Formal Syntheses of Naturally Occurring Welwitindolinones
Fu, Tsung-hao, McElroy, William T, Shamszad, Mariam, Martin, Stephen F
Published in Organic letters (03.08.2012)
Published in Organic letters (03.08.2012)
Get full text
Journal Article
Studies toward welwitindolinones: formal syntheses of N-methylwelwitindolinone C isothiocyanate and related natural products
Fu, Tsung-hao, McElroy, William T., Shamszad, Mariam, Heidebrecht, Richard W., Gulledge, Brian, Martin, Stephen F.
Published in Tetrahedron (08.07.2013)
Published in Tetrahedron (08.07.2013)
Get full text
Journal Article
Efforts towards the optimization of a bi-aryl class of potent IRAK4 inhibitors
Hanisak, Jennifer, Seganish, W. Michael, McElroy, William T., Tang, Haiquin, Zhang, Rui, Tsui, Hon-Chung, Fischmann, Theirry, Tulshian, Deen, Tata, James, Sondey, Christopher, Devito, Kristine, Fossetta, James, Garlisi, Charles G., Lundell, Daniel, Niu, Xiaoda
Published in Bioorganic & medicinal chemistry letters (01.09.2016)
Published in Bioorganic & medicinal chemistry letters (01.09.2016)
Get full text
Journal Article
Discovery of orally active pyrazoloquinolines as potent PDE10 inhibitors for the management of schizophrenia
Yang, Shu-Wei, Smotryski, Jennifer, McElroy, William T., Tan, Zheng, Ho, Ginny, Tulshian, Deen, Greenlee, William J., Guzzi, Mario, Zhang, Xiaoping, Mullins, Deborra, Xiao, Li, Hruza, Alan, Chan, Tze-Ming, Rindgen, Diane, Bleickardt, Carina, Hodgson, Robert
Published in Bioorganic & medicinal chemistry letters (01.01.2012)
Published in Bioorganic & medicinal chemistry letters (01.01.2012)
Get full text
Journal Article
Potent and Selective Amidopyrazole Inhibitors of IRAK4 That Are Efficacious in a Rodent Model of Inflammation
McElroy, William T., Tan, Zheng, Ho, Ginny, Paliwal, Sunil, Li, Guoqing, Seganish, W. Michael, Tulshian, Deen, Tata, James, Fischmann, Thierry O., Sondey, Christopher, Bian, Hong, Bober, Loretta, Jackson, James, Garlisi, Charles G., Devito, Kristine, Fossetta, James, Lundell, Daniel, Niu, Xiaoda
Published in ACS medicinal chemistry letters (11.06.2015)
Published in ACS medicinal chemistry letters (11.06.2015)
Get full text
Journal Article
Discovery and hit-to-lead optimization of 2,6-diaminopyrimidine inhibitors of interleukin-1 receptor-associated kinase 4
McElroy, William T., Seganish, W. Michael, Herr, R. Jason, Harding, James, Yang, Jinhai, Yet, Larry, Komanduri, Venukrishnan, Prakash, Koraboina Chandra, Lavey, Brian, Tulshian, Deen, Greenlee, William J., Sondey, Christopher, Fischmann, Thierry O., Niu, Xiaoda
Published in Bioorganic & medicinal chemistry letters (01.05.2015)
Published in Bioorganic & medicinal chemistry letters (01.05.2015)
Get full text
Journal Article
High-Throughput Screening to Identify Small Molecules That Selectively Inhibit APOL1 Protein Level in Podocytes
Choy, Jonathan, Kan, Yanqing, Cifelli, Steve, Johnson, Josephine, Chen, Michelle, Shiao, Lin-Lin, Zhou, Haihong, Previs, Stephen, Lei, Ying, Johnstone, Richard, Liaw, Andy, Saigal, Ashmita, Hu, Lufei, Ramos, Robert, Visconti, Richard, McElroy, William T., Kreamer, Anthony, Wildey, Mary-Jo, Peier, Andrea, Shin, Myung K., Imbriglio, Jason, Ren, Zhao, Hoek, Maarten, Weinglass, Adam, Ai, Xi
Published in SLAS discovery (01.10.2021)
Published in SLAS discovery (01.10.2021)
Get full text
Journal Article
Initial optimization and series evolution of diaminopyrimidine inhibitors of interleukin-1 receptor associated kinase 4
Seganish, W. Michael, McElroy, William T., Herr, R. Jason, Brumfield, Stephanie, Greenlee, William J., Harding, James, Komanduri, Venukrishnan, Matasi, Julius, Prakash, Koraboina Chandra, Tulshian, Deen, Yang, Jinhai, Yet, Larry, Devito, Kristine, Fossetta, James, Garlisi, Charles G., Lundell, Daniel, Niu, Xiaoda, Sondey, Christopher
Published in Bioorganic & medicinal chemistry letters (15.08.2015)
Published in Bioorganic & medicinal chemistry letters (15.08.2015)
Get full text
Journal Article
Discovery and Structure Enabled Synthesis of 2,6-Diaminopyrimidin-4-one IRAK4 Inhibitors
Seganish, W. Michael, Fischmann, Thierry O, Sherborne, Brad, Matasi, Julius, Lavey, Brian, McElroy, William T, Tulshian, Deen, Tata, James, Sondey, Christopher, Garlisi, Charles G, Devito, Kristine, Fossetta, James, Lundell, Daniel, Niu, Xiaoda
Published in ACS medicinal chemistry letters (13.08.2015)
Published in ACS medicinal chemistry letters (13.08.2015)
Get full text
Journal Article
Live Cell Membranome cDNA Screen: A Novel Homogenous Live Cell Binding Assay to Study Membrane Protein-Ligand Interaction
Shen, Xun, Smith, Elizabeth, Ai, Xi, McElroy, William T., Liaw, Andy, Kreamer, Tony, Chang, Meiping, Devito, Kristine, Hudak, Edward, Xu, Serena, Pei, Yi, Sur, Sylvie, Peier, Andrea, Li, Jing
Published in SLAS discovery (01.12.2019)
Published in SLAS discovery (01.12.2019)
Get full text
Journal Article
Application of Palladium-Catalyzed Allylic Arylation to the Synthesis of a (±)-7-Deoxypancratistatin Analogue
Shukla, Krupa H, Boehmler, Debra J, Bogacyzk, Suzanne, Duvall, Bridget R, Peterson, William A, McElroy, William T, DeShong, Philip
Published in Organic letters (14.09.2006)
Published in Organic letters (14.09.2006)
Get full text
Journal Article
Pyrazoloquinolines as PDE10A inhibitors: Discovery of a tool compound
McElroy, William T., Tan, Zheng, Basu, Kallol, Yang, Shu-Wei, Smotryski, Jennifer, Ho, Ginny D., Tulshian, Deen, Greenlee, William J., Mullins, Deborra, Guzzi, Mario, Zhang, Xiaoping, Bleickardt, Carina, Hodgson, Robert
Published in Bioorganic & medicinal chemistry letters (01.02.2012)
Published in Bioorganic & medicinal chemistry letters (01.02.2012)
Get full text
Journal Article