Conformational pathway provides unique sensitivity to a synaptic mGluR
Habrian, Chris H., Levitz, Joshua, Vyklicky, Vojtech, Fu, Zhu, Hoagland, Adam, McCort-Tranchepain, Isabelle, Acher, Francine, Isacoff, Ehud Y.
Published in Nature communications (05.12.2019)
Published in Nature communications (05.12.2019)
Get full text
Journal Article
The mGlu7 receptor provides protective effects against epileptogenesis and epileptic seizures
Girard, Benoit, Tuduri, Pola, Moreno, Maria Paula, Sakkaki, Sophie, Barboux, Cedric, Bouschet, Tristan, Varrault, Annie, Vitre, Jihane, McCort-Tranchepain, Isabelle, Dairou, Julien, Acher, Francine, Fagni, Laurent, Marchi, Nicola, Perroy, Julie, Bertaso, Federica
Published in Neurobiology of disease (01.09.2019)
Published in Neurobiology of disease (01.09.2019)
Get full text
Journal Article
Natural amines inhibit activation of human plasmacytoid dendritic cells through CXCR4 engagement
Smith, Nikaïa, Pietrancosta, Nicolas, Davidson, Sophia, Dutrieux, Jacques, Chauveau, Lise, Cutolo, Pasquale, Dy, Michel, Scott-Algara, Daniel, Manoury, Bénédicte, Zirafi, Onofrio, McCort-Tranchepain, Isabelle, Durroux, Thierry, Bachelerie, Françoise, Schwartz, Olivier, Münch, Jan, Wack, Andreas, Nisole, Sébastien, Herbeuval, Jean-Philippe
Published in Nature communications (09.02.2017)
Published in Nature communications (09.02.2017)
Get full text
Journal Article
LSP2-9166, an orthosteric mGlu4 and mGlu7 receptor agonist, reduces cocaine self-administration under a progressive ratio schedule in rats
De Sa Nogueira, David, Bourdy, Romain, Filliol, Dominique, Quessada, Cyril, McCort-Tranchepain, Isabelle, Acher, Francine, Zwiller, Jean, Romieu, Pascal, Befort, Katia
Published in Neuroscience letters (01.11.2021)
Published in Neuroscience letters (01.11.2021)
Get full text
Journal Article
Activation of the Mu-Delta Opioid Receptor Heteromers Blocks Morphine Rewarding Effects
Requana Aradas, Ariadna, Djaboub, Youssra, Mccort-Tranchepain, Isabelle, Hajasova, Zuzana, Clémenceau, Loïc, Canestrelli, Corinne, Mann, Anika, Schulz, Stefan, Delaval, Angélique, Acher, Francine, Massotte, Dominique, Noble, Florence, Marie, Nicolas
Published in The international journal of neuropsychopharmacology (01.07.2023)
Published in The international journal of neuropsychopharmacology (01.07.2023)
Get full text
Journal Article
MFSD1 with its accessory subunit GLMP functions as a general dipeptide uniporter in lysosomes
Jungnickel, Katharina Esther Julia, Guelle, Océane, Iguchi, Miharu, Dong, Wentao, Kotov, Vadim, Gabriel, Florian, Debacker, Cécile, Dairou, Julien, McCort-Tranchepain, Isabelle, Laqtom, Nouf N., Chan, Sze Ham, Ejima, Akika, Sato, Kenji, Massa López, David, Saftig, Paul, Mehdipour, Ahmad Reza, Abu-Remaileh, Monther, Gasnier, Bruno, Löw, Christian, Damme, Markus
Published in Nature cell biology (01.07.2024)
Published in Nature cell biology (01.07.2024)
Get full text
Journal Article
Novel Inhibitory Site Revealed by XAP044 Mode of Action on the Metabotropic Glutamate 7 Receptor Venus Flytrap Domain
Cristiano, Nunzia, Cabayé, Alexandre, Brabet, Isabelle, Glatthar, Ralf, Tora, Amelie, Goudet, Cyril, Bertrand, Hugues-Olivier, Goupil-Lamy, Anne, Flor, Peter J., Pin, Jean-Philippe, McCort-Tranchepain, Isabelle, Acher, Francine C.
Published in Journal of medicinal chemistry (25.07.2024)
Published in Journal of medicinal chemistry (25.07.2024)
Get full text
Journal Article
Activation of the Mu-Delta Opioid Receptor Heteromers Blocks Morphine Rewarding Effects
Requana Aradas, Ariadna, Djaboub, Youssra, McCort-Tranchepain, Isabelle, Hajasova, Zuzana, Clémenceau, Loïc, Canestrelli, Corinne, Mann, Anika, Schulz, Stefan, Delaval, Angélique, Acher, Francine, Massotte, Dominique, Noble, Florence, Marie, Nicolas
Published in The international journal of neuropsychopharmacology (31.07.2023)
Published in The international journal of neuropsychopharmacology (31.07.2023)
Get full text
Journal Article
Amino Acids Bearing Aromatic or Heteroaromatic Substituents as a New Class of Ligands for the Lysosomal Sialic Acid Transporter Sialin
Dubois, Lilian, Pietrancosta, Nicolas, Cabaye, Alexandre, Fanget, Isabelle, Debacker, Cécile, Gilormini, Pierre-André, Dansette, Patrick M, Dairou, Julien, Biot, Christophe, Froissart, Roseline, Goupil-Lamy, Anne, Bertrand, Hugues-Olivier, Acher, Francine C, McCort-Tranchepain, Isabelle, Gasnier, Bruno, Anne, Christine
Published in Journal of medicinal chemistry (13.08.2020)
Published in Journal of medicinal chemistry (13.08.2020)
Get full text
Journal Article
Increased Potency and Selectivity for Group III Metabotropic Glutamate Receptor Agonists Binding at Dual sites
Selvam, Chelliah, Lemasson, Isabelle A, Brabet, Isabelle, Oueslati, Nadia, Karaman, Berin, Cabaye, Alexandre, Tora, Amélie S, Commare, Bruno, Courtiol, Tiphanie, Cesarini, Sara, McCort-Tranchepain, Isabelle, Rigault, Delphine, Mony, Laetitia, Bessiron, Thomas, McLean, Heather, Leroux, Frédéric R, Colobert, Françoise, Daniel, Hervé, Goupil-Lamy, Anne, Bertrand, Hugues-Olivier, Goudet, Cyril, Pin, Jean-Philippe, Acher, Francine C
Published in Journal of medicinal chemistry (08.03.2018)
Published in Journal of medicinal chemistry (08.03.2018)
Get full text
Journal Article
Synthesis and Biological Properties of New Constrained CCK-B Antagonists: Discrimination of Two Affinity States of the CCK-B Receptor on Transfected CHO Cells
Bellier, Bruno, McCort-Tranchepain, Isabelle, Ducos, Bertrand, Danascimento, Sophie, Meudal, Hervé, Noble, Florence, Garbay, Christiane, Roques, Bernard P
Published in Journal of medicinal chemistry (21.11.1997)
Published in Journal of medicinal chemistry (21.11.1997)
Get full text
Journal Article
MFSD1 in complex with its accessory subunit GLMP functions as a general dipeptide uniporter in lysosomes
Katharina Esther Julia Jungnickel, Guelle, Oceane, Iguchi, Miharu, Dong, Wentao, Kotov, Vadim, Gabriel, Florian, Debacker, Cecile, Dairou, Julien, Mccort-Tranchepain, Isabelle, Laqtom, Nouf N, Sze Ham Chan, Ejima, Akika, Sato, Kenji, David Massa Lopez, Saftig, Paul, Mehdipour, Ahmad Reza, Abu-Remaileh, Monther, Gasnier, Bruno, Low, Christian, Damme, Markus
Published in bioRxiv (15.12.2023)
Published in bioRxiv (15.12.2023)
Get full text
Paper