Kinetically Selective Inhibitors of Histone Deacetylase 2 (HDAC2) as Cognition Enhancers
Wagner, F F, Zhang, Y-L, Fass, D M, Joseph, N, Gale, J P, Weïwer, M, McCarren, P, Fisher, S L, Kaya, T, Zhao, W-N, Reis, S A, Hennig, K M, Thomas, M, Lemercier, B C, Lewis, M C, Guan, J S, Moyer, M P, Scolnick, E, Haggarty, S J, Tsai, L-H, Holson, E B
Published in Chemical science (Cambridge) (01.01.2015)
Published in Chemical science (Cambridge) (01.01.2015)
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Conformational Studies of Methyl 3-O-Methyl-α-d-arabinofuranoside: An Approach for Studying the Conformation of Furanose Rings
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McKinney, D., Ranaghan, M., McMillan, B., Brousseau, M., O’Keefe, M., Moroco, J., Singh, R., Besnik, B., McCarren, P., Mulvaney, K., Sellers, W., Ianari, A.
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An Isochemogenic Set of Inhibitors To Define the Therapeutic Potential of Histone Deacetylases in β‑Cell Protection
Wagner, Florence F, Lundh, Morten, Kaya, Taner, McCarren, Patrick, Zhang, Yan-Ling, Chattopadhyay, Shrikanta, Gale, Jennifer P, Galbo, Thomas, Fisher, Stewart L, Meier, Bennett C, Vetere, Amedeo, Richardson, Sarah, Morgan, Noel G, Christensen, Dan Ploug, Gilbert, Tamara J, Hooker, Jacob M, Leroy, Mélanie, Walpita, Deepika, Mandrup-Poulsen, Thomas, Wagner, Bridget K, Holson, Edward B
Published in ACS chemical biology (19.02.2016)
Published in ACS chemical biology (19.02.2016)
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Kinetically selective inhibitors of histone deacetylase 2 (HDAC2) as cognition enhancersElectronic supplementary information (ESI) available: Compound synthesis and characterization; 1HNMR spectra, HPLC or UPLC spectral traces; HDAC enzymatic assay protocol; IC50s for representative compounds for HDACs 1-9; full kinetic parameters for BRD4884 and BRD6688; progression and dissociation curves for BRD6688; pharmacokinetic graphs and parameters for representative compounds; kinetic selectivity profi
Wagner, F. F, Zhang, Y.-L, Fass, D. M, Joseph, N, Gale, J. P, Weïwer, M, McCarren, P, Fisher, S. L, Kaya, T, Zhao, W.-N, Reis, S. A, Hennig, K. M, Thomas, M, Lemercier, B. C, Lewis, M. C, Guan, J. S, Moyer, M. P, Scolnick, E, Haggarty, S. J, Tsai, L.-H, Holson, E. B
Year of Publication 01.12.2014
Year of Publication 01.12.2014
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Kinetically selective inhibitors of histone deacetylase 2 (HDAC2) as cognition enhancers† †Electronic supplementary information (ESI) available: Compound synthesis and characterization; 1HNMR spectra, HPLC or UPLC spectral traces; HDAC enzymatic assay protocol; IC50s for representative compounds for HDACs 1–9; full kinetic parameters for BRD4884 and BRD6688; progression and dissociation curves for BRD6688; pharmacokinetic graphs and parameters for representative compounds; kinetic selectivity pr
Wagner, F. F., Zhang, Y.-L., Fass, D. M., Joseph, N., Gale, J. P., Weïwer, M., McCarren, P., Fisher, S. L., Kaya, T., Zhao, W.-N., Reis, S. A., Hennig, K. M., Thomas, M., Lemercier, B. C., Lewis, M. C., Guan, J. S., Moyer, M. P., Scolnick, E., Haggarty, S. J., Tsai, L.-H., Holson, E. B.
Published in Chemical science (Cambridge) (09.10.2014)
Published in Chemical science (Cambridge) (09.10.2014)
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Nitroxyl Disulfides, Novel Intermediates in Transnitrosation Reactions
Houk, K. N, Hietbrink, Bruce N, Bartberger, Michael D, McCarren, Patrick R, Choi, Bo Yoon, Voyksner, Robert D, Stamler, Jonathan S, Toone, Eric J
Published in Journal of the American Chemical Society (11.06.2003)
Published in Journal of the American Chemical Society (11.06.2003)
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Pulmonary penetration of alpha 1-proteinase inhibitor administered parenterally to dogs
Smith, R M, Spragg, R G, Moser, K M, Cochrane, C G, McCarren, J P
Published in The American review of respiratory disease (01.12.1987)
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Arabinofuranosyl Oligosaccharides from Mycobacteria: Synthesis and Effect of Glycosylation on Ring Conformation and Hydroxymethyl Group Rotamer Populations
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Published in Journal of the American Chemical Society (23.02.2000)
Published in Journal of the American Chemical Society (23.02.2000)
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Computational Studies of the Arabinofuranose Ring: Conformational Preferences of Fully Relaxed Methyl α-d-arabinofuranoside
McCarren, Patrick R, Gordon, Matthew T, Lowary, Todd L, Hadad, Christopher M
Published in The journal of physical chemistry. A, Molecules, spectroscopy, kinetics, environment, & general theory (21.06.2001)
Published in The journal of physical chemistry. A, Molecules, spectroscopy, kinetics, environment, & general theory (21.06.2001)
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