Synthesis and Profiling of a Diverse Collection of Azetidine-Based Scaffolds for the Development of CNS-Focused Lead-like Libraries
Lowe, Jason T, Lee, Maurice D, Akella, Lakshmi B, Davoine, Emeline, Donckele, Etienne J, Durak, Landon, Duvall, Jeremy R, Gerard, Baudouin, Holson, Edward B, Joliton, Adrien, Kesavan, Sarathy, Lemercier, Berenice C, Liu, Haibo, Marié, Jean-Charles, Mulrooney, Carol A, Muncipinto, Giovanni, Welzel-O’Shea, Morgan, Panko, Laura M, Rowley, Ann, Suh, Byung-Chul, Thomas, Meryl, Wagner, Florence F, Wei, Jingqiang, Foley, Michael A, Marcaurelle, Lisa A
Published in Journal of organic chemistry (07.09.2012)
Published in Journal of organic chemistry (07.09.2012)
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An Aldol-Based Build/Couple/Pair Strategy for the Synthesis of Medium- and Large-Sized Rings: Discovery of Macrocyclic Histone Deacetylase Inhibitors
Marcaurelle, Lisa A, Comer, Eamon, Dandapani, Sivaraman, Duvall, Jeremy R, Gerard, Baudouin, Kesavan, Sarathy, Lee, Maurice D, Liu, Haibo, Lowe, Jason T, Marie, Jean-Charles, Mulrooney, Carol A, Pandya, Bhaumik A, Rowley, Ann, Ryba, Troy D, Suh, Byung-Chul, Wei, Jingqiang, Young, Damian W, Akella, Lakshmi B, Ross, Nathan T, Zhang, Yan-Ling, Fass, Daniel M, Reis, Surya A, Zhao, Wen-Ning, Haggarty, Stephen J, Palmer, Michelle, Foley, Michael A
Published in Journal of the American Chemical Society (01.12.2010)
Published in Journal of the American Chemical Society (01.12.2010)
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Novel tricyclic glycal-based TRIB1 inducers that reprogram LDL metabolism in hepatic cells
Nagiec, Marek M, Duvall, Jeremy R, Skepner, Adam P, Howe, Eleanor A, Bastien, Jessica, Comer, Eamon, Marie, Jean-Charles, Johnston, Stephen E, Negri, Joseph, Eichhorn, Michelle, Vantourout, Julien, Clish, Clary, Musunuru, Kiran, Foley, Michael, Perez, Jose R, Palmer, Michelle A. J
Published in MedChemComm (01.11.2018)
Published in MedChemComm (01.11.2018)
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Accessing Skeletal Diversity Using Catalyst Control: Formation of n and n + 1 Macrocyclic Triazole Rings
Kelly, Ann Rowley, Wei, Jingqiang, Kesavan, Sarathy, Marié, Jean-Charles, Windmon, Nicole, Young, Damian W, Marcaurelle, Lisa A
Published in Organic letters (04.06.2009)
Published in Organic letters (04.06.2009)
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Enantioselective Synthesis of 3,4-Chromanediones via Asymmetric Rearrangement of 3-Allyloxyflavones
Marié, Jean-Charles, Xiong, Yuan, Min, Geanna K, Yeager, Adam R, Taniguchi, Tohru, Berova, Nina, Schaus, Scott E, Porco, John A
Published in Journal of organic chemistry (02.07.2010)
Published in Journal of organic chemistry (02.07.2010)
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Stereoselective access to tubuphenylalanine and tubuvaline: improved Mn-mediated radical additions and assembly of a tubulysin tetrapeptide analog
Friestad, Gregory K., Banerjee, Koushik, Marie, Jean -Charles, Mali, Umesh, Yao, Lei
Published in Journal of antibiotics (01.04.2016)
Published in Journal of antibiotics (01.04.2016)
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Synthesis of Stereochemically and Skeletally Diverse Fused Ring Systems from Functionalized C‑Glycosides
Gerard, Baudouin, Lee, Maurice D, Dandapani, Sivaraman, Duvall, Jeremy R, Fitzgerald, Mark E, Kesavan, Sarathy, Lowe, Jason T, Marié, Jean-Charles, Pandya, Bhaumik A, Suh, Byung-Chul, O’Shea, Morgan Welzel, Dombrowski, Michael, Hamann, Diane, Lemercier, Berenice, Murillo, Tiffanie, Akella, Lakshmi B, Foley, Michael A, Marcaurelle, Lisa A
Published in Journal of organic chemistry (07.06.2013)
Published in Journal of organic chemistry (07.06.2013)
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A computational model to investigate astrocytic glutamate uptake influence on synaptic transmission and neuronal spiking
Allam, Sushmita L, Ghaderi, Viviane S, Bouteiller, Jean-Marie C, Legendre, Arnaud, Ambert, Nicolas, Greget, Renaud, Bischoff, Serge, Baudry, Michel, Berger, Theodore W
Published in Frontiers in computational neuroscience (01.10.2012)
Published in Frontiers in computational neuroscience (01.10.2012)
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Identification of Highly Specific Diversity-Oriented Synthesis-Derived Inhibitors of Clostridium difficile
Duvall, Jeremy R, Bedard, Leanne, Naylor-Olsen, Adel M, Manson, Abigail L, Bittker, Joshua A, Sun, Wenye, Fitzgerald, Mark E, He, Zhenmin, Lee, Maurice D, Marie, Jean-Charles, Muncipinto, Giovanni, Rush, Diane, Xu, Deming, Xu, Huisheng, Zhang, Mingliang, Earl, Ashlee M, Palmer, Michelle A, Foley, Michael A, Vacca, Joseph P, Scherer, Christina A
Published in ACS infectious diseases (12.05.2017)
Published in ACS infectious diseases (12.05.2017)
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Diversity-Oriented Synthesis Yields a New Drug Lead for Treatment of Chagas Disease
Dandapani, Sivaraman, Germain, Andrew R, Jewett, Ivan, le Quement, Sebastian, Marie, Jean-Charles, Muncipinto, Giovanni, Duvall, Jeremy R, Carmody, Leigh C, Perez, Jose R, Engel, Juan C, Gut, Jiri, Kellar, Danielle, Siqueira-Neto, Jair Lage, McKerrow, James H, Kaiser, Marcel, Rodriguez, Ana, Palmer, Michelle A, Foley, Michael, Schreiber, Stuart L, Munoz, Benito
Published in ACS medicinal chemistry letters (13.02.2014)
Published in ACS medicinal chemistry letters (13.02.2014)
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Selective ring opening of silylated vinyloxiranes and reactivity of azido-alcohols
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Silylated Vinyloxiranes - Recent Advances and Synthetic Applications
Marion, Frédéric, Calvet, Sandrine, Marié, Jean-Charles, Courillon, Christine, Malacria, Max
Published in European Journal of Organic Chemistry (01.01.2006)
Published in European Journal of Organic Chemistry (01.01.2006)
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ChemInform Abstract: Enantioselective Synthesis of 3,4-Chromanediones via Asymmetric Rearrangement of 3-Allyloxyflavones
Marie, Jean-Charles, Xiong, Yuan, Min, Geanna K., Yeager, Adam R., Taniguchi, Tohru, Berova, Nina, Schaus, Scott E., Porco, John A. Jr
Published in ChemInform (09.11.2010)
Published in ChemInform (09.11.2010)
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