Discovery of a series of potent and selective human H4 antagonists using ligand efficiency and libraries to explore structure–activity relationship (SAR)
Masood, M. Abid, Selby, Matthew D., Bell, Andrew S., Mansfield, Andrew C., Gardner, Mark, Smith, Graham F., Lane, Charlotte, Kenyon-Edwards, Helen, Osborne, Rachel, Jones, Rhys M., Liu, Wai L., Brown, Christopher D., Clarke, Nicholas, Perrucio, Francesca, Mowbray, Charles E.
Published in Bioorganic & medicinal chemistry letters (01.11.2011)
Published in Bioorganic & medicinal chemistry letters (01.11.2011)
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[3+2] Dipolar cycloadditions of an unstabilised azomethine ylide under continuous flow conditions
Grafton, Mark, Mansfield, Andrew C., Fray, M. Jonathan
Published in Tetrahedron letters (17.02.2010)
Published in Tetrahedron letters (17.02.2010)
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2-heteroaryl and 2-heterocyclic benzoxazoles as PDE IV inhibitors for the treatment of asthma
WHITEHEAD; JOHN W F, MANSFIELD; ANDREW C, CHASIN; MARK, CAVALLA; DAVID J, WALTON; LESLEY
Year of Publication 26.12.2000
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Year of Publication 26.12.2000
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