Discovery and structure–activity study of a novel benzoxaborole anti-inflammatory agent (AN2728) for the potential topical treatment of psoriasis and atopic dermatitis
Akama, Tsutomu, Baker, Stephen J., Zhang, Yong-Kang, Hernandez, Vincent, Zhou, Huchen, Sanders, Virginia, Freund, Yvonne, Kimura, Richard, Maples, Kirk R., Plattner, Jacob J.
Published in Bioorganic & medicinal chemistry letters (15.04.2009)
Published in Bioorganic & medicinal chemistry letters (15.04.2009)
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Journal Article
Boron-based phosphodiesterase inhibitors show novel binding of boron to PDE4 bimetal center
Freund, Yvonne R., Akama, Tsutomu, Alley, M.R.K., Antunes, Joana, Dong, Chen, Jarnagin, Kurt, Kimura, Richard, Nieman, James A., Maples, Kirk R., Plattner, Jacob J., Rock, Fernando, Sharma, Rashmi, Singh, Rajeshwar, Sanders, Virginia, Zhou, Yasheen
Published in FEBS letters (21.09.2012)
Published in FEBS letters (21.09.2012)
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Journal Article
Translational research involving oxidative stress and diseases of aging
Floyd, Robert A., Towner, Rheal A., He, Ting, Hensley, Kenneth, Maples, Kirk R.
Published in Free radical biology & medicine (01.09.2011)
Published in Free radical biology & medicine (01.09.2011)
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Journal Article
Identification of a novel boron-containing antibacterial agent (AN0128) with anti-inflammatory activity, for the potential treatment of cutaneous diseases
Baker, Stephen J., Akama, Tsutomu, Zhang, Yong-Kang, Sauro, Vittorio, Pandit, Chetan, Singh, Rajeshwar, Kully, Maureen, Khan, Jehangir, Plattner, Jacob J., Benkovic, Stephen J., Lee, Ving, Maples, Kirk R.
Published in Bioorganic & medicinal chemistry letters (01.12.2006)
Published in Bioorganic & medicinal chemistry letters (01.12.2006)
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Journal Article
Novel Semisynthetic Derivative of Antibiotic Eremomycin Active against Drug-Resistant Gram-Positive Pathogens Including Bacillus anthracis
Maples, Kirk R, Wheeler, Conrad, Ip, Emily, Plattner, Jacob J, Chu, Daniel, Zhang, Yong-Kang, Preobrazhenskaya, Maria N, Printsevskaya, Svetlana S, Solovieva, Svetlana E, Olsufyeva, Evgenia N, Heine, Henry, Lovchik, Julie, Lyons, C. Richard
Published in Journal of medicinal chemistry (26.07.2007)
Published in Journal of medicinal chemistry (26.07.2007)
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Journal Article
NXY-059 maintains Akt activation and inhibits release of cytochrome C after focal cerebral ischemia
Yoshimoto, Tetsuyuki, Kanakaraj, Palanisamy, Ying Ma, Jing, Cheng, Mingshan, Kerr, Irene, Malaiyandi, Latha, Watson, Jenny A, Siesjö, Bo K, Maples, Kirk R
Published in Brain research (30.08.2002)
Published in Brain research (30.08.2002)
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Journal Article
BORON-CONTAINING SMALL MOLECULE
HERNANDEZ VINCENT S, PLATTNER JACOB J, AKAMA TSUTOMU, LEYDEN JAMES J, ZHANG YONG-KANG, SANDERS VIRGINIA, MAPLES KIRK R, BAKER STEPHEN J, BELLINGER-KAWAHARA CAROLYN, HOLD KARIN M
Year of Publication 15.06.2017
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Year of Publication 15.06.2017
Patent
BORON-CONTAINING SMALL MOLECULE
HERNANDEZ VINCENT S, PLATTNER JACOB J, AKAMA TSUTOMU, LEYDEN JAMES J, ZHANG YONG-KANG, SANDERS VIRGINIA, MAPLES KIRK R, BAKER STEPHEN J, BELLINGER-KAWAHARA CAROLYN, HOLD KARIN M
Year of Publication 04.02.2016
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Year of Publication 04.02.2016
Patent
BORON-CONTAINING SMALL MOLECULES AS ANTI-INFLAMMATORY AGENTS
AKAMA TSUTOMU, SANDERS VIRGINIA, MAPLES KIRK R, MARCELO SALES, MICHAEL RICHARD KEVIN ALLEY, RAJESHWAR SINGH, CHARLES Z DING, JAMES A NIEMANN, PLATTNER JACOB J, XIA YI, ZHANG YONG-KANG, CHEN DAITAO, FREUND YVONNE, STEPHEN J BAKER, RASHMI SHARMA, XIAOSONG LU, ROBERT JACOBS
Year of Publication 09.03.2017
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Year of Publication 09.03.2017
Patent
BORON-CONTAINING SMALL MOLECULES
STEPHEN J BENKOVIC, AKAMA TSUTOMU, MICHAEL DIPIERRO, AARON M STEMPHOSKI, MAO WEIMIN, SANDERS VIRGINIA, KARIN M HOLD, MAPLES KIRK R, MICHAEL RICHARD KEVIN ALLEY, FERNANDO ROCK, VINCENT S HERNANDEZ, PLATTNER JACOB J, ISAAC KENNEDY, GEORGE PETROS YIANNIKOUROS, ZHOU HUCHEN, ZHANG YONG-KANG, SIEAD ZEGAR, STEPHEN J BAKER, IGOR LIKHOTVORIK
Year of Publication 01.12.2016
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Year of Publication 01.12.2016
Patent