Search Results - "Margathe, Jean-Francois" :: K.UTB vyhledávací portál | TBU Library Retrieval Portal

Development of original metabolically stable apelin-17 analogs with diuretic and cardiovascular effects

Development of original metabolically stable apelin-17 analogs with diuretic and cardiovascular effects

by Gerbier, Romain, Alvear-Perez, Rodrigo, Margathe, Jean-Francois, Flahault, Adrien, Couvineau, Pierre, Gao, Ji, De Mota, Nadia, Dabire, Hubert, Li, Bo, Ceraudo, Emilie, Hus-Citharel, Annette, Esteoulle, Lucie, Bisoo, Cynthia, Hibert, Marcel, Berdeaux, Alain, Iturrioz, Xavier, Bonnet, Dominique, Llorens-Cortes, Catherine
Published in The FASEB journal (01.02.2017)

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Diastereoselective synthesis of novel aza-diketopiperazines via a domino cyclohydrocarbonylation/addition process

Diastereoselective synthesis of novel aza-diketopiperazines via a domino cyclohydrocarbonylation/addition process

by Regenass, Pierre, Margathe, Jean-Francois, Mann, Andre, Suffert, Jean, Hibert, Marcel, Girard, Nicolas, Bonnet, Dominique
Published in Chemical communications (Cambridge, England) (04.09.2014)

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Structure–Activity Relationship Studies toward the Discovery of Selective Apelin Receptor Agonists

Structure–Activity Relationship Studies toward the Discovery of Selective Apelin Receptor Agonists

by Margathe, Jean-François, Iturrioz, Xavier, Alvear-Perez, Rodrigo, Marsol, Claire, Riché, Stéphanie, Chabane, Hadjila, Tounsi, Nassera, Kuhry, Maxime, Heissler, Denis, Hibert, Marcel, Llorens-Cortes, Catherine, Bonnet, Dominique
Published in Journal of medicinal chemistry (10.04.2014)

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Selective Nonpeptidic Fluorescent Ligands for Oxytocin Receptor: Design, Synthesis, and Application to Time-Resolved FRET Binding Assay

Selective Nonpeptidic Fluorescent Ligands for Oxytocin Receptor: Design, Synthesis, and Application to Time-Resolved FRET Binding Assay

by Karpenko, Iuliia A, Margathe, Jean-François, Rodriguez, Thiéric, Pflimlin, Elsa, Dupuis, Elodie, Hibert, Marcel, Durroux, Thierry, Bonnet, Dominique
Published in Journal of medicinal chemistry (12.03.2015)

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Time-Resolved FRET Binding Assay to Investigate Hetero-Oligomer Binding Properties: Proof of Concept with Dopamine D1/D3 Heterodimer

Time-Resolved FRET Binding Assay to Investigate Hetero-Oligomer Binding Properties: Proof of Concept with Dopamine D1/D3 Heterodimer

by Hounsou, Candide, Margathe, Jean-François, Oueslati, Nadia, Belhocine, Abderazak, Dupuis, Elodie, Thomas, Cécile, Mann, André, Ilien, Brigitte, Rognan, Didier, Trinquet, Eric, Hibert, Marcel, Pin, Jean-Philippe, Bonnet, Dominique, Durroux, Thierry
Published in ACS chemical biology (20.02.2015)

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Convenient Access to Fluorescent Probes by Chemoselective Acylation of Hydrazinopeptides: Application to the Synthesis of the First Far-Red Ligand for Apelin Receptor Imaging

Convenient Access to Fluorescent Probes by Chemoselective Acylation of Hydrazinopeptides: Application to the Synthesis of the First Far-Red Ligand for Apelin Receptor Imaging

by Margathe, Jean-François, Iturrioz, Xavier, Regenass, Pierre, Karpenko, Iuliia A., Humbert, Nicolas, de Rocquigny, Hugues, Hibert, Marcel, Llorens-Cortes, Catherine, Bonnet, Dominique
Published in Chemistry : a European journal (22.01.2016)

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Chemoselective Acylation of Hydrazinopeptides to Access Fluorescent Probes for Time-Resolved FRET Assays on GPCRs

Chemoselective Acylation of Hydrazinopeptides to Access Fluorescent Probes for Time-Resolved FRET Assays on GPCRs

by Ramanoudjame, Sridévi M, Esteoulle, Lucie, Riché, Stéphanie, Margathe, Jean-François, Durroux, Thierry, Karpenko, Iuliia A, Bonnet, Dominique
Published in Methods in molecular biology (Clifton, N.J.) (2019)

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A Time‐Resolved FRET Cell‐Based Binding Assay for the Apelin Receptor

A Time‐Resolved FRET Cell‐Based Binding Assay for the Apelin Receptor

by Valencia, Christel, Dujet, Céline, Margathe, Jean‐François, Iturrioz, Xavier, Roux, Thomas, Trinquet, Eric, Villa, Pascal, Hibert, Marcel, Dupuis, Elodie, Llorens‐Cortes, Catherine, Bonnet, Dominique
Published in ChemMedChem (21.06.2017)

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Combinatorial Aid for Underprivileged Scaffolds: Solution and Solid-phase Strategies for a Rapid and Efficient Access To Novel Aza-diketopiperazines (Aza-DKP)

Combinatorial Aid for Underprivileged Scaffolds: Solution and Solid-phase Strategies for a Rapid and Efficient Access To Novel Aza-diketopiperazines (Aza-DKP)

by Bonnet, Dominique, Margathe, Jean-François, Radford, Sally, Pflimlin, Elsa, Riché, Stéphanie, Doman, Pete, Hibert, Marcel, Ganesan, A
Published in ACS combinatorial science (14.05.2012)

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융합된 바이사이클릭 RAF 억제제 및 이의 사용 방법

융합된 바이사이클릭 RAF 억제제 및 이의 사용 방법

by JONES CLIFFORD DAVID, MARGATHE JEAN FRANCOIS, BELFIELD ANDREW, COLLETTO CHIARA
Year of Publication 03.05.2023

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Patent

융합된 바이사이클릭 RAF 억제제의 키랄 합성

융합된 바이사이클릭 RAF 억제제의 키랄 합성

by JONES CLIFFORD DAVID, MARGATHE JEAN FRANCOIS, HAWKINS NEIL, GLOSSOP STEVEN CHRISTOPHER, BELFIELD ANDREW, COLLETTO CHIARA
Year of Publication 03.05.2023

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Patent

Solid-Phase, Multicomponent Reactions of Methyleneaziridines: Synthesis of 1,3-Disubstituted Propanones

Solid-Phase, Multicomponent Reactions of Methyleneaziridines: Synthesis of 1,3-Disubstituted Propanones

by Margathe, Jean-François, Shipman, Michael, Smith, Stephen C
Published in Organic letters (27.10.2005)

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ChemInform Abstract: Diastereoselective Synthesis of Novel Aza-Diketopiperazines via a Domino Cyclohydrocarbonylation/Addition Process

ChemInform Abstract: Diastereoselective Synthesis of Novel Aza-Diketopiperazines via a Domino Cyclohydrocarbonylation/Addition Process

by Regenass, Pierre, Margathe, Jean-Francois, Mann, Andre, Suffert, Jean, Hibert, Marcel, Girard, Nicolas, Bonnet, Dominique
Published in ChemInform (01.01.2015)

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Diastereoselective synthesis of novel aza-diketopiperazines viaa domino cyclohydrocarbonylation/addition process

Diastereoselective synthesis of novel aza-diketopiperazines viaa domino cyclohydrocarbonylation/addition process

by Regenass, Pierre, Margathe, Jean-Francois, Mann, Andre, Suffert, Jean, Hibert, Marcel, Girard, Nicolas, Bonnet, Dominique
Published in Chemical communications (Cambridge, England) (01.07.2014)

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FUSED BICYCLIC RAF INHIBITORS AND METHODS FOR USE THEREOF

FUSED BICYCLIC RAF INHIBITORS AND METHODS FOR USE THEREOF

by COLLETTO, CHIARA, JONES, CLIFFORD DAVID, BELFIELD, ANDREW, MARGATHE, JEAN-FRANCOIS
Year of Publication 03.02.2022

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Patent

CHIRAL SYNTHESIS OF FUSED BICYCLIC RAF INHIBITORS

CHIRAL SYNTHESIS OF FUSED BICYCLIC RAF INHIBITORS

by COLLETTO, CHIARA, HAWKINS, NEIL, JONES, CLIFFORD DAVID, BELFIELD, ANDREW, GLOSSOP, STEVEN CHRISTOPHER, MARGATHE, JEAN-FRANCOIS
Year of Publication 03.02.2022

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Patent

Time-Resolved FRET Binding Assay to Investigate Hetero-Oligomer Binding Properties: Proof of Concept with Dopamine D 1 /D 3 Heterodimer

Time-Resolved FRET Binding Assay to Investigate Hetero-Oligomer Binding Properties: Proof of Concept with Dopamine D 1 /D 3 Heterodimer

by Hounsou, Candide, Margathe, Jean-François, Oueslati, Nadia, Belhocine, Abderazak, Dupuis, Elodie, Thomas, Cécile, Mann, André, Ilien, Brigitte, Rognan, Didier, Trinquet, Eric, Hibert, Marcel, Pin, Jean-Philippe, Bonnet, Dominique, Durroux, Thierry
Published in ACS chemical biology (20.02.2015)

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Journal Article

COMPOUNDS USEFUL AS CSF1 MODULATORS

COMPOUNDS USEFUL AS CSF1 MODULATORS

by MORRISON, ANGUS, BELFIELD, ANDREW, AVERY, CRAIG, MARGATHE, JEAN-FRANCOIS, JOHNSON, ALICE, BINGHAM, MATILDA, ARMER, RICHARD, HUGHES, SHAUN
Year of Publication 07.04.2016

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Patent

FUSED BICYCLIC RAF INHIBITORS AND METHODS FOR USE THEREOF

FUSED BICYCLIC RAF INHIBITORS AND METHODS FOR USE THEREOF

by Jones, Clifford David, BELFIELD, Andrew, Margathe, Jean-François, Colletto, Chiara
Year of Publication 18.04.2024

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Patent

Fused bicyclic RAF inhibitors and methods for use thereof

Fused bicyclic RAF inhibitors and methods for use thereof

by Jones, Clifford David, Belfield, Andrew, Margathe, Jean-François, Colletto, Chiara
Year of Publication 02.01.2024

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Patent