Discovery of a Potent and Selective Tyrosine Kinase 2 Inhibitor: TAK-279
Leit, Silvana, Greenwood, Jeremy, Carriero, Samantha, Mondal, Sayan, Abel, Robert, Ashwell, Mark, Blanchette, Heather, Boyles, Nicholas A., Cartwright, Mark, Collis, Alan, Feng, Shulu, Ghanakota, Phani, Harriman, Geraldine C., Hosagrahara, Vinayak, Kaila, Neelu, Kapeller, Rosanna, Rafi, Salma B., Romero, Donna L., Tarantino, Paul M., Timaniya, Jignesh, Toms, Angela V., Wester, Ronald T., Westlin, William, Srivastava, Bhaskar, Miao, Wenyan, Tummino, Peter, McElwee, Joshua J., Edmondson, Scott D., Masse, Craig E.
Published in Journal of medicinal chemistry (10.08.2023)
Published in Journal of medicinal chemistry (10.08.2023)
Get full text
Journal Article
Syntheses and Biological Evaluation of (+)-Lactacystin and Analogs
Masse, Craig E., Morgan, Adam J., Adams, Julian, Panek, James S.
Published in European journal of organic chemistry (01.07.2000)
Published in European journal of organic chemistry (01.07.2000)
Get full text
Journal Article
A General Method for the Enantioselective Synthesis of Pantolactone Derivatives
Evans, David A, Wu, Jimmy, Masse, Craig E, MacMillan, David W. C
Published in Organic letters (03.10.2002)
Published in Organic letters (03.10.2002)
Get full text
Journal Article
Potent and selective TYK2-JH1 inhibitors highly efficacious in rodent model of psoriasis
Leit, Silvana, Greenwood, Jeremy R., Mondal, Sayan, Carriero, Samantha, Dahlgren, Markus, Harriman, Geraldine C., Kennedy-Smith, Joshua J., Kapeller, Rosana, Lawson, Jon P., Romero, Donna L., Toms, Angela V., Shelley, Mee, Wester, Ronald T., Westlin, William, McElwee, Joshua J., Miao, Wenyan, Edmondson, Scott D., Masse, Craig E.
Published in Bioorganic & medicinal chemistry letters (01.10.2022)
Published in Bioorganic & medicinal chemistry letters (01.10.2022)
Get full text
Journal Article
Anti‐leukaemic activity of the TYK2 selective inhibitor NDI‐031301 in T‐cell acute lymphoblastic leukaemia
Akahane, Koshi, Li, Zhaodong, Etchin, Julia, Berezovskaya, Alla, Gjini, Evisa, Masse, Craig E., Miao, Wenyan, Rocnik, Jennifer, Kapeller, Rosana, Greenwood, Jeremy R., Tiv, Hong, Sanda, Takaomi, Weinstock, David M., Look, A. Thomas
Published in British journal of haematology (01.04.2017)
Published in British journal of haematology (01.04.2017)
Get full text
Journal Article
X‑ray Crystal Structures of Escherichia coli RNA Polymerase with Switch Region Binding Inhibitors Enable Rational Design of Squaramides with an Improved Fraction Unbound to Human Plasma Protein
Molodtsov, Vadim, Fleming, Paul R, Eyermann, Charles J, Ferguson, Andrew D, Foulk, Melinda A, McKinney, David C, Masse, Craig E, Buurman, Ed T, Murakami, Katsuhiko S
Published in Journal of medicinal chemistry (09.04.2015)
Published in Journal of medicinal chemistry (09.04.2015)
Get full text
Journal Article
The Exceptional Chelating Ability of Dimethylaluminum Chloride and Methylaluminum Dichloride. The Merged Stereochemical Impact of α- and β-Stereocenters in Chelate-Controlled Carbonyl Addition Reactions with Enolsilane and Hydride Nucleophiles
Evans, David A, Allison, Brett D, Yang, Michael G, Masse, Craig E
Published in Journal of the American Chemical Society (07.11.2001)
Published in Journal of the American Chemical Society (07.11.2001)
Get full text
Journal Article
Lewis Acid-Mediated Carbocyclization Reactions of Chiral (E)-Crotylsilanes
Masse, Craig E, Dakin, Les A, Knight, Bradford S, Panek, James S
Published in Journal of organic chemistry (26.12.1997)
Published in Journal of organic chemistry (26.12.1997)
Get full text
Journal Article
Design and synthesis of deuterated boceprevir analogs with enhanced pharmacokinetic properties
Morgan, Adam J., Nguyen, Sophia, Uttamsingh, Vinita, Bridson, Gary, Harbeson, Scott, Tung, Roger, Masse, Craig E.
Published in Journal of labelled compounds & radiopharmaceuticals (01.07.2011)
Published in Journal of labelled compounds & radiopharmaceuticals (01.07.2011)
Get full text
Journal Article
TYK2 억제제 및 이의 용도
GREENWOOD JEREMY ROBERT, COWEN SCOTT D, MASSE CRAIG E, MONDAL SAYAN, MCLEAN THOMAS H
Year of Publication 02.04.2020
Get full text
Year of Publication 02.04.2020
Patent
ACC INHIBITORS AND USES THEREOF
GREENWOOD JEREMY ROBERT, MASSE CRAIG E, BHAT SATHESH, HARRIMAN GERALDINE C, HARWOOD JAMES
Year of Publication 30.12.2019
Get full text
Year of Publication 30.12.2019
Patent
ACC INHIBITORS AND USES THEREOF
GREENWOOD JEREMY ROBERT, MASSE CRAIG E, BHAT SATHESH, HARRIMAN GERALDINE C, HARWOOD JAMES
Year of Publication 19.04.2019
Get full text
Year of Publication 19.04.2019
Patent