Discovery of a Potent, Selective, and Orally Active Human Epidermal Growth Factor Receptor-2 Sheddase Inhibitor for the Treatment of Cancer
Yao, Wenqing, Zhuo, Jincong, Burns, David M, Xu, Meizhong, Zhang, Colin, Li, Yun-Long, Qian, Ding-Quan, He, Chunhong, Weng, Lingkai, Shi, Eric, Lin, Qiyan, Agrios, Costas, Burn, Timothy C, Caulder, Eian, Covington, Maryanne B, Fridman, Jordan S, Friedman, Steven, Katiyar, Kamna, Hollis, Gregory, Li, Yanlong, Liu, Changnian, Liu, Xiangdong, Marando, Cindy A, Newton, Robert, Pan, Max, Scherle, Peggy, Taylor, Nancy, Vaddi, Kris, Wasserman, Zelda R, Wynn, Richard, Yeleswaram, Swamy, Jalluri, Ravi, Bower, Michael, Zhou, Bing-Bing, Metcalf, Brian
Published in Journal of medicinal chemistry (22.02.2007)
Published in Journal of medicinal chemistry (22.02.2007)
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Conversion of an MMP-potent scaffold to an MMP-selective HER-2 sheddase inhibitor via scaffold hybridization and subtle P'1 permutations
BURNS, David M, CHUNHONG HE, FRIDMAN, Jordan S, HOLLIS, Gregory, VADDI, Kris, YELESWARAM, Swamy, NEWTON, Robert, FRIEDMAN, Steve, METCALF, Brian, WENQING YAO, YANLONG LI, SCHERLE, Peggy, XIANGDONG LIU, MARANDO, Cindy A, COVINGTON, Mayanne B, GENGJIE YANG, PAN, Max, TURNER, Sharon
Published in Bioorganic & medicinal chemistry letters (15.01.2008)
Published in Bioorganic & medicinal chemistry letters (15.01.2008)
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Compelling P1 substituent affect on metalloprotease binding profile enables the design of a novel cyclohexyl core scaffold with excellent MMP selectivity and HER-2 sheddase inhibition
Burns, David M., Li, Yun-Long, Shi, Eric, He, Chunhong, Xu, Meizhong, Zhuo, Jincong, Zhang, Colin, Qian, Ding-Quan, Li, Yanlong, Wynn, Richard, Covington, Maryanne B., Katiyar, Kamna, Marando, Cindy A., Fridman, Jordan S., Scherle, Peggy, Friedman, Steve, Metcalf, Brian, Yao, Wenqing
Published in Bioorganic & medicinal chemistry letters (01.07.2009)
Published in Bioorganic & medicinal chemistry letters (01.07.2009)
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Design and identification of selective HER-2 sheddase inhibitors via P1′ manipulation and unconventional P2′ perturbations to induce a molecular metamorphosis
Yao, Wenqing, Zhuo, Jincong, Burns, David M., Li, Yun-Long, Qian, Ding-Quan, Zhang, Colin, He, Chunhong, Xu, Meizhong, Shi, Eric, Li, Yanlong, Marando, Cindy A., Covington, Maryanne B., Yang, Gengjie, Liu, Xiangdong, Pan, Max, Fridman, Jordan S., Scherle, Peggy, Wasserman, Zelda R., Hollis, Gregory, Vaddi, Kris, Yeleswaram, Swamy, Newton, Robert, Friedman, Steve, Metcalf, Brian
Published in Bioorganic & medicinal chemistry (2008)
Published in Bioorganic & medicinal chemistry (2008)
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Journal Article
Conversion of an MMP-potent scaffold to an MMP-selective HER-2 sheddase inhibitor via scaffold hybridization and subtle permutations
Burns, David M., He, Chunhong, Li, Yanlong, Scherle, Peggy, Liu, Xiangdong, Marando, Cindy A., Covington, Mayanne B., Yang, Gengjie, Pan, Max, Turner, Sharon, Fridman, Jordan S., Hollis, Gregory, Vaddi, Kris, Yeleswaram, Swamy, Newton, Robert, Friedman, Steve, Metcalf, Brian, Yao, Wenqing
Published in Bioorganic & medicinal chemistry (01.01.2008)
Published in Bioorganic & medicinal chemistry (01.01.2008)
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Journal Article
Liver transplantation as definitive treatment for a factor V Leiden mutation
Dunn, Stephen P., Tsai, Anthony, Griffin, Gregory, Toth, Stephen, Casas-Melley, Adela T., Falkenstein, Kathleen P., Marando, Cindy A., Krueger, Leslie J.
Published in The Journal of pediatrics (01.03.2005)
Published in The Journal of pediatrics (01.03.2005)
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Conversion of an MMP-potent scaffold to an MMP-selective HER-2 sheddase inhibitor via scaffold hybridization and subtle P 1 ′ permutations
Burns, David M., He, Chunhong, Li, Yanlong, Scherle, Peggy, Liu, Xiangdong, Marando, Cindy A., Covington, Mayanne B., Yang, Gengjie, Pan, Max, Turner, Sharon, Fridman, Jordan S., Hollis, Gregory, Vaddi, Kris, Yeleswaram, Swamy, Newton, Robert, Friedman, Steve, Metcalf, Brian, Yao, Wenqing
Published in Bioorganic & medicinal chemistry letters (15.01.2008)
Published in Bioorganic & medicinal chemistry letters (15.01.2008)
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Corrigendum to “Compelling P1 substituent affect on metalloprotease binding profile enables the design of a novel cyclohexyl core scaffold with excellent MMP selectivity and HER-2 sheddase inhibition” [Bioorg. Med. Chem. Lett. 19 (2009) 3525]
Burns, David M., Li, Yun-Long, Xu, Meizhong, Shi, Eric, He, Chunhong, Zhuo, Jincong, Zhang, Colin, Qian, Ding-Quan, Li, Yanlong, Wynn, Richard, Covington, Maryanne B., Katiyar, Kamna, Marando, Cindy A., Fridman, Jordan S., Scherle, Peggy, Friedman, Steve, Metcalf, Brian, Yao, Wenqing
Published in Bioorganic & medicinal chemistry letters (01.10.2009)
Published in Bioorganic & medicinal chemistry letters (01.10.2009)
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Journal Article
Liver transplantation as definitive treatment for A factory V Leiden mutation
DUNN, Stephen P, TSAI, Anthony, GRIFFIN, Gregory, TOTH, Stephen, CASAS-MELLEY, Adela T, FALKENSTEIN, Kathleen P, MARANDO, Cindy A, KRUEGER, Leslie J
Published in The Journal of pediatrics (2005)
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Published in The Journal of pediatrics (2005)
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