Reversal of tumoral immune resistance by inhibition of tryptophan 2,3-dioxygenase
Pilotte, Luc, Larrieu, Pierre, Stroobant, Vincent, Colau, Didier, Dolušić, Eduard, Frédérick, Raphaël, De Plaen, Etienne, Uyttenhove, Catherine, Wouters, Johan, Masereel, Bernard, Van den Eynde, Benoît J
Published in Proceedings of the National Academy of Sciences - PNAS (14.02.2012)
Published in Proceedings of the National Academy of Sciences - PNAS (14.02.2012)
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Journal Article
Targeting tumor-associated carbonic anhydrase IX in cancer therapy
Thiry, Anne, Dogné, Jean-Michel, Masereel, Bernard, Supuran, Claudiu T.
Published in Trends in pharmacological sciences (Regular ed.) (01.11.2006)
Published in Trends in pharmacological sciences (Regular ed.) (01.11.2006)
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Journal Article
Tryptophan 2,3-Dioxygenase (TDO) Inhibitors. 3-(2-(Pyridyl)ethenyl)indoles as Potential Anticancer Immunomodulators
Dolušić, Eduard, Larrieu, Pierre, Moineaux, Laurence, Stroobant, Vincent, Pilotte, Luc, Colau, Didier, Pochet, Lionel, Van den Eynde, Benoît, Masereel, Bernard, Wouters, Johan, Frédérick, Raphaël
Published in Journal of medicinal chemistry (11.08.2011)
Published in Journal of medicinal chemistry (11.08.2011)
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Journal Article
Validation and standardization of the ETP-based activated protein C resistance test for the clinical investigation of steroid contraceptives in women: an unmet clinical and regulatory need
Douxfils, Jonathan, Morimont, Laure, Delvigne, Anne-Sophie, Devel, Philippe, Masereel, Bernard, Haguet, Hélène, Bouvy, Céline, Dogné, Jean-Michel
Published in Clinical chemistry and laboratory medicine (28.01.2020)
Published in Clinical chemistry and laboratory medicine (28.01.2020)
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Journal Article
Specific inhibition of carbonic anhydrase IX activity enhances the in vivo therapeutic effect of tumor irradiation
Dubois, Ludwig, Peeters, Sarah, Lieuwes, Natasja G, Geusens, Nele, Thiry, Anne, Wigfield, Simon, Carta, Fabrizio, Mcintyre, Alan, Scozzafava, Andrea, Dogné, Jean-Michel, Supuran, Claudiu T, Harris, Adrian L, Masereel, Bernard, Lambin, Philippe
Published in Radiotherapy and oncology (01.06.2011)
Published in Radiotherapy and oncology (01.06.2011)
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Journal Article
Carbonic anhydrase inhibitors as anticonvulsant agents
Thiry, Anne, Dogné, Jean-Michel, Supuran, Claudiu T, Masereel, Bernard
Published in Current topics in medicinal chemistry (01.05.2007)
Published in Current topics in medicinal chemistry (01.05.2007)
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Journal Article
Novel 3-Carboxamide-coumarins as Potent and Selective FXIIa Inhibitors
Robert, Séverine, Bertolla, Carine, Masereel, Bernard, Dogné, Jean-Michel, Pochet, Lionel
Published in Journal of medicinal chemistry (12.06.2008)
Published in Journal of medicinal chemistry (12.06.2008)
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Journal Article
Recent Developments of Carbonic Anhydrase Inhibitors as Potential Anticancer Drugs
Thiry, Anne, Supuran, Claudiu T, Masereel, Bernard, Dogné, Jean-Michel
Published in Journal of medicinal chemistry (12.06.2008)
Published in Journal of medicinal chemistry (12.06.2008)
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Journal Article
Discovery and preliminary SARs of keto-indoles as novel indoleamine 2,3-dioxygenase (IDO) inhibitors
Dolušić, Eduard, Larrieu, Pierre, Blanc, Sébastien, Sapunaric, Frédéric, Pouyez, Jenny, Moineaux, Laurence, Colette, Delphine, Stroobant, Vincent, Pilotte, Luc, Colau, Didier, Ferain, Thierry, Fraser, Graeme, Galleni, Moreno, Frère, Jean-Marie, Masereel, Bernard, Van den Eynde, Benoît, Wouters, Johan, Frédérick, Raphaël
Published in European journal of medicinal chemistry (01.07.2011)
Published in European journal of medicinal chemistry (01.07.2011)
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Coumarin and Isocoumarin as Serine Protease Inhibitors
Pochet, Lionel, Frederick, Raphael, Masereel, Bernard
Published in Current pharmaceutical design (01.11.2004)
Published in Current pharmaceutical design (01.11.2004)
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Journal Article
Effects of SiC nanoparticles orally administered in a rat model: Biodistribution, toxicity and elemental composition changes in feces and organs
Lozano, Omar, Laloy, Julie, Alpan, Lütfiye, Mejia, Jorge, Rolin, Stéphanie, Toussaint, Olivier, Dogné, Jean-Michel, Lucas, Stéphane, Masereel, Bernard
Published in Toxicology and applied pharmacology (15.10.2012)
Published in Toxicology and applied pharmacology (15.10.2012)
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Journal Article
Is thrombin generation the new rapid, reliable and relevant pharmacological tool for the development of anticoagulant drugs?
Robert, Séverine, Ghiotto, Jérémie, Pirotte, Bernard, David, Jean-Louis, Masereel, Bernard, Pochet, Lionel, Dogné, Jean-Michel
Published in Pharmacological research (01.03.2009)
Published in Pharmacological research (01.03.2009)
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Indanesulfonamides as Carbonic Anhydrase Inhibitors. Toward Structure-Based Design of Selective Inhibitors of the Tumor-Associated Isozyme CA IX
Thiry, Anne, Ledecq, Marie, Cecchi, Alessandro, Dogné, Jean-Michel, Wouters, Johan, Supuran, Claudiu T, Masereel, Bernard
Published in Journal of medicinal chemistry (04.05.2006)
Published in Journal of medicinal chemistry (04.05.2006)
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Journal Article
Dual carbonic anhydrase--cyclooxygenase-2 inhibitors
Dogné, Jean-Michel, Thiry, Anne, Pratico, Domenico, Masereel, Bernard, Supuran, Claudiu T
Published in Current topics in medicinal chemistry (01.05.2007)
Published in Current topics in medicinal chemistry (01.05.2007)
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Journal Article
Antibody-functionalized polymer-coated gold nanoparticles targeting cancer cells: an in vitro and in vivo study
Marega, Riccardo, Karmani, Linda, Flamant, Lionel, Nageswaran, Praveen Ganesh, Valembois, Vanessa, Masereel, Bernard, Feron, Olivier, Borght, Thierry Vander, Lucas, Stephane, Michiels, Carine, Gallez, Bernard, Bonifazi, Davide
Published in Journal of materials chemistry (01.01.2012)
Published in Journal of materials chemistry (01.01.2012)
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Journal Article
Data in support of a harmine-derived beta-carboline in vitro effects in cancer cells through protein synthesis
Carvalho, Annelise, Chu, Jennifer, Meinguet, Céline, Kiss, Robert, Vandenbussche, Guy, Masereel, Bernard, Wouters, Johan, Kornienko, Alexander, Pelletier, Jerry, Mathieu, Véronique
Published in Data in brief (01.06.2017)
Published in Data in brief (01.06.2017)
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Journal Article
New Developments on Thromboxane and Prostacyclin Modulators Part II: Prostacyclin Modulators
DE LEVAL, Xavier, HANSON, Julien, DAVID, Jean-Louis, MASEREEL, Bernard, PIROTTE, Bernard, DOGNE, Jean-Michel
Published in Current medicinal chemistry (01.05.2004)
Published in Current medicinal chemistry (01.05.2004)
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New Developments on Thromboxane and Prostacyclin Modulators Part I: Thromboxane Modulators
DOGNE, Jean-Michel, DE LEVAL, Xavier, KOLH, Philippe, HANSON, Julien, FREDERICH, Michel, LAMBERMONT, Bernard, GHUYSEN, Alexandre, CASINI, Angela, MASEREEL, Bernard, RUAN, Ke-He, PIROTTE, Bernard
Published in Current medicinal chemistry (01.05.2004)
Published in Current medicinal chemistry (01.05.2004)
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