Orally Active MMP-1 Sparing α-Tetrahydropyranyl and α-Piperidinyl Sulfone Matrix Metalloproteinase (MMP) Inhibitors with Efficacy in Cancer, Arthritis, and Cardiovascular Disease
Becker, Daniel P, Barta, Thomas E, Bedell, Louis J, Boehm, Terri L, Bond, Brian R, Carroll, Jeffery, Carron, Chris P, DeCrescenzo, Gary A, Easton, Alan M, Freskos, John N, Funckes-Shippy, Chris L, Heron, Marcia, Hockerman, Susan, Howard, Carol Pearcy, Kiefer, James R, Li, Madeleine H, Mathis, Karl J, McDonald, Joseph J, Mehta, Pramod P, Munie, Grace E, Sunyer, Teresa, Swearingen, Craig A, Villamil, Clara I, Welsch, Dean, Williams, Jennifer M, Yu, Ying, Yao, Jun
Published in Journal of medicinal chemistry (23.09.2010)
Published in Journal of medicinal chemistry (23.09.2010)
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Journal Article
Structural and Inhibition Analysis Reveals the Mechanism of Selectivity of a Series of Aggrecanase Inhibitors
Tortorella, Micky D., Tomasselli, Alfredo G., Mathis, Karl J., Schnute, Mark E., Woodard, Scott S., Munie, Grace, Williams, Jennifer M., Caspers, Nicole, Wittwer, Arthur J., Malfait, Anne-Marie, Shieh, Huey-Sheng
Published in The Journal of biological chemistry (04.09.2009)
Published in The Journal of biological chemistry (04.09.2009)
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Journal Article
The titerless infected-cells preservation and scale-up (TIPS) method for large-scale production of NO-sensitive human soluble guanylate cyclase (sGC) from insect cells infected with recombinant baculovirus
Wasilko, David J., Edward Lee, S., Stutzman-Engwall, Kim J., Reitz, Beverly A., Emmons, Thomas L., Mathis, Karl J., Bienkowski, Michael J., Tomasselli, Alfredo G., David Fischer, H.
Published in Protein expression and purification (01.06.2009)
Published in Protein expression and purification (01.06.2009)
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Journal Article
High Resolution Crystal Structure of the Catalytic Domain of ADAMTS-5 (Aggrecanase-2)
Shieh, Huey-Sheng, Mathis, Karl J., Williams, Jennifer M., Hills, Robert L., Wiese, Joe F., Benson, Timothy E., Kiefer, James R., Marino, Margaret H., Carroll, Jeffery N., Leone, Joseph W., Malfait, Anne-Marie, Arner, Elizabeth C., Tortorella, Micky D., Tomasselli, Alfredo
Published in The Journal of biological chemistry (18.01.2008)
Published in The Journal of biological chemistry (18.01.2008)
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Journal Article
2-(6-Phenyl-1H-indazol-3-yl)-1H-benzo[d]imidazoles: design and synthesis of a potent and isoform selective PKC-zeta inhibitor
Trujillo, John I, Kiefer, James R, Huang, Wei, Thorarensen, Atli, Xing, Li, Caspers, Nicole L, Day, Jacqueline E, Mathis, Karl J, Kretzmer, Kuniko K, Reitz, Beverley A, Weinberg, Robin A, Stegeman, Roderick A, Wrightstone, Ann, Christine, Lori, Compton, Robert, Li, Xiong
Published in Bioorganic & medicinal chemistry letters (01.02.2009)
Published in Bioorganic & medicinal chemistry letters (01.02.2009)
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Journal Article
Structure-based drug design enables conversion of a DFG-in binding CSF-1R kinase inhibitor to a DFG-out binding mode
Meyers, Marvin J., Pelc, Matthew, Kamtekar, Satwik, Day, Jacqueline, Poda, Gennadiy I., Hall, Molly K., Michener, Marshall L., Reitz, Beverly A., Mathis, Karl J., Pierce, Betsy S., Parikh, Mihir D., Mischke, Deborah A., Long, Scott A., Parlow, John J., Anderson, David R., Thorarensen, Atli
Published in Bioorganic & medicinal chemistry letters (01.03.2010)
Published in Bioorganic & medicinal chemistry letters (01.03.2010)
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Journal Article
Structure analysis reveals the flexibility of the ADAMTS‐5 active site
Shieh, Huey‐Sheng, Tomasselli, Alfredo G., Mathis, Karl J., Schnute, Mark E., Woodard, Scott S., Caspers, Nicole, Williams, Jennifer M., Kiefer, James R., Munie, Grace, Wittwer, Arthur, Malfait, Anne‐Marie, Tortorella, Micky D.
Published in Protein science (01.04.2011)
Published in Protein science (01.04.2011)
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Journal Article
MMP-13 selective α-sulfone hydroxamates: A survey of P1′ heterocyclic amide isosteres
Barta, Thomas E., Becker, Daniel P., Bedell, Louis J., Easton, Alan M., Hockerman, Susan L., Kiefer, James, Munie, Grace E., Mathis, Karl J., Li, Madeleine H., Rico, Joseph G., Villamil, Clara I., Williams, Jennifer M.
Published in Bioorganic & medicinal chemistry letters (15.05.2011)
Published in Bioorganic & medicinal chemistry letters (15.05.2011)
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Journal Article
Surgical management of vertebral malformation in a Manx cat
Havlicek, Martin, Mathis, Karl R., Beck, Jason A., Allan, Graeme S.
Published in Journal of feline medicine and surgery (01.06.2009)
Published in Journal of feline medicine and surgery (01.06.2009)
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Journal Article
High yield purification of soluble guanylate cyclase from bovine lung
Mathis, Karl J., Emmons, Thomas L., Curran, Daniel F., Day, Jacqueline E., Tomasselli, Alfredo G.
Published in Protein expression and purification (01.07.2008)
Published in Protein expression and purification (01.07.2008)
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Journal Article
Purification and characterization of recombinant human soluble guanylate cyclase produced from baculovirus-infected insect cells
Emmons, Thomas L., Mathis, Karl J., Shuck, Mary E., Reitz, Beverly A., Curran, Daniel F., Walker, Mark C., Leone, Joseph W., Day, Jacqueline E., Bienkowski, Michael J., Fischer, H. David, Tomasselli, Alfredo G.
Published in Protein expression and purification (01.06.2009)
Published in Protein expression and purification (01.06.2009)
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Journal Article
Computed Tomographic Diagnosis of Traumatic Atlanto-occipital Rotatory Luxation and Successful Closed Reduction in a Dog
Lye, Gordon, Mathis, Karl, Hill, Sarah, Cattin, Ryan, Hartman, Angela
Published in VCOT Open (01.07.2020)
Published in VCOT Open (01.07.2020)
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Journal Article
Canine cauda equina neuritis secondary to neospora
Lye, Gordon, Mathis, Karl, Hill, Sarah, Hardy, Lorna, Cattin, Ryan
Published in Veterinary record case reports (01.02.2020)
Published in Veterinary record case reports (01.02.2020)
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Journal Article
Mammalian cell production and purification of progenipoietin, a dual-agonist chimaeric haematopoietic growth factor
Wood, David C, Mathis, Karl J, Joy, William D, Minnerly, John C, Pegg, Lyle E, Welply, Joseph K
Published in Biotechnology and applied biochemistry (01.02.2003)
Published in Biotechnology and applied biochemistry (01.02.2003)
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Secretion of active kringle-2-serine protease in Escherichia coli
Obukowicz, Mark G, Gustafson, Mark E, Junger, Kurt D, Leimgruber, Richard M, Wittwer, Arthur J, Wun, Tze Chein, Warren, Thomas G, Bishop, Bruce F, Mathis, Karl J
Published in Biochemistry (Easton) (01.10.1990)
Published in Biochemistry (Easton) (01.10.1990)
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Journal Article
What is your diagnosis? Gastroesophageal intussusception
Mathis, Karl R, Nykamp, Stephanie G, Ringwood, Brendon P, Martin, Dawn M
Published in Journal of the American Veterinary Medical Association (15.02.2013)
Published in Journal of the American Veterinary Medical Association (15.02.2013)
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