A Small-Molecule Inhibitor of PIM Kinases as a Potential Treatment for Urothelial Carcinomas
Foulks, Jason M, Carpenter, Kent J, Luo, Bai, Xu, Yong, Senina, Anna, Nix, Rebecca, Chan, Ashley, Clifford, Adrianne, Wilkes, Marcus, Vollmer, David, Brenning, Benjamin, Merx, Shannon, Lai, Shuping, McCullar, Michael V, Ho, Koc-Kan, Albertson, Daniel J, Call, Lee T, Bearss, Jared J, Tripp, Sheryl, Liu, Ting, Stephens, Bret J, Mollard, Alexis, Warner, Steven L, Bearss, David J, Kanner, Steven B
Published in Neoplasia (New York, N.Y.) (01.05.2014)
Published in Neoplasia (New York, N.Y.) (01.05.2014)
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Discovery of 4-phenyl-2-phenylaminopyridine based TNIK inhibitors
Ho, Koc-Kan, Parnell, K. Mark, Yuan, Yi, Xu, Yong, Kultgen, Steven G, Hamblin, Steven, Hendrickson, Thomas F, Luo, Bai, Foulks, Jason M, McCullar, Michael V, Kanner, Steven B
Published in Bioorganic & medicinal chemistry letters (15.01.2013)
Published in Bioorganic & medicinal chemistry letters (15.01.2013)
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Synthesis and structure–activity relationship of 2-arylamino-4-aryl-pyrimidines as potent PAK1 inhibitors
Xu, Yong, Foulks, Jason M., Clifford, Adrianne, Brenning, Benjamin, Lai, Shuping, Luo, Bai, Parnell, K. Mark, Merx, Shannon, McCullar, Michael V., Kanner, Steven B., Ho, Koc-Kan
Published in Bioorganic & medicinal chemistry letters (15.07.2013)
Published in Bioorganic & medicinal chemistry letters (15.07.2013)
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Intraperitoneal delivery of human natural killer cells for treatment of ovarian cancer
Knorr, D, Pribyl, L, Bendzick, L, McCullar, V, Miller, J, Kaufman, D
Published in Gynecologic oncology (01.07.2013)
Published in Gynecologic oncology (01.07.2013)
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Epigenetic drug discovery: targeting DNA methyltransferases
Foulks, Jason M, Parnell, K Mark, Nix, Rebecca N, Chau, Suzanna, Swierczek, Krzysztof, Saunders, Michael, Wright, Kevin, Hendrickson, Thomas F, Ho, Koc-Kan, McCullar, Michael V, Kanner, Steven B
Published in Journal of biomolecular screening (01.01.2012)
Published in Journal of biomolecular screening (01.01.2012)
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Pharmacologic activation of PKM2 slows lung tumor xenograft growth
Parnell, K Mark, Foulks, Jason M, Nix, Rebecca N, Clifford, Adrianne, Bullough, Jeremy, Luo, Bai, Senina, Anna, Vollmer, David, Liu, Jihua, McCarthy, Virgil, Xu, Yong, Saunders, Michael, Liu, Xiao-Hui, Pearce, Scott, Wright, Kevin, O'Reilly, Marc, McCullar, Michael V, Ho, Koc-Kan, Kanner, Steven B
Published in Molecular cancer therapeutics (01.08.2013)
Published in Molecular cancer therapeutics (01.08.2013)
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Discovery of 3-(trifluoromethyl)-1H-pyrazole-5-carboxamide activators of the M2 isoform of pyruvate kinase (PKM2)
Xu, Yong, Liu, Xiao-Hui, Saunders, Michael, Pearce, Scott, Foulks, Jason M., Parnell, K. Mark, Clifford, Adrianne, Nix, Rebecca N., Bullough, Jeremy, Hendrickson, Thomas F., Wright, Kevin, McCullar, Michael V., Kanner, Steven B., Ho, Koc-Kan
Published in Bioorganic & medicinal chemistry letters (15.01.2014)
Published in Bioorganic & medicinal chemistry letters (15.01.2014)
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Synthesis and Biological Evaluation of Pyrazolo[1,5‑a]pyrimidine Compounds as Potent and Selective Pim‑1 Inhibitors
Xu, Yong, Brenning, Benjamin G, Kultgen, Steven G, Foulks, Jason M, Clifford, Adrianne, Lai, Shuping, Chan, Ashley, Merx, Shannon, McCullar, Michael V, Kanner, Steven B, Ho, Koc-Kan
Published in ACS medicinal chemistry letters (08.01.2015)
Published in ACS medicinal chemistry letters (08.01.2015)
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GSK3 Inhibition Drives Maturation of NK Cells and Enhances Their Antitumor Activity
Cichocki, Frank, Valamehr, Bahram, Bjordahl, Ryan, Zhang, Bin, Rezner, Betsy, Rogers, Paul, Gaidarova, Svetlana, Moreno, Stacey, Tuininga, Katie, Dougherty, Phillip, McCullar, Valarie, Howard, Peter, Sarhan, Dhifaf, Taras, Emily, Schlums, Heinrich, Abbot, Stewart, Shoemaker, Daniel, Bryceson, Yenan T, Blazar, Bruce R, Wolchko, Scott, Cooley, Sarah, Miller, Jeffrey S
Published in Cancer research (Chicago, Ill.) (15.10.2017)
Published in Cancer research (Chicago, Ill.) (15.10.2017)
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Discovery of Novel Putative Inhibitors of UDP-GlcNAc 2‑Epimerase as Potent Antibacterial Agents
Xu, Yong, Brenning, Benjamin, Clifford, Adrianne, Vollmer, David, Bearss, Jared, Jones, Carissa, McCarthy, Virgil, Shi, Chongtie, Wolfe, Bradley, Aavula, Bhasker, Warner, Steve, Bearss, David J, McCullar, Michael V, Schuch, Raymond, Pelzek, Adam, Bhaskaran, Shyam S, Stebbins, C. Erec, Goldberg, Allan R, Fischetti, Vincent A, Vankayalapati, Hariprasad
Published in ACS medicinal chemistry letters (12.12.2013)
Published in ACS medicinal chemistry letters (12.12.2013)
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Tim-3 Is an Inducible Human Natural Killer (NK) Cell Receptor That Enhances Interferon Gamma Production in Response to Galectin-9 (GAL-9)
Gleason, M.K, Lenvik, T.R, McCullar, V, Felices, M, O'Brien, M.S, Cooley, S.A, Verneris, M.R, Cichocki, F, Holman, C.J, Panoskaltsis-Mortari, A, Niki, T, Hirashima, M, Blazar, B.R, Miller, J.S
Published in Biology of blood and marrow transplantation (2012)
Published in Biology of blood and marrow transplantation (2012)
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43: A subpopulation of human NK cells lacking inhibitory receptors for self MHC is developmentally immature rather than autoreactive
Cooley, S.A, Xiao, F, Bergemann, T.L, Pitt, M, Gleason, M, McCullar, V, McQueen, K, Guethlein, L, Parham, P, Miller, J.S
Published in Biology of blood and marrow transplantation (2007)
Published in Biology of blood and marrow transplantation (2007)
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Abstract 3226: PKM2 metabolic activator slows lung cancer xenograft growth
Parnell, Mark, Foulks, Jason M., Nix, Rebecca, Luo, Bai, Senina, Anna, Xu, Yong, Saunders, Michael, Ho, Koc-Kan, McCullar, Michael V., Kanner, Steven B.
Published in Cancer research (Chicago, Ill.) (15.04.2012)
Published in Cancer research (Chicago, Ill.) (15.04.2012)
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