2,6-Naphthyridines as potent and selective inhibitors of the novel protein kinase C isozymes
van Eis, Maurice J., Evenou, Jean-Pierre, Floersheim, Philipp, Gaul, Christoph, Cowan-Jacob, Sandra W., Monovich, Lauren, Rummel, Gabriele, Schuler, Walter, Stark, Wilhelm, Strauss, Andre, Matt, Anette von, Vangrevelinghe, Eric, Wagner, Juergen, Soldermann, Nicolas
Published in Bioorganic & medicinal chemistry letters (15.12.2011)
Published in Bioorganic & medicinal chemistry letters (15.12.2011)
Get full text
Journal Article
Aromatic Quinolinecarboxamides as Selective, Orally Active Antibody Production Inhibitors for Prevention of Acute Xenograft Rejection
Papageorgiou, Christos, von Matt, Anette, Joergensen, Joanne, Andersen, Elsebeth, Wagner, Katrin, Beerli, Christian, Than, Thai, Borer, Xaver, Florineth, Andrea, Rihs, Gretty, Schreier, Max H, Weckbecker, Gisbert, Heusser, Christoph
Published in Journal of medicinal chemistry (07.06.2001)
Published in Journal of medicinal chemistry (07.06.2001)
Get full text
Journal Article
Discovery of novel pyrrolidineoxy-substituted heteroaromatics as potent and selective PI3K delta inhibitors with improved physicochemical properties
Hoegenauer, Klemens, Soldermann, Nicolas, Hebach, Christina, Hollingworth, Gregory J., Lewis, Ian, von Matt, Anette, Smith, Alexander B., Wolf, Romain M., Wilcken, Rainer, Haasen, Dorothea, Burkhart, Christoph, Zécri, Frédéric
Published in Bioorganic & medicinal chemistry letters (01.12.2016)
Published in Bioorganic & medicinal chemistry letters (01.12.2016)
Get full text
Journal Article
Identification of Orally Available Naphthyridine Protein Kinase D Inhibitors
Meredith, Erik L, Ardayfio, Ophelia, Beattie, Kimberly, Dobler, Markus R, Enyedy, Istvan, Gaul, Christoph, Hosagrahara, Vinayak, Jewell, Charles, Koch, Keith, Lee, Wendy, Lehmann, HansJoerg, McKinsey, Timothy A, Miranda, Karl, Pagratis, Nikos, Pancost, Margaret, Patnaik, Anup, Phan, Dillon, Plato, Craig, Qian, Ming, Rajaraman, Vasumathy, Rao, Chang, Rozhitskaya, Olga, Ruppen, Thomas, Shi, Jie, Siska, Sarah J, Springer, Clayton, van Eis, Maurice, Vega, Richard B, von Matt, Anette, Yang, Lihua, Yoon, Taeyoung, Zhang, Ji-Hu, Zhu, Na, Monovich, Lauren G
Published in Journal of medicinal chemistry (12.08.2010)
Published in Journal of medicinal chemistry (12.08.2010)
Get full text
Journal Article
New pyrazolo[1,5a]pyrimidines as orally active inhibitors of Lck
Gommermann, Nina, Buehlmayer, Peter, von Matt, Anette, Breitenstein, Werner, Masuya, Keiichi, Pirard, Bernard, Furet, Pascal, Cowan-Jacob, Sandra W., Weckbecker, Gisbert
Published in Bioorganic & medicinal chemistry letters (15.06.2010)
Published in Bioorganic & medicinal chemistry letters (15.06.2010)
Get full text
Journal Article
NLRP3 inflammasome inhibitors
SMITH, Nichola, FOOKS SOLOVAY, Catherine, VELCICKY, Juraj, FARADY, Christopher, MATTES, Henri, GOMMERMANN, Nina, STIEFL, Nikolaus Johannes, VON MATT, Anette, VANGREVELINGHE, Eric, MACKAY, Angela, JANSER, Philipp
Year of Publication 02.03.2023
Get full text
Year of Publication 02.03.2023
Patent
NLRP3 INFLAMMASOME INHIBITORS
SMITH, Nichola, VELCICKY, Juraj, FARADY, Christopher, MATTES, Henri, GOMMERMANN, Nina, STIEFL, Nikolaus Johannes, SOLOVAY, Catherine Fooks, VANGREVELINGHE, Eric, MACKAY, Angela, von MATT, Anette, JANSER, Philipp
Year of Publication 11.08.2022
Get full text
Year of Publication 11.08.2022
Patent
NLRP3 INFLAMMASOME INHIBITORS
SMITH, Nichola, FOOKS SOLOVAY, Catherine, VELCICKY, Juraj, FARADY, Christopher, MATTES, Henri, GOMMERMANN, Nina, STIEFL, Nikolaus Johannes, VON MATT, Anette, VANGREVELINGHE, Eric, MACKAY, Angela, JANSER, Philipp
Year of Publication 23.03.2022
Get full text
Year of Publication 23.03.2022
Patent
NLRP3 inflammasome inhibitors
Gommermann, Nina, Mattes, Henri, Mackay, Angela, Solovay, Catherine Fooks, Velcicky, Juraj, Farady, Christopher, Stiefl, Nikolaus Johannes, von Matt, Anette, Janser, Philipp, Smith, Nichola, Vangrevelinghe, Eric
Year of Publication 22.02.2022
Get full text
Year of Publication 22.02.2022
Patent
NLRP3 INFLAMMASOME INHIBITORS
SMITH, Nichola, FOOKS SOLOVAY, Catherine, VELCICKY, Juraj, FARADY, Christopher, MATTES, Henri, GOMMERMANN, Nina, STIEFL, Nikolaus Johannes, VON MATT, Anette, VANGREVELINGHE, Eric, MACKAY, Angela, JANSER, Philipp
Year of Publication 30.12.2021
Get full text
Year of Publication 30.12.2021
Patent
NLRP3 inflammasome inhibitors
Gommermann, Nina, Mattes, Henri, Mackay, Angela, Solovay, Catherine Fooks, Velcicky, Juraj, Farady, Christopher, Stiefl, Nikolaus Johannes, von Matt, Anette, Janser, Philipp, Smith, Nichola, Vangrevelinghe, Eric
Year of Publication 28.12.2021
Get full text
Year of Publication 28.12.2021
Patent
NLRP3 inflammasome inhibitors
SMITH, Nichola, FOOKS SOLOVAY, Catherine, VELCICKY, Juraj, FARADY, Christopher, MATTES, Henri, GOMMERMANN, Nina, STIEFL, Nikolaus Johannes, VON MATT, Anette, VANGREVELINGHE, Eric, MACKAY, Angela, JANSER, Philipp
Year of Publication 18.11.2021
Get full text
Year of Publication 18.11.2021
Patent
Tetrahydro-Pyrido-Pyrimidine Derivatives
Hoegenauer, Klemens, Tufilli, Nicola, Hollingworth, Gregory John, Graveleau, Nadege, Smith, Alexander Baxter, von Matt, Anette, Wolf, Romain, Hebach, Christina, Soldermann, Nicolas, Strang, Ross Sinclair, Zecri, Frederic, Fernandes Gomes Dos Santos, Paulo, Cooke, Nigel Graham, Stowasser, Frank
Year of Publication 25.08.2022
Get full text
Year of Publication 25.08.2022
Patent
NLRP3 INFLAMMASOME INHIBITORS
MACKAY, ANGELA, STIEFL, NIKOLAUS JOHANNES, GOMMERMANN, NINA, FARADY, CHRISTOPHER, JANSER, PHILIPP, FOOKS SOLOVAY, CATHERINE, MATTES, HENRI, VANGREVELINGHE, ERIC, SMITH, NICHOLA, VON MATT, ANETTE, VELCICKY, JURAJ
Year of Publication 26.11.2020
Get full text
Year of Publication 26.11.2020
Patent
NLRP3 INFLAMMASOME INHIBITORS
SMITH, Nichola, VELCICKY, Juraj, FARADY, Christopher, MATTES, Henri, GOMMERMANN, Nina, STIEFL, Nikolaus Johannes, SOLOVAY, Catherine Fooks, VANGREVELINGHE, Eric, MACKAY, Angela, von MATT, Anette, JANSER, Philipp
Year of Publication 19.11.2020
Get full text
Year of Publication 19.11.2020
Patent
NLRP3 INFLAMMASOME INHIBITORS
SMITH, Nichola, VELCICKY, Juraj, FARADY, Christopher, MATTES, Henri, GOMMERMANN, Nina, STIEFL, Nikolaus Johannes, SOLOVAY, Catherine Fooks, VANGREVELINGHE, Eric, MACKAY, Angela, von MATT, Anette, JANSER, Philipp
Year of Publication 19.11.2020
Get full text
Year of Publication 19.11.2020
Patent
Tetrahydro-Pyrido-Pyrimidine Derivatives
Hoegenauer, Klemens, Tufilli, Nicola, Hollingworth, Gregory John, Graveleau, Nadege, Smith, Alexander Baxter, von Matt, Anette, Wolf, Romain, Hebach, Christina, Soldermann, Nicolas, Strang, Ross Sinclair, Zecri, Frederic, Fernandes Gomes Dos Santos, Paulo, Cooke, Nigel Graham, Stowasser, Frank
Year of Publication 17.12.2020
Get full text
Year of Publication 17.12.2020
Patent
USE OF INHIBITORS OF THE ACTIVITY OR FUNCTION OF PI3K
KALIS, CHRISTOPH, STRANG, ROSS, WOLF, ROMAIN, HOGENAUER, KLEMENS, SOLDERMANN, NICOLAS, ZECRI, FREDERIC, STOWASSER, FRANK, TUFILLI, NICOLA, SMITH, ALEXANDER BAXTER, FERNANDES GOMES DOS SANTOS, PAULO ANTONIO, COOKE, NIGEL GRAHAM, FURET, PASCAL, HEBACH, CHRISTINA, HOLLINGWORTH, GREGORY, LEWIS, IAN, VON MATT, ANETTE, STAUFFER, FREDERIC
Year of Publication 25.08.2020
Get full text
Year of Publication 25.08.2020
Patent
Tetrahydro-Pyrido-Pyrimidine Derivatives as PI3Kdelta inhibitors
Hoegenauer, Klemens, Tufilli, Nicola, Hollingworth, Gregory John, Graveleau, Nadege, Smith, Alexander Baxter, von Matt, Anette, Wolf, Romain, Hebach, Christina, Soldermann, Nicolas, Strang, Ross Sinclair, Zecri, Frederic, Fernandes Gomes Dos Santos, Paulo, Cooke, Nigel Graham, Stowasser, Frank
Year of Publication 18.07.2019
Get full text
Year of Publication 18.07.2019
Patent