Tetrazine Dynamic Covalent Polymer Networks
Rivero, David S, Paiva-Feener, Rafael E, Santos, Tanausú, Martín-Encinas, Endika, Carrillo, Romen
Published in Macromolecules (23.11.2021)
Published in Macromolecules (23.11.2021)
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Journal Article
Antileishmanial Effect of 1,5- and 1,8-Substituted Fused Naphthyridines
Melcón-Fernandez, Estela, Martín-Encinas, Endika, Palacios, Francisco, Galli, Gulio, Reguera, Rosa M, Martínez-Valladares, María, Balaña-Fouce, Rafael, Alonso, Concepción, Pérez-Pertejo, Yolanda
Published in Molecules (Basel, Switzerland) (22.12.2023)
Published in Molecules (Basel, Switzerland) (22.12.2023)
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Journal Article
Synthesis, biological and computational evaluation of novel cyanomethyl vinyl ether derivatives
Martín-Encinas, Endika, Fuertes, María, Delgado-Hernández, Samuel, García-Tellado, Fernando, Tejedor, David, Alonso, Concepción
Published in Frontiers in pharmacology (04.03.2024)
Published in Frontiers in pharmacology (04.03.2024)
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Journal Article
Dynamic Nucleophilic Aromatic Substitution of Tetrazines
Santos, Tanausú, Rivero, David S., Pérez‐Pérez, Yaiza, Martín‐Encinas, Endika, Pasán, Jorge, Daranas, Antonio Hernández, Carrillo, Romen
Published in Angewandte Chemie (16.08.2021)
Published in Angewandte Chemie (16.08.2021)
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Journal Article
Novel topoisomerase I inhibitors. Syntheses and biological evaluation of phosphorus substituted quinoline derivates with antiproliferative activity
Alonso, Concepción, Fuertes, María, Martín-Encinas, Endika, Selas, Asier, Rubiales, Gloria, Tesauro, Cinzia, Knudssen, Birgitta K., Palacios, Francisco
Published in European journal of medicinal chemistry (10.04.2018)
Published in European journal of medicinal chemistry (10.04.2018)
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Journal Article
Fused chromeno and quinolino[1,8]naphthyridines: Synthesis and biological evaluation as topoisomerase I inhibitors and antiproliferative agents
Martín-Encinas, Endika, Rubiales, Gloria, Knudsen, Birgitta R., Palacios, Francisco, Alonso, Concepción
Published in Bioorganic & medicinal chemistry (15.06.2021)
Published in Bioorganic & medicinal chemistry (15.06.2021)
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Journal Article
Synthesis of novel hybrid quinolino[4,3-b][1,5]naphthyridines and quinolino[4,3-b][1,5]naphthyridin-6(5H)-one derivatives and biological evaluation as topoisomerase I inhibitors and antiproliferatives
Martín-Encinas, Endika, Selas, Asier, Tesauro, Cinzia, Rubiales, Gloria, Knudsen, Birgitta R., Palacios, Francisco, Alonso, Concepción
Published in European journal of medicinal chemistry (01.06.2020)
Published in European journal of medicinal chemistry (01.06.2020)
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Journal Article
Synthesis of novel antiproliferative hybrid bis-(3-indolyl)methane phosphonate derivatives
Maestro, Aitor, Martín-Encinas, Endika, Alonso, Concepción, Martinez de Marigorta, Edorta, Rubiales, Gloria, Vicario, Javier, Palacios, Francisco
Published in European journal of medicinal chemistry (05.10.2018)
Published in European journal of medicinal chemistry (05.10.2018)
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Journal Article
Hydrogen sulphide-triggered theranostic prodrugs based on the dynamic chemistry of tetrazines
Perretti, Marcelle D, Pérez-Pérez, Yaiza, Soler-Carracedo, Kevin, Martín-Encinas, Endika, Alonso, Concepción, Scoccia, Jimena, Carrillo, Romen
Published in Chemical communications (Cambridge, England) (03.05.2022)
Published in Chemical communications (Cambridge, England) (03.05.2022)
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Journal Article
Fused 1,5-Naphthyridines: Synthetic Tools and Applications
Masdeu, Carme, Fuertes, Maria, Martin-Encinas, Endika, Selas, Asier, Rubiales, Gloria, Palacios, Francisco, Alonso, Concepcion
Published in Molecules (Basel, Switzerland) (31.07.2020)
Published in Molecules (Basel, Switzerland) (31.07.2020)
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Journal Article
Novel phosphine sulphide gold() complexes: topoisomerase I inhibitors and antiproliferative agents
Martín-Encinas, Endika, Conejo-Rodríguez, Verónica, Miguel, Jesús A, Martínez-Ilarduya, Jesús M, Rubiales, Gloria, Knudsen, Birgitta R, Palacios, Francisco, Alonso, Concepción
Published in Dalton transactions : an international journal of inorganic chemistry (21.06.2020)
Published in Dalton transactions : an international journal of inorganic chemistry (21.06.2020)
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Journal Article
A Dual-Sensor-Based Screening System for In Vitro Selection of TDP1 Inhibitors
Jakobsen, Ann-Katrine, Keller, Josephine Geertsen, Gonzalez, María, Martin-Encinas, Endika, Palacios, Francisco, Alonso, Concepcion, Knudsen, Birgitta Ruth, Stougaard, Magnus
Published in Sensors (Basel, Switzerland) (15.07.2021)
Published in Sensors (Basel, Switzerland) (15.07.2021)
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Journal Article
Straightforward synthesis and biological evaluation as topoisomerase I inhibitors and antiproliferative agents of hybrid Chromeno[4,3-b][1,5]Naphthyridines and Chromeno[4,3-b][1,5]Naphthyridin-6-ones
Martín-Encinas, Endika, Rubiales, Gloria, Knudssen, Birgitta R., Palacios, Francisco, Alonso, Concepción
Published in European journal of medicinal chemistry (15.09.2019)
Published in European journal of medicinal chemistry (15.09.2019)
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Journal Article
Naphthyridine Derivatives Induce Programmed Cell Death in Naegleria fowleri
Rizo-Liendo, Aitor, Arberas-Jiménez, Iñigo, Martin-Encinas, Endika, Sifaoui, Ines, Reyes-Batlle, María, Chao-Pellicer, Javier, Alonso, Concepción, Palacios, Francisco, Piñero, José E., Lorenzo-Morales, Jacob
Published in Pharmaceuticals (Basel, Switzerland) (01.10.2021)
Published in Pharmaceuticals (Basel, Switzerland) (01.10.2021)
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Journal Article
Kanptotezina eta haren deribatuak minbiziaren aurkako borrokan: Topoisomerasa I inhibitzaileak
Lopez-Aguileta, Leyre, Alonso, Concepción, Palacios, Francisco, Selas, Asier, Martín-Encinas, Endika
Published in EKAIA Euskal Herriko Unibertsitateko Zientzia eta Teknologia Aldizkaria (24.11.2022)
Published in EKAIA Euskal Herriko Unibertsitateko Zientzia eta Teknologia Aldizkaria (24.11.2022)
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