Granulosa cell endothelin-2 expression is fundamental for ovulatory follicle rupture
Cacioppo, Joseph A, Lin, Po-Ching Patrick, Hannon, Patrick R, McDougle, Daniel R, Gal, Arnon, Ko, CheMyong
Published in Scientific reports (11.04.2017)
Published in Scientific reports (11.04.2017)
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Functional studies of N‐terminally modified CYP2J2 epoxygenase in model lipid bilayers
McDougle, Daniel R., Palaria, Amrita, Magnetta, Eric, Meling, Daryl D., Das, Aditi
Published in Protein science (01.07.2013)
Published in Protein science (01.07.2013)
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Anti-inflammatory ω-3 endocannabinoid epoxides
McDougle, Daniel R., Watson, Josephine E., Abdeen, Amr A., Adili, Reheman, Caputo, Megan P., Krapf, John E., Johnson, Rodney W., Kilian, Kristopher A., Holinstat, Michael, Das, Aditi
Published in Proceedings of the National Academy of Sciences - PNAS (25.07.2017)
Published in Proceedings of the National Academy of Sciences - PNAS (25.07.2017)
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Incorporation of charged residues in the CYP2J2 F-G loop disrupts CYP2J2–lipid bilayer interactions
McDougle, Daniel R., Baylon, Javier L., Meling, Daryl D., Kambalyal, Amogh, Grinkova, Yelena V., Hammernik, Jared, Tajkhorshid, Emad, Das, Aditi
Published in Biochimica et biophysica acta (01.10.2015)
Published in Biochimica et biophysica acta (01.10.2015)
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Preclinical evaluation of intravenous NAX 810‐2, a novel GalR2‐preferring analog, for anticonvulsant efficacy and pharmacokinetics
Metcalf, Cameron S., Klein, Brian D., McDougle, Daniel R., Zhang, Liuyin, Kaufmann, Dan, Bulaj, Grzegorz, White, H. Steve
Published in Epilepsia (Copenhagen) (01.02.2017)
Published in Epilepsia (Copenhagen) (01.02.2017)
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CYP2J2 epoxygenase membrane anchor plays an important role in facilitating electron transfer from CPR
Meling, Daryl D., McDougle, Daniel R., Das, Aditi
Published in Journal of inorganic biochemistry (01.01.2015)
Published in Journal of inorganic biochemistry (01.01.2015)
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Preclinical Analgesic and Safety Evaluation of the GalR2-preferring Analog, NAX 810-2
Metcalf, Cameron S., Smith, Misty D., Klein, Brian D., McDougle, Daniel R., Zhang, Liuyin, Bulaj, Grzegorz
Published in Neurochemical research (01.07.2017)
Published in Neurochemical research (01.07.2017)
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Analgesic properties of a peripherally acting and GalR2 receptor-preferring galanin analog in inflammatory, neuropathic, and acute pain models
Metcalf, Cameron S, Klein, Brian D, McDougle, Daniel R, Zhang, Liuyin, Smith, Misty D, Bulaj, Grzegorz, White, H Steve
Published in The Journal of pharmacology and experimental therapeutics (01.01.2015)
Published in The Journal of pharmacology and experimental therapeutics (01.01.2015)
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Journal Article
Cyclooxygenase-2 catalysis and inhibition in lipid bilayer nanodiscs
Orlando, Benjamin J., McDougle, Daniel R., Lucido, Michael J., Eng, Edward T., Graham, Leigh Ann, Schneider, Claus, Stokes, David L., Das, Aditi, Malkowski, Michael G.
Published in Archives of biochemistry and biophysics (15.03.2014)
Published in Archives of biochemistry and biophysics (15.03.2014)
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Incorporation of Monodisperse Oligoethyleneglycol Amino Acids into Anticonvulsant Analogues of Galanin and Neuropeptide Y Provides Peripherally Acting Analgesics
Zhang, Liuyin, Klein, Brian D, Metcalf, Cameron S, Smith, Misty D, McDougle, Daniel R, Lee, Hee-Kyoung, White, H. Steve, Bulaj, Grzegorz
Published in Molecular pharmaceutics (04.02.2013)
Published in Molecular pharmaceutics (04.02.2013)
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Introduction of lipidization-cationization motifs affords systemically bioavailable neuropeptide Y and neurotensin analogs with anticonvulsant activities
Green, Brad R., White, Karen L., McDougle, Daniel R., Zhang, Liuyin, Klein, Brian, Scholl, Erika A., Pruess, Timothy H., White, H. Steve, Bulaj, Grzegorz
Published in Journal of peptide science (01.09.2010)
Published in Journal of peptide science (01.09.2010)
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Journal Article
Pre-Clinical Evaluation of Intravenous NAX 810-2, a Novel GalR2-Preferring Analog, for Anticonvulsant Efficacy and Pharmacokinetics
Metcalf, Cameron S., Klein, Brian D., McDougle, Daniel R., Zhang, Liuyin, Kaufmann, Dan, Bulaj, Grzegorz, White, H. Steve
Published in Epilepsia (Copenhagen) (18.01.2017)
Published in Epilepsia (Copenhagen) (18.01.2017)
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