YM155, a novel small-molecule survivin suppressant, induces regression of established human hormone-refractory prostate tumor xenografts
NAKAHARA, Takahito, TAKEUCHI, Masahiro, SASAMATA, Masao, KINOYAMA, Isao, MINEMATSU, Tsuyoshi, SHIRASUNA, Kenna, MATSUHISA, Akira, KITA, Aya, TOMINAGA, Fumiko, YAMANAKA, Kentaro, KUDOH, Masafumi
Published in Cancer research (Chicago, Ill.) (01.09.2007)
Published in Cancer research (Chicago, Ill.) (01.09.2007)
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The selective anaplastic lymphoma receptor tyrosine kinase inhibitor ASP3026 induces tumor regression and prolongs survival in non-small cell lung cancer model mice
Mori, Masamichi, Ueno, Yoko, Konagai, Satoshi, Fushiki, Hiroshi, Shimada, Itsuro, Kondoh, Yutaka, Saito, Rika, Mori, Kenichi, Shindou, Nobuaki, Soga, Takatoshi, Sakagami, Hideki, Furutani, Takashi, Doihara, Hitoshi, Kudoh, Masafumi, Kuromitsu, Sadao
Published in Molecular cancer therapeutics (01.02.2014)
Published in Molecular cancer therapeutics (01.02.2014)
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YM-359445, an Orally Bioavailable Vascular Endothelial Growth Factor Receptor-2 Tyrosine Kinase Inhibitor, Has Highly Potent Antitumor Activity against Established Tumors
Amino, Nobuaki, Ideyama, Yukitaka, Yamano, Mayumi, Kuromitsu, Sadao, Tajinda, Katsuinori, Samizu, Kiyohiro, Hisamichi, Hiroyuki, Matsuhisa, Akira, Shirasuna, Kenna, Kudoh, Masafumi, Shibasaki, Masayuki
Published in Clinical cancer research (01.03.2006)
Published in Clinical cancer research (01.03.2006)
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N-Arylpiperazine-1-carboxamide Derivatives: a Novel Series of Orally Active Nonsteroidal Androgen Receptor Antagonists
Kinoyama, Isao, Taniguchi, Nobuaki, Kawaminami, Eiji, Nozawa, Eisuke, Koutoku, Hiroshi, Furutani, Takashi, Kudoh, Masafumi, Okada, Minoru
Published in Chemical & Pharmaceutical Bulletin (2005)
Published in Chemical & Pharmaceutical Bulletin (2005)
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A role of androgen receptor protein in cell growth of an androgen-independent prostate cancer cell line
Furutani, T.(Astellas Pharma Inc., Tsukuba, Ibaraki (Japan). Drug Discovery Research), Takeyama, K, Koutoku, H, Ito, S, Taniguchi, N, Suzuki, E, Kudoh, M, Shibasaki, M, Shikama, H, Kato, S
Published in Bioscience, biotechnology, and biochemistry (01.11.2005)
Published in Bioscience, biotechnology, and biochemistry (01.11.2005)
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YM-231146, a Novel Orally Bioavailable Inhibitor of Vascular Endothelial Growth Factor Receptor-2, Is Effective against Paclitaxel Resistant Tumors
Amino, Nobuaki, Ideyama, Yukitaka, Yamano, Mayumi, Kuromitsu, Sadao, Tajinda, Katsunori, Samizu, Kiyohiro, Matsuhisa, Akira, Shirasuna, Kenna, Kudoh, Masafumi, Shibasaki, Masayuki
Published in Biological & Pharmaceutical Bulletin (01.11.2005)
Published in Biological & Pharmaceutical Bulletin (01.11.2005)
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Human Expanded Polyglutamine Androgen Receptor Mutants in Neurodegeneration as a Novel Ligand Target
Furutani, Takashi, Takeyama, Ken-ichi, Tanabe, Masahiko, Koutoku, Hiroshi, Ito, Saya, Taniguchi, Nobuaki, Suzuki, Eriko, Kudoh, Masafumi, Shibasaki, Masayuki, Shikama, Hisataka, Kato, Shigeaki
Published in The Journal of pharmacology and experimental therapeutics (01.11.2005)
Published in The Journal of pharmacology and experimental therapeutics (01.11.2005)
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Synthesis and Pharmacological Evaluation of Novel Arylpiperazine Derivatives as Nonsteroidal Androgen Receptor Antagonists
Kinoyama, Isao, Taniguchi, Nobuaki, Yoden, Toru, Koutoku, Hiroshi, Furutani, Takashi, Kudoh, Masafumi, Okada, Minoru
Published in Chemical & Pharmaceutical Bulletin (01.11.2004)
Published in Chemical & Pharmaceutical Bulletin (01.11.2004)
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RETRACTION: Human Expanded Polyglutamine Androgen Receptor Mutants in Neurodegeneration as a Novel Ligand Target
Furutani, Takashi, Takeyama, Ken-ichi, Tanabe, Masahiko, Koutoku, Hiroshi, Ito, Saya, Taniguchi, Nobuaki, Suzuki, Eriko, Kudoh, Masafumi, Shibasaki, Masayuki, Shikama, Hisataka, Kato, Shigeaki
Published in The Journal of pharmacology and experimental therapeutics (01.11.2005)
Published in The Journal of pharmacology and experimental therapeutics (01.11.2005)
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Journal Article
Studies on Aromatase Inhibitors. I. Synthesis and Biological Evaluation of 4-Amino-4H-1, 2, 4-triazole Derivatives
OKADA, Minoru, YODEN, Toru, KAWAMINAMI, Eiji, SHIMADA, Yoshiaki, KUDOH, Masafumi, ISOMURA, Yasuo, SHIKAMA, Hisataka, FUJIKURA, Takashi
Published in Chemical & pharmaceutical bulletin (1996)
Published in Chemical & pharmaceutical bulletin (1996)
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Inhibitory effect of a novel non-steroidal aromatase inhibitor, YM511 on the proliferation of MCF-7 human breast cancer cell
Kudoh, Masafumi, Susaki, Yoko, Ideyama, Yukitaka, Nanya, Taiki, Mori, Masamichi, Shikama, Hisataka, Fujikura, Takashi
Published in The Journal of steroid biochemistry and molecular biology (01.05.1996)
Published in The Journal of steroid biochemistry and molecular biology (01.05.1996)
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Studies on Aromatase Inhibitors. III. Synthesis and Biological Evaluation of ((4-Bromobenzyl)(4-cyanophenyl)amino)azoles and Their Azine Analogs
OKADA, Minoru, YODEN, Toru, KAWAMINAMI, Eiji, SHIMADA, Yoshiaki, KUDOH, Masafumi, ISOMURA, Yasuo
Published in Chemical & pharmaceutical bulletin (1997)
Published in Chemical & pharmaceutical bulletin (1997)
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YM-201627: An orally active antitumor agent with selective inhibition of vascular endothelial cell proliferation
Amino, Nobuaki, Ideyama, Yukitaka, Yamano, Mayumi, Kuromitsu, Sadao, Tajinda, Katsunori, Samizu, Kiyohiro, Matsuhisa, Akira, Kudoh, Masafumi, Shibasaki, Masayuki
Published in Cancer letters (08.07.2006)
Published in Cancer letters (08.07.2006)
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Bag1 proteins regulate growth and survival of ZR-75-1 human breast cancer cells
KUDOH, Masafumi, KNEE, Deborah A, TAKAYAMA, Shinichi, REED, John C
Published in Cancer research (Chicago, Ill.) (15.03.2002)
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Published in Cancer research (Chicago, Ill.) (15.03.2002)
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(+)-(2R,5S)-4-[4-Cyano-3-(trifluoromethyl)phenyl]-2,5-dimethyl-N-[6-(trifluoromethyl)pyridin-3- yl]piperazine-1-carboxamide (YM580) as an Orally Potent and Peripherally Selective Nonsteroidal Androgen Receptor Antagonist
Kinoyama, Isao, Taniguchi, Nobuaki, Toyoshima, Akira, Nozawa, Eisuke, Kamikubo, Takashi, Imamura, Masakazu, Matsuhisa, Akira, Samizu, Kiyohiro, Kawanimani, Eiji, Niimi, Tatsuya, Hamada, Noritaka, Koutoku, Hiroshi, Furutani, Takashi, Kudoh, Masafumi, Okada, Minoru, Ohta, Mitsuaki, Tsukamoto, Shin-ichi
Published in Journal of medicinal chemistry (26.01.2006)
Published in Journal of medicinal chemistry (26.01.2006)
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Journal Article
Stabilization of androgen receptor protein is induced by agonist, not by antagonists
Furutani, Takashi, Watanabe, Tomoyuki, Tanimoto, Kyouko, Hashimoto, Takamichi, Koutoku, Hiroshi, Kudoh, Masafumi, Shimizu, Yasuaki, Kato, Shigeaki, Shikama, Hisataka
Published in Biochemical and biophysical research communications (21.06.2002)
Published in Biochemical and biophysical research communications (21.06.2002)
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Journal Article
YM116, 2-(1H-Imidazol-4-ylmethyl)-9H-carbazole, Decreases Adrenal Androgen Synthesis by Inhibiting C17-20 Lyase Activity in NCI-H295 Human Adrenocortical Carcinoma Cells
Ideyama, Yukitaka, Kudoh, Masafumi, Tanimoto, Kyoko, Susaki, Yoko, Nanya, Taiki, Nakahara, Takahito, Ishikawa, Hiroko, Fujikura, Takashi, Akaza, Hideyuki, Shikama, Hisataka
Published in Japanese Journal of Pharmacology (1999)
Published in Japanese Journal of Pharmacology (1999)
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YM-359445, an orally bioavailable vascular endothelial growth factor receptor-2 tyrosine klinase inhibitor, has highly potent antitumor activity against established tumors
AMINO, Nobuaki, IDEYAMA, Yukitaka, SHIBASAKI, Masayuki, YAMANO, Mayumi, KUROMITSU, Sadao, TAJINDA, Katsuinori, SAMIZU, Kiyohiro, HISAMICHI, Hiroyuki, MATSUHISA, Akira, SHIRASUNA, Kenna, KUDOH, Masafumi
Published in Clinical cancer research (2006)
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Published in Clinical cancer research (2006)
Journal Article
N-Arylpiperazine-1-carboxamide Derivatives
Kinoyama, Isao, Taniguchi, Nobuaki, Kawaminami, Eiji, Nozawa, Eisuke, Koutoku, Hiroshi, Furutani, Takashi, Kudoh, Masafumi, Okada, Minoru
Published in Chemical & pharmaceutical bulletin (01.04.2005)
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Published in Chemical & pharmaceutical bulletin (01.04.2005)
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