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Year of Publication 19.07.2024
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Year of Publication 19.07.2024
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Modified oligonucleotides and methods of use
MARTINEZ MONTERO SAUL, GRYAZNOV SERGEI, BEIGELMAN LEONID, RAJWANSHI VIVEK, HONG JIN
Year of Publication 24.01.2024
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Year of Publication 24.01.2024
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변형된 짧은 간섭 핵산 (SINA) 분자 및 그의 용도
DEVAL JEROME, LUONG XUAN, MARTINEZ MONTERO SAUL, BEIGELMAN LEONID, DE COSTA N. TILANI S, BHATTACHARYA ANEERBAN
Year of Publication 24.04.2024
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Year of Publication 24.04.2024
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Modified oligonucleotides and methods of use
MARTINEZ MONTERO SAUL, GRYAZNOV SERGEI, BEIGELMAN LEONID, RAJWANSHI VIVEK, HONG JIN
Year of Publication 08.03.2023
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Year of Publication 08.03.2023
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Adjusting the Structure of 2′-Modified Nucleosides and Oligonucleotides via C4′-α‑F or C4′-α-OMe Substitution: Synthesis and Conformational Analysis
Malek-Adamian, Elise, Patrascu, Mihai Burai, Jana, Sunit Kumar, Martínez-Montero, Saúl, Moitessier, Nicolas, Damha, Masad J
Published in Journal of organic chemistry (07.09.2018)
Published in Journal of organic chemistry (07.09.2018)
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변형 올리고뉴클레오티드 및 타우병증에서의 사용 방법
VAN OUTRYVE D'YDEWALLE CONSTANTIN, MARTINEZ MONTERO SAUL, GRYAZNOV SERGEI, BEIGELMAN LEONID, EBNETH ANDREAS, RAJWANSHI VIVEK KUMAR
Year of Publication 23.11.2020
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Year of Publication 23.11.2020
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4′‑C‑Methoxy-2′-deoxy-2′-fluoro Modified Ribonucleotides Improve Metabolic Stability and Elicit Efficient RNAi-Mediated Gene Silencing
Malek-Adamian, Elise, Guenther, Dale C, Matsuda, Shigeo, Martínez-Montero, Saúl, Zlatev, Ivan, Harp, Joel, Burai Patrascu, Mihai, Foster, Donald J, Fakhoury, Johans, Perkins, Lydia, Moitessier, Nicolas, Manoharan, Rajar M, Taneja, Nate, Bisbe, Anna, Charisse, Klaus, Maier, Martin, Rajeev, Kallanthottathil G, Egli, Martin, Manoharan, Muthiah, Damha, Masad J
Published in Journal of the American Chemical Society (18.10.2017)
Published in Journal of the American Chemical Society (18.10.2017)
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변형된 올리고뉴클레오티드 및 사용 방법
MARTINEZ MONTERO SAUL, GRYAZNOV SERGEI, BEIGELMAN LEONID, RAJWANSHI VIVEK, HONG JIN
Year of Publication 07.05.2019
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Year of Publication 07.05.2019
Patent
Locked 2′-Deoxy-2′,4′-Difluororibo Modified Nucleic Acids: Thermal Stability, Structural Studies, and siRNA Activity
Martínez-Montero, Saúl, Deleavey, Glen F, Martín-Pintado, Nerea, Fakhoury, Johans F, González, Carlos, Damha, Masad J
Published in ACS chemical biology (18.09.2015)
Published in ACS chemical biology (18.09.2015)
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Synthesis and Properties of 2′-Deoxy-2′,4′-difluoroarabinose-Modified Nucleic Acids
Martínez-Montero, Saúl, Deleavey, Glen F, Dierker-Viik, Arden, Lindovska, Petra, Ilina, Tatiana, Portella, Guillem, Orozco, Modesto, Parniak, Michael A, González, Carlos, Damha, Masad J
Published in Journal of organic chemistry (20.03.2015)
Published in Journal of organic chemistry (20.03.2015)
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Seven-Membered Ring Nucleoside Analogues: Stereoselective Synthesis and Studies on Their Conformational Properties
Habibian, Maryam, Martínez-Montero, Saúl, Portella, Guillem, Chua, Zhijie, Bohle, D. Scott, Orozco, Modesto, Damha, Masad J
Published in Organic letters (06.11.2015)
Published in Organic letters (06.11.2015)
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CAL-B-Catalyzed Acylation of Nucleosides and Role of the Sugar Conformation: An Improved Understanding of the Enzyme-Substrate Recognition
Martínez-Montero, Saúl, Fernández, Susana, Sanghvi, Yogesh S., Gotor, Vicente, Ferrero, Miguel
Published in European journal of organic chemistry (01.10.2012)
Published in European journal of organic chemistry (01.10.2012)
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Journal Article
Synthesis, Structure, and Conformational Analysis of Nucleoside Analogues Comprising Six-Membered 1,3-Oxathiane Sugar Rings
Abou Assi, Hala, Martínez-Montero, Saúl, Dixit, Dilip M., Chua, Zhijie, Bohle, D. Scott, Damha, Masad J.
Published in European journal of organic chemistry (01.03.2015)
Published in European journal of organic chemistry (01.03.2015)
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Synthesis, evaluation of anti-HIV-1 and anti-HCV activity of novel 2′,3′-dideoxy-2′,2′-difluoro-4′-azanucleosides
Martínez-Montero, Saúl, Fernández, Susana, Sanghvi, Yogesh S., Theodorakis, Emmanuel A., Detorio, Mervi A., Mcbrayer, Tamara R., Whitaker, Tony, Schinazi, Raymond F., Gotor, Vicente, Ferrero, Miguel
Published in Bioorganic & medicinal chemistry (01.12.2012)
Published in Bioorganic & medicinal chemistry (01.12.2012)
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Enzymatic Parallel Kinetic Resolution of Mixtures of d/l 2′-Deoxy and Ribonucleosides: An Approach for the Isolation of β-l-Nucleosides
Martínez-Montero, Saúl, Fernández, Susana, Sanghvi, Yogesh S, Gotor, Vicente, Ferrero, Miguel
Published in Journal of organic chemistry (01.10.2010)
Published in Journal of organic chemistry (01.10.2010)
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THU-198 In vitro and in vivo pharmacological characterization of human PNPLA3-targeting short interfering RNA molecules for the treatment of metabolic dysfunction-associated steatohepatitis
Song, Jieun, Deval, Jerome, Adame, Lillian, Jaisinghani, Ruchika, Tso, Emily, Lin, Daniel, Bhattacharya, Aneerban, Stoycheva, Antitsa, Sousa, Jacquelyn, Parish, Craig, Montero, Saul Martinez, Rajwanshi, Vivek, Daguison, Shane, Gohil, Vikrant, Zhang, Qingling, Williamson, Toni, Chanda, Sushmita, Talukdar, Saswata, Smith, David, Beigelman, Leonid, Symons, Julian, Zhou, Yingjiang, Luong, Xuan
Published in Journal of hepatology (01.06.2024)
Published in Journal of hepatology (01.06.2024)
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Incorporation of novel ASO chemistries significantly improves the potency and durability of HBVASOs in the AAV-HBV mouse model
Hong, Jin, Eltepu, Laxman, Montero, Saul Martinez, Tan, Hua, Hyunsoon, Kang, Rajwanshi, Vivek, Cortez, John, Cai, Dawei, Liu, Cheng, Rosler, Elen, Smith, David, Symons, Julian, Blatt, Lawrence, Beigelman, Leonid
Published in Journal of hepatology (01.07.2022)
Published in Journal of hepatology (01.07.2022)
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Nucleotide Sugar Pucker Preference Mitigates Excision by HIV‑1 RT
Yamada, Ken, Wahba, Alexander S, Bernatchez, Jean A, Ilina, Tatiana, Martínez-Montero, Saúl, Habibian, Maryam, Deleavey, Glen F, Götte, Matthias, Parniak, Michael A, Damha, Masad J
Published in ACS chemical biology (18.09.2015)
Published in ACS chemical biology (18.09.2015)
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Antibody-Antisense Oligonucleotide Conjugate Downregulates a Key Gene in Glioblastoma Stem Cells
Arnold, Amy E., Malek-Adamian, Elise, Le, Phuong U., Meng, Anika, Martínez-Montero, Saúl, Petrecca, Kevin, Damha, Masad J., Shoichet, Molly S.
Published in Molecular therapy. Nucleic acids (01.06.2018)
Published in Molecular therapy. Nucleic acids (01.06.2018)
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Design and Divergent Synthesis of Aza Nucleosides from a Chiral Imino Sugar
Martı́nez-Montero, Saúl, Fernández, Susana, Sanghvi, Yogesh S, Chattopadhyaya, Jyoti, Ganesan, Muthupandian, Ramesh, Namakkal G, Gotor, Vicente, Ferrero, Miguel
Published in Journal of organic chemistry (18.05.2012)
Published in Journal of organic chemistry (18.05.2012)
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