Paradox-Breaking RAF Inhibitors that Also Target SRC Are Effective in Drug-Resistant BRAF Mutant Melanoma
Girotti, Maria Romina, Lopes, Filipa, Preece, Natasha, Niculescu-Duvaz, Dan, Zambon, Alfonso, Davies, Lawrence, Whittaker, Steven, Saturno, Grazia, Viros, Amaya, Pedersen, Malin, Suijkerbuijk, Bart M.J.M., Menard, Delphine, McLeary, Robert, Johnson, Louise, Fish, Laura, Ejiama, Sarah, Sanchez-Laorden, Berta, Hohloch, Juliane, Carragher, Neil, Macleod, Kenneth, Ashton, Garry, Marusiak, Anna A., Fusi, Alberto, Brognard, John, Frame, Margaret, Lorigan, Paul, Marais, Richard, Springer, Caroline
Published in Cancer cell (12.01.2015)
Published in Cancer cell (12.01.2015)
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Journal Article
Mixed lineage kinases activate MEK independently of RAF to mediate resistance to RAF inhibitors
Marusiak, Anna A, Edwards, Zoe C, Hugo, Willy, Trotter, Eleanor W, Girotti, Maria R, Stephenson, Natalie L, Kong, Xiangju, Gartside, Michael G, Fawdar, Shameem, Hudson, Andrew, Breitwieser, Wolfgang, Hayward, Nicholas K, Marais, Richard, Lo, Roger S, Brognard, John
Published in Nature communications (22.05.2014)
Published in Nature communications (22.05.2014)
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Journal Article
MLK4 regulates DNA damage response and promotes triple-negative breast cancer chemoresistance
Mehlich, Dawid, Łomiak, Michał, Sobiborowicz, Aleksandra, Mazan, Alicja, Dymerska, Dagmara, Szewczyk, Łukasz M, Mehlich, Anna, Borowiec, Agnieszka, Prełowska, Monika K, Gorczyński, Adam, Jabłoński, Paweł, Iżycka-Świeszewska, Ewa, Nowis, Dominika, Marusiak, Anna A
Published in Cell death & disease (27.11.2021)
Published in Cell death & disease (27.11.2021)
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Journal Article
Targeted genetic dependency screen facilitates identification of actionable mutations in FGFR4, MAP3K9, and PAK5 in lung cancer
Fawdar, Shameem, Trotter, Eleanor W., Li, Yaoyong, Stephenson, Natalie L., Hanke, Franziska, Marusiak, Anna A., Edwards, Zoe C., Ientile, Sara, Waszkowycz, Bohdan, Miller, Crispin J., Brognard, John
Published in Proceedings of the National Academy of Sciences - PNAS (23.07.2013)
Published in Proceedings of the National Academy of Sciences - PNAS (23.07.2013)
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Drivers of cancer metastasis – Arise early and remain present
Dymerska, Dagmara, Marusiak, Anna A.
Published in Biochimica et biophysica acta. Reviews on cancer (01.03.2024)
Published in Biochimica et biophysica acta. Reviews on cancer (01.03.2024)
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Journal Article
Somatically mutated ABL1 is an actionable and essential NSCLC survival gene
Testoni, Ewelina, Stephenson, Natalie L, Torres‐Ayuso, Pedro, Marusiak, Anna A, Trotter, Eleanor W, Hudson, Andrew, Hodgkinson, Cassandra L, Morrow, Christopher J, Dive, Caroline, Brognard, John
Published in EMBO molecular medicine (01.02.2016)
Published in EMBO molecular medicine (01.02.2016)
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Inhibition of the ʟ-glutamine transporter ASCT2 sensitizes plasma cell myeloma cells to proteasome inhibitors
Prelowska, Monika K., Mehlich, Dawid, Ugurlu, M. Talha, Kedzierska, Hanna, Cwiek, Aleksandra, Kosnik, Artur, Kaminska, Klaudia, Marusiak, Anna A., Nowis, Dominika
Published in Cancer letters (01.06.2021)
Published in Cancer letters (01.06.2021)
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Selective Degradation of MLK3 by a Novel CEP1347-VHL-02 PROTAC Compound Limits the Oncogenic Potential of TNBC
Karpińska, Kamila, Mehlich, Dawid, Sabbasani, Venkata R., Łomiak, Michał, Torres-Ayuso, Pedro, Wróbel, Katarzyna, Truong, Vi Nguyen-Phuong, Serwa, Remigiusz, Swenson, Rolf E., Brognard, John, Marusiak, Anna A.
Published in Journal of medicinal chemistry (12.09.2024)
Published in Journal of medicinal chemistry (12.09.2024)
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PIM1 targeted degradation prevents the emergence of chemoresistance in prostate cancer
Torres-Ayuso, Pedro, Katerji, Meghri, Mehlich, Dawid, Lookingbill, Sophia A., Sabbasani, Venkata R., Liou, Hope, Casillas, Andrea L., Chauhan, Shailender S., Serwa, Remigiusz, Rubin, Maxine R., Marusiak, Anna A., Swenson, Rolf E., Warfel, Noel A., Brognard, John
Published in Cell chemical biology (15.02.2024)
Published in Cell chemical biology (15.02.2024)
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Journal Article
Upregulation of MLK4 promotes migratory and invasive potential of breast cancer cells
Marusiak, Anna A, Prelowska, Monika K, Mehlich, Dawid, Lazniewski, Michal, Kaminska, Klaudia, Gorczynski, Adam, Korwat, Aleksandra, Sokolowska, Olga, Kedzierska, Hanna, Golab, Jakub, Biernat, Wojciech, Plewczynski, Dariusz, Brognard, John, Nowis, Dominika
Published in Oncogene (01.04.2019)
Published in Oncogene (01.04.2019)
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Corrigendum to “Inhibition of the ʟ-glutamine transporter ASCT2 sensitizes plasma cell myeloma cells to proteasome inhibitors” [Canc. Lett. 507 (2021) 13–25]
Prelowska, Monika K., Mehlich, Dawid, Ugurlu, M. Talha, Kedzierska, Hanna, Cwiek, Aleksandra, Kosnik, Artur, Kaminska, Klaudia, Marusiak, Anna A., Nowis, Dominika
Published in Cancer letters (01.02.2022)
Published in Cancer letters (01.02.2022)
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Journal Article
Protein Kinase Cδ Deficiency Causes Mendelian Systemic Lupus Erythematosus With B Cell‐Defective Apoptosis and Hyperproliferation
Belot, Alexandre, Kasher, Paul R., Trotter, Eleanor W., Foray, Anne‐Perrine, Debaud, Anne‐Laure, Rice, Gillian I., Szynkiewicz, Marcin, Zabot, Marie‐Therese, Rouvet, Isabelle, Bhaskar, Sanjeev S., Daly, Sarah B., Dickerson, Jonathan E., Mayer, Josephine, O'Sullivan, James, Juillard, Laurent, Urquhart, Jill E., Fawdar, Shameem, Marusiak, Anna A., Stephenson, Natalie, Waszkowycz, Bohdan, Beresford, Michael W., Biesecker, Leslie G., Black, Graeme C. M., René, Céline, Eliaou, Jean‐François, Fabien, Nicole, Ranchin, Bruno, Cochat, Pierre, Gaffney, Patrick M., Rozenberg, Flore, Lebon, Pierre, Malcus, Christophe, Crow, Yanick J., Brognard, John, Bonnefoy, Nathalie
Published in Arthritis & rheumatology (Hoboken, N.J.) (01.08.2013)
Published in Arthritis & rheumatology (Hoboken, N.J.) (01.08.2013)
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Journal Article
Protein Kinase C[delta] Deficiency Causes Mendelian Systemic Lupus Erythematosus With B Cell-Defective Apoptosis and Hyperproliferation
Belot, Alexandre, Kasher, Paul R, Trotter, Eleanor W, ay, Anne-Perrine, Debaud, Anne-Laure, Rice, Gillian I, Szynkiewicz, Marcin, Zabot, Marie-Therese, Rouvet, Isabelle, Bhaskar, Sanjeev S, Daly, Sarah B, Dickerson, Jonathan E, Mayer, Josephine, O'Sullivan, James, Juillard, Laurent, Urquhart, Jill E, Fawdar, Shameem, Marusiak, Anna A, Stephenson, Natalie, Waszkowycz, Bohdan, W. Beresford, Michael, Biesecker, Leslie G, C. M. Black, Graeme, René, Céline, Eliaou, Jean-François, Fabien, Nicole, Ranchin, Bruno, Cochat, Pierre, Gaffney, Patrick M, Rozenberg, Flore, Lebon, Pierre, Malcus, Christophe, Crow, Yanick J, Brognard, John, Bonnefoy, Nathalie
Published in Arthritis & rheumatology (Hoboken, N.J.) (01.08.2013)
Published in Arthritis & rheumatology (Hoboken, N.J.) (01.08.2013)
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Journal Article
Differential responses to kinase inhibition in FGFR2-addicted triple negative breast cancer cells: a quantitative phosphoproteomics study
Cunningham, Debbie L, Sarhan, Adil R, Creese, Andrew J, Larkins, Katherine P B, Zhao, Hongyan, Ferguson, Harriet R, Brookes, Katie, Marusiak, Anna A, Cooper, Helen J, Heath, John K
Published in Scientific reports (14.05.2020)
Published in Scientific reports (14.05.2020)
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Journal Article
Recurrent MLK4 Loss-of-Function Mutations Suppress JNK Signaling to Promote Colon Tumorigenesis
Marusiak, Anna A, Stephenson, Natalie L, Baik, Hayeon, Trotter, Eleanor W, Li, Yaoyong, Blyth, Karen, Mason, Susan, Chapman, Phil, Puto, Lorena A, Read, Jon A, Brassington, Claire, Pollard, Hannah K, Phillips, Chris, Green, Isabelle, Overman, Ross, Collier, Matthew, Testoni, Ewelina, Miller, Crispin J, Hunter, Tony, Sansom, Owen J, Brognard, John
Published in Cancer research (Chicago, Ill.) (01.02.2016)
Published in Cancer research (Chicago, Ill.) (01.02.2016)
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Journal Article
Abstract 4408: Mutant ABL1 is a genetic dependency in non-small cell lung cancer amenable to pharmacological intervention
Torres-Ayuso, PEDRO, Testoni, Ewelina, Stephenson, Natalie L., Marusiak, Anna A., Trotter, Eleanor W., Hudson, Andrew, Hodgkinson, Cassandra L., Morrow, Christopher J., Dive, Caroline, Brognard, John
Published in Cancer research (Chicago, Ill.) (15.07.2016)
Published in Cancer research (Chicago, Ill.) (15.07.2016)
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Journal Article
Paradox-Breaking RAF Inhibitors that Also Target SRC Are Effective in Drug-Resistant BRAF Mutant Melanoma
Girotti, Maria Romina, Lopes, Filipa, Preece, Natasha, Niculescu-Duvaz, Dan, Zambon, Alfonso, Davies, Lawrence, Whittaker, Steven, Saturno, Grazia, Viros, Amaya, Pedersen, Malin, Suijkerbuijk, Bart M.J.M., Menard, Delphine, McLeary, Robert, Johnson, Louise, Fish, Laura, Ejiama, Sarah, Sanchez-Laorden, Berta, Hohloch, Juliane, Carragher, Neil, Macleod, Kenneth, Ashton, Garry, Marusiak, Anna A., Fusi, Alberto, Brognard, John, Frame, Margaret, Lorigan, Paul, Marais, Richard, Springer, Caroline
Published in Cancer cell (13.03.2017)
Published in Cancer cell (13.03.2017)
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