Design and optimization of cyclized NK1 antagonists with controlled atropisomeric properties
Albert, JS, Ohnmacht, C, Bernstein, PR, Rumsey, WL, Aharony, D, Masek, BB, Dembofsky, BT, Koether, GM, Potts, W, Evenden, JL
Published in Tetrahedron (10.05.2004)
Published in Tetrahedron (10.05.2004)
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Naphtho[2,1-b][1,5] and [1,2-f][1,4]oxazocines as selective NK1 antagonists
OHNMACHT, Cyrus J, ALBERT, Jeffrey S, BERNSTEIN, Peter R, RUMSEY, William L, MASEK, Brian B, DEMBOFSKY, Bruce T, KOETHER, Gerard M, ANDISIK, Donald W, AHARONY, David
Published in Bioorganic & medicinal chemistry (15.05.2004)
Published in Bioorganic & medicinal chemistry (15.05.2004)
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Molecular shape comparison of angiotensin II receptor antagonists
Masek, Brian B, Merchant, Arshad, Matthew, James B
Published in Journal of medicinal chemistry (30.04.1993)
Published in Journal of medicinal chemistry (30.04.1993)
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New nonpeptide angiotensin II receptor antagonists. 1. Synthesis, biological properties, and structure-activity relationships of 2-alkyl benzimidazole derivatives
Thomas, A P, Allott, C P, Gibson, K H, Major, J S, Masek, B B, Oldham, A A, Ratcliffe, A H, Roberts, D A, Russell, S T, Thomason, D A
Published in Journal of medicinal chemistry (06.03.1992)
Published in Journal of medicinal chemistry (06.03.1992)
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New nonpeptide angiotensin II receptor antagonists. 2. Synthesis, biological properties, and structure-activity relationships of 2-alkyl-4-(biphenylylmethoxy)quinoline derivatives
Bradbury, Robert H, Allott, Christopher P, Dennis, Michael, Fisher, Eric, Major, John S, Masek, Brian B, Oldham, Alec A, Pearce, Robert J, Rankine, Neil
Published in Journal of medicinal chemistry (01.10.1992)
Published in Journal of medicinal chemistry (01.10.1992)
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N-aryl-3,3,3-trifluoro-2-hydroxy-2-methylpropanamides: K-ATP potassium channel openers. Modifications on the western region
Ohnmacht, CJ, Russell, K, Empfield, Frank, CA, Gibson, KH, Mayhugh, DR, McLaren, FM, Shapiro, HS, Brown, FJ, Trainor, DA, Ceccarelli, C, Lin, MM, Masek, BB, Forst, JM, Harris, RJ, Hulsizer, JM, Lewis, JJ, Silverman, SM, Smith, RW, Warwick, PJ, Kau, ST, Chun, AL, Grant, TL, Howe, BB, Li, JH, Trivedi, S, Halterman, TJ, Yochim, C, Dyroff, MC, Kirkland, M, Neilson, KL
Published in Journal of medicinal chemistry (08.11.1996)
Published in Journal of medicinal chemistry (08.11.1996)
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EAI-TupletScore, a pharmacophore and shape driven ligand-based de-novo design algorithm
Smith, KM, Masek, BB, Clark, RD, Mansley, T, Abrahamian, E, Nagy, S
Published in Chemistry Central journal (05.06.2009)
Published in Chemistry Central journal (05.06.2009)
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N -Aryl-3,3,3-trifluoro-2-hydroxy-2-methylpropanamides: K ATP Potassium Channel Openers. Modifications on the Western Region
Ohnmacht, Cyrus J., Russell, Keith, Empfield, James R., Frank, Cathy A., Gibson, Keith H., Mayhugh, Daniel R., McLaren, Frances M., Shapiro, Howard S., Brown, Frederick J., Trainor, Diane A., Ceccarelli, Christopher, Lin, Margaret M., Masek, Brian B., Forst, Janet M., Harris, Robert J., Hulsizer, James M., Lewis, Joseph J., Silverman, Stuart M., Smith, Reed W., Warwick, Paul J., Kau, Sen T., Chun, Alexa L., Grant, Thomas L., Howe, Burton B., Li, Jack H., Trivedi, Shephali, Halterman, Tracy J., Yochim, Christopher, Dyroff, Martin C., M.Kirkland, and, Neilson, Kathleen L.
Published in Journal of medicinal chemistry (14.03.1997)
Published in Journal of medicinal chemistry (14.03.1997)
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