, Sorif, Hamblin, J. Nicole, Hessel, Edith M
Published in Journal of medicinal chemistry (23.09.2021)
Published in Journal of medicinal chemistry (23.09.2021)
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