Design and synthesis of potent and selective 1,3,4-trisubstituted-2-oxopiperazine based melanocortin-4 receptor agonists
Tian, Xinrong, Mishra, Rajesh K., Switzer, Adrian G., Hu, X. Eric, Kim, Nick, Mazur, Adam W., Ebetino, Frank H., Wos, John A., Crossdoersen, Doreen, Pinney, Beth B., Farmer, Julie A., Sheldon, Russell J.
Published in Bioorganic & medicinal chemistry letters (01.09.2006)
Published in Bioorganic & medicinal chemistry letters (01.09.2006)
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Journal Article
Design, Synthesis, and Evaluation of Proline and Pyrrolidine Based Melanocortin Receptor Agonists. A Conformationally Restricted Dipeptide Mimic Approach
Tian, Xinrong, Field, Timothy B, Switzer, Adrian G, Mazur, Adam W, Ebetino, Frank H, Wos, John A, Berberich, Steve M, Jayasinghe, Lalith R, Obringer, Cindy M, Dowty, Martin E, Pinney, Beth B, Farmer, Julie A, Crossdoersen, Doreen, Sheldon, Russell J
Published in Journal of medicinal chemistry (27.07.2006)
Published in Journal of medicinal chemistry (27.07.2006)
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Journal Article
Design, synthesis, and evaluation of proline based melanocortin receptor ligands
Tian, Xinrong, Field, Timothy, Mazur, Adam W., Ebetino, Frank H., Wos, John A., Crossdoersen, Doreen, Pinney, Beth B., Sheldon, Russell J.
Published in Bioorganic & medicinal chemistry letters (02.06.2005)
Published in Bioorganic & medicinal chemistry letters (02.06.2005)
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Journal Article
Sauvagine analogs selective for corticotropin releasing factor 2 receptor: effect of substitutions at positions 35 and 39 on CRF2R selectivity
Mazur, Adam W., Wang, Feng, Tscheiner, Michelle, Donnelly, Elizabeth, Isfort, Robert J.
Published in Peptides (New York, N.Y. : 1980) (01.05.2005)
Published in Peptides (New York, N.Y. : 1980) (01.05.2005)
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Journal Article
Discovery of Corticotropin Releasing Factor 2 Receptor Selective Sauvagine Analogues for Treatment of Skeletal Muscle Atrophy
Isfort, Robert J, Wang, Feng, Tscheiner, Michelle, Donnelly, Elizabeth, Bauer, Mary Beth, Lefever, Frank, Hinkle, Richard T, Mazur, Adam W
Published in Journal of medicinal chemistry (13.01.2005)
Published in Journal of medicinal chemistry (13.01.2005)
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Journal Article
Modifications of the human urocortin 2 peptide that improve pharmacological properties
Isfort, Robert J., Wang, Feng, Tscheiner, Michelle, Dolan, Elizabeth, Bauer, Mary Beth, Lefever, Frank, Reichart, Deborah, Wehmeyer, Kenneth R., Reilman, Raymond A., Keck, Bradly D., Hinkle, Richard T., Mazur, Adam W.
Published in Peptides (New York, N.Y. : 1980) (01.07.2006)
Published in Peptides (New York, N.Y. : 1980) (01.07.2006)
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Journal Article
Novel tetrahydropyran-based peptidomimetics from a bioisosteric transformation of a tripeptide. Evidence of their activity at melanocortin receptors
Mazur, Adam W, Kulesza, Anna, Mishra, Rajesh K, Cross-Doersen, Doreen, Russell, Anne F, Ebetino, Frank H
Published in Bioorganic & medicinal chemistry (17.07.2003)
Published in Bioorganic & medicinal chemistry (17.07.2003)
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Journal Article
Discovery of Substituted Human Urocortin 1 Analogs with Improved CRF2 Receptor Selectivity and Increased Efficacy in Preventing Skeletal Muscle Atrophy
Isfort, Robert J, Wang, Feng, Tscheiner, Michelle, Dolan, Elizabeth, Bauer, Mary Beth, Lefever, Frank, Reichart, Deborah, Hinkle, Richard T, Wehmeyer, Kenneth R, Reilman, Raymond A, Keck, Bradly D, Mazur, Adam W
Published in International journal of peptide research and therapeutics (01.09.2007)
Published in International journal of peptide research and therapeutics (01.09.2007)
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Journal Article
Digestibility of selected carbohydrates by anaerobic bacteria
Mazur, Adam W, Mohlenkamp, M. Joseph, Hiler, George, Wilkins, Tracy D, Van Tassell, Roger L
Published in Journal of agricultural and food chemistry (01.11.1993)
Published in Journal of agricultural and food chemistry (01.11.1993)
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Preparation of ‘carba’ dipeptides bearing a basic side-chain at the C-terminus: synthesis of enantiopure Boc- d-Phe-Ψ[CH 2CH 2]- l-Arg(NO 2)-OH and Boc- d-Phe-Ψ[CH 2CH 2]- d-Arg(NO 2)-OH
Kende, Andrew S., Dong, Han-Qing, Mazur, Adam W., Ebetino, Frank H.
Published in Tetrahedron letters (27.08.2001)
Published in Tetrahedron letters (27.08.2001)
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