Fragment-Based Discovery of Pyrimido[1,2-b]indazole PDE10A Inhibitors
Chino, Ayaka, Seo, Ryushi, Amano, Yasushi, Namatame, Ichiji, Hamaguchi, Wataru, Honbou, Kazuya, Mihara, Takuma, Yamazaki, Mayako, Tomishima, Masaki, Masuda, Naoyuki
Published in Chemical & pharmaceutical bulletin (2018)
Published in Chemical & pharmaceutical bulletin (2018)
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Stepwise Construction of Head-to-Tail-Type Oligothiophenes via Iterative Palladium-Catalyzed CH Arylation and Halogen Exchange
Masuda, Naoyuki, Tanba, Shunsuke, Sugie, Atsushi, Monguchi, Daiki, Koumura, Nagatoshi, Hara, Kohjiro, Mori, Atsunori
Published in Organic letters (04.06.2009)
Published in Organic letters (04.06.2009)
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Addressing phototoxicity observed in a novel series of biaryl derivatives: Discovery of potent, selective and orally active phosphodiesterase 10A inhibitor ASP9436
Hamaguchi, Wataru, Masuda, Naoyuki, Miyamoto, Satoshi, Kikuchi, Shigetoshi, Narazaki, Fumie, Shiina, Yasuhiro, Seo, Ryushi, Amano, Yasushi, Mihara, Takuma, Moriguchi, Hiroyuki, Hattori, Kouji
Published in Bioorganic & medicinal chemistry (01.07.2015)
Published in Bioorganic & medicinal chemistry (01.07.2015)
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Dinuclear Copper(II) 3,4,5-Tri-O-benzylgallate
Mikuriya, Masahiro, Yamakawa, Chihiro, Masuda, Naoyuki, Yoshioka, Daisuke, Yamaguchi, Sayuri, Yamada, Hidetoshi, Mizuta, Tsutomu, Kawata, Naomi, Tanaka, Hidekazu, Handa, Makoto
Published in Open Chemistry Journal (22.03.2019)
Published in Open Chemistry Journal (22.03.2019)
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Potent and orally bioavailable CCR4 antagonists: Synthesis and structure–activity relationship study of 2-aminoquinazolines
Yokoyama, Kazuhiro, Ishikawa, Noriko, Igarashi, Susumu, Kawano, Noriyuki, Masuda, Naoyuki, Hamaguchi, Wataru, Yamasaki, Shingo, Koganemaru, Yohei, Hattori, Kazuyuki, Miyazaki, Takahiro, Ogino, Shin-ichi, Matsumoto, Yuzo, Takeuchi, Makoto, Ohta, Mitsuaki
Published in Bioorganic & medicinal chemistry (2009)
Published in Bioorganic & medicinal chemistry (2009)
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ITERATIVE EXTENSION OF THIOPHENE RING LEADING TO HEAD-TO-TAIL-TYPE OLIGOTHIOPHENES VIA STEPWISE CH ARYLATION AND HALOGEN EXCHANGE SEQUENCE
Tanba, Shunsuke, Sugie, Atsushi, Masuda, Naoyuki, Monguchi, Daiki, Koumura, Nagatoshi, Hara, Kohjiro, Mori, Atsunori
Published in Heterocycles (31.12.2010)
Published in Heterocycles (31.12.2010)
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KDR-5169, a new gastrointestinal prokinetic agent, enhances gastric contractile and emptying activities in dogs and rats
Tazawa, Shigeki, Masuda, Naoyuki, Koizumi, Takashi, Kitazawa, Makio, Nakane, Tokio, Miyata, Hiroshi
Published in European journal of pharmacology (11.01.2002)
Published in European journal of pharmacology (11.01.2002)
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Binding Modes of Two Novel Non-Nucleoside Reverse Transcriptase Inhibitors, YM-215389 and YM-228855, to HIV Type-1 Reverse Transcriptase
Kodama, Eiichi, Orita, Masaya, Masuda, Naoyuki, Yamamoto, Osamu, Fujii, Masahiro, Ohgami, Tetsuro, Kageyama, Shunji, Ohta, Mitsuaki, Hatta, Toshifumi, Inoue, Hiroshi, Suzuki, Hiroshi, Sudo, Kenji, Shimizu, Yasuaki, Matsuoka, Masao
Published in Antiviral chemistry & chemotherapy (01.06.2008)
Published in Antiviral chemistry & chemotherapy (01.06.2008)
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Novel benzimidazole derivatives as phosphodiesterase 10A (PDE10A) inhibitors with improved metabolic stability
Chino, Ayaka, Masuda, Naoyuki, Amano, Yasushi, Honbou, Kazuya, Mihara, Takuma, Yamazaki, Mayako, Tomishima, Masaki
Published in Bioorganic & medicinal chemistry (01.07.2014)
Published in Bioorganic & medicinal chemistry (01.07.2014)
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Synthesis, SAR study, and biological evaluation of novel 2,3-dihydro-1H-imidazo[1,2-a]benzimidazole derivatives as phosphodiesterase 10A inhibitors
Chino, Ayaka, Honda, Shugo, Morita, Masataka, Yonezawa, Koichi, Hamaguchi, Wataru, Amano, Yasushi, Moriguchi, Hiroyuki, Yamazaki, Mayako, Aota, Masaki, Tomishima, Masaki, Masuda, Naoyuki
Published in Bioorganic & medicinal chemistry (15.08.2019)
Published in Bioorganic & medicinal chemistry (15.08.2019)
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