Design and Application of a DNA-Encoded Macrocyclic Peptide Library
Zhu, Zhengrong, Shaginian, Alex, Grady, LaShadric C, O’Keeffe, Thomas, Shi, Xiangguo E, Davie, Christopher P, Simpson, Graham L, Messer, Jeffrey A, Evindar, Ghotas, Bream, Robert N, Thansandote, Praew P, Prentice, Naomi R, Mason, Andrew M, Pal, Sandeep
Published in ACS chemical biology (19.01.2018)
Published in ACS chemical biology (19.01.2018)
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MrgX2 is a promiscuous receptor for basic peptides causing mast cell pseudo‐allergic and anaphylactoid reactions
Grimes, Jak, Desai, Sapna, Charter, Neil W., Lodge, James, Moita Santos, Rita, Isidro‐Llobet, Albert, Mason, Andrew M., Wu, Zining, Wolfe, Lawrence A., Anantharaman, Lakshmi, Green, Andrew, Bridges, Angela M., Dalmas Wilk, Deidre A., Brown, Andrew J.
Published in Pharmacology research & perspectives (01.12.2019)
Published in Pharmacology research & perspectives (01.12.2019)
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Efficient two directional syntheses of a homophthalate ester and novel resorcylate oligomers
Patel, Bhavesh H., Heath, Scott F.A., Mason, Andrew M., Barrett, Anthony G.M.
Published in Tetrahedron letters (27.04.2011)
Published in Tetrahedron letters (27.04.2011)
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The discovery of GSK221149A: A potent and selective oxytocin antagonist
Liddle, John, Allen, Michael J., Borthwick, Alan D., Brooks, David P., Davies, David E., Edwards, Richard M., Exall, Anne M., Hamlett, Chris, Irving, Wendy R., Mason, Andrew M., McCafferty, Gerald P., Nerozzi, Fabrizio, Peace, Simon, Philp, Joanne, Pollard, Derek, Pullen, Mark A., Shabbir, Shaila S., Sollis, Steve L., Westfall, Timothy D., Woollard, Pat M., Wu, Charlene, Hickey, Deirdre M.B.
Published in Bioorganic & medicinal chemistry (2008)
Published in Bioorganic & medicinal chemistry (2008)
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In Vivo Half-Life Extension of BMP1/TLL Metalloproteinase Inhibitors Using Small-Molecule Human Serum Albumin Binders
Vantourout, Julien C, Mason, Andrew M, Yuen, Josephine, Simpson, Graham L, Evindar, Ghotas, Kuai, Letian, Hobbs, Michael, Edgar, Emma, Needle, Saul, Bai, Xiaopeng, Wilson, Steve, Scott-Stevens, Paul, Traylen, William, Lambert, Kim, Young, Neil, Bunally, Shenaz, Summerfield, Scott G, Snell, Richard, Lad, Rakesh, Shi, Eric, Skinner, Steven, Shewchuk, Lisa, Watson, Allan J.B, Chung, Chun-wa, Pal, Sandeep, Holt, Dennis A, Kallander, Lara S, Prendergast, Joanne, Rivera, Katrina, Washburn, David G, Harpel, Mark R, Arico-Muendel, Christopher, Isidro-Llobet, Albert
Published in Bioconjugate chemistry (17.02.2021)
Published in Bioconjugate chemistry (17.02.2021)
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Design, synthesis and evaluation of E2‐25K derived stapled peptides
Watson, Morag E., Scott, Daniel, Jamieson, Craig, Layfield, Robert, Mason, Andrew M.
Published in Peptide science (Hoboken, N.J.) (01.01.2021)
Published in Peptide science (Hoboken, N.J.) (01.01.2021)
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Pyridyl-2,5-Diketopiperazines as Potent, Selective, and Orally Bioavailable Oxytocin Antagonists: Synthesis, Pharmacokinetics, and In Vivo Potency
Borthwick, Alan D, Liddle, John, Davies, Dave E, Exall, Anne M, Hamlett, Christopher, Hickey, Deirdre M, Mason, Andrew M, Smith, Ian E. D, Nerozzi, Fabrizio, Peace, Simon, Pollard, Derek, Sollis, Steve L, Allen, Michael J, Woollard, Patrick M, Pullen, Mark A, Westfall, Timothy D, Stanislaus, Dinesh J
Published in Journal of medicinal chemistry (26.01.2012)
Published in Journal of medicinal chemistry (26.01.2012)
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Structure- and property-based design of factor Xa inhibitors: Pyrrolidin-2-ones with acyclic alanyl amides as P4 motifs
Young, Robert J., Campbell, Matthew, Borthwick, Alan D., Brown, David, Burns-Kurtis, Cynthia L., Chan, Chuen, Convery, Máire A., Crowe, Miriam C., Dayal, Satish, Diallo, Hawa, Kelly, Henry A., Paul King, N., Kleanthous, Savvas, Mason, Andrew M., Mordaunt, Jackie E., Patel, Champa, Pateman, Anthony J., Senger, Stefan, Shah, Gita P., Smith, Paul W., Watson, Nigel S., Weston, Helen E., Zhou, Ping
Published in Bioorganic & medicinal chemistry letters (01.12.2006)
Published in Bioorganic & medicinal chemistry letters (01.12.2006)
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Journal Article
Structure and property based design of factor Xa inhibitors: Pyrrolidin-2-ones with biaryl P4 motifs
Young, Robert J., Borthwick, Alan D., Brown, David, Burns-Kurtis, Cynthia L., Campbell, Matthew, Chan, Chuen, Charbaut, Marie, Chung, Chun-wa, Convery, Máire A., Kelly, Henry A., Paul King, N., Kleanthous, Savvas, Mason, Andrew M., Pateman, Anthony J., Patikis, Angela N., Pinto, Ivan L., Pollard, Derek R., Senger, Stefan, Shah, Gita P., Toomey, John R., Watson, Nigel S., Weston, Helen E.
Published in Bioorganic & medicinal chemistry (2008)
Published in Bioorganic & medicinal chemistry (2008)
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Journal Article
Structure and property based design of factor Xa inhibitors: Biaryl pyrrolidin-2-ones incorporating basic heterocyclic motifs
Young, Robert J., Borthwick, Alan D., Brown, David, Burns-Kurtis, Cynthia L., Campbell, Matthew, Chan, Chuen, Charbaut, Marie, Convery, Máire A., Diallo, Hawa, Hortense, Eric, Irving, Wendy R., Kelly, Henry A., King, N. Paul, Kleanthous, Savvas, Mason, Andrew M., Pateman, Anthony J., Patikis, Angela N., Pinto, Ivan L., Pollard, Derek R., Senger, Stefan, Shah, Gita P., Toomey, John R., Watson, Nigel S., Weston, Helen E., Zhou, Ping
Published in Bioorganic & medicinal chemistry (2008)
Published in Bioorganic & medicinal chemistry (2008)
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Journal Article
Design and synthesis of orally active pyrrolidin-2-one-based factor Xa inhibitors
Watson, Nigel S., Brown, David, Campbell, Matthew, Chan, Chuen, Chaudry, Laiq, Convery, Máire A., Fenwick, Rebecca, Hamblin, J. Nicole, Haslam, Claudine, Kelly, Henry A., King, N. Paul, Kurtis, Cynthia L., Leach, Andrew R., Manchee, Gary R., Mason, Andrew M., Mitchell, Charlotte, Patel, Champa, Patel, Vipulkumar K., Senger, Stefan, Shah, Gita P., Weston, Helen E., Whitworth, Caroline, Young, Robert J.
Published in Bioorganic & medicinal chemistry letters (15.07.2006)
Published in Bioorganic & medicinal chemistry letters (15.07.2006)
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Design and Synthesis of Pyrrolidine-5,5-trans-lactams (5-Oxohexahydropyrrolo[3,2-b]pyrroles) as Novel Mechanism-Based Inhibitors of Human Cytomegalovirus Protease. 2. Potency and Chirality
Borthwick, Alan D, Crame, Andrew J, Ertl, Peter F, Exall, Anne M, Haley, Terry M, Hart, Graham J, Mason, Andrew M, Pennell, Andrew M. K, Singh, Onkar M. P, Weingarten, Gordon G, Woolven, James M
Published in Journal of medicinal chemistry (03.01.2002)
Published in Journal of medicinal chemistry (03.01.2002)
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Journal Article
Design and Synthesis of Pyrrolidine-5,5-trans-lactams (5-Oxo-hexahydro-pyrrolo[3,2-b]pyrroles) as Novel Mechanism-Based Inhibitors of Human Cytomegalovirus Protease. 1. The α-Methyl-trans-lactam Template
Borthwick, Alan D, Angier, S. Jane, Crame, Andrew J, Exall, Anne M, Haley, Terry M, Hart, Graham J, Mason, Andrew M, Pennell, Andrew M. K, Weingarten, Gordon G
Published in Journal of medicinal chemistry (16.11.2000)
Published in Journal of medicinal chemistry (16.11.2000)
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Pyrrolidine-5,5- trans-lactams as novel mechanism-based inhibitors of human cytomegalovirus protease. Part 3: potency and plasma stability
Borthwick, Alan D, Exall, Anne M, Haley, Terry M, Jackson, Deborah L, Mason, Andrew M, Weingarten, Gordon G
Published in Bioorganic & medicinal chemistry letters (08.07.2002)
Published in Bioorganic & medicinal chemistry letters (08.07.2002)
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