Antagonists of the human A2A receptor. Part 5: Highly bio-available pyrimidine-4-carboxamides
GILLESPIE, Roger J, BAMFORD, Samantha J, GAUR, Suneel, JORDAN, Allan M, LERPINIERE, Joanne, MANSELL, Howard L, STRATTON, Gemma C
Published in Bioorganic & medicinal chemistry letters (01.05.2009)
Published in Bioorganic & medicinal chemistry letters (01.05.2009)
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Antagonists of the human A(2A) receptor. Part 5: Highly bio-available pyrimidine-4-carboxamides
Gillespie, Roger J, Bamford, Samantha J, Gaur, Suneel, Jordan, Allan M, Lerpiniere, Joanne, Mansell, Howard L, Stratton, Gemma C
Published in Bioorganic & medicinal chemistry letters (15.05.2009)
Published in Bioorganic & medicinal chemistry letters (15.05.2009)
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Antagonists of the human A2A receptor. Part 6: Further optimization of pyrimidine-4-carboxamides
GILLESPIE, Roger J, BAMFORD, Samantha J, MANSELL, Howard L, NG, Sean, SAADI, Mona, SIMMONITE, Heather, STRATTON, Gemma C, TODD, Richard S, WILLIAMSON, Douglas S, YULE, Ian A, CLAY, Alex, GAUR, Suneel, HAYMES, Tim, JACKSON, Philip S, JORDAN, Allan M, KLENKE, Burlchard, LEONARDI, Stefania, LIU, Jeanette
Published in Bioorganic & medicinal chemistry (15.09.2009)
Published in Bioorganic & medicinal chemistry (15.09.2009)
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Journal Article
Antagonists of the human A(2A) receptor. Part 6: Further optimization of pyrimidine-4-carboxamides
Gillespie, Roger J, Bamford, Samantha J, Clay, Alex, Gaur, Suneel, Haymes, Tim, Jackson, Philip S, Jordan, Allan M, Klenke, Burkhard, Leonardi, Stefania, Liu, Jeanette, Mansell, Howard L, Ng, Sean, Saadi, Mona, Simmonite, Heather, Stratton, Gemma C, Todd, Richard S, Williamson, Douglas S, Yule, Ian A
Published in Bioorganic & medicinal chemistry (15.09.2009)
Published in Bioorganic & medicinal chemistry (15.09.2009)
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Pyrrolo(iso)quinoline derivatives as 5-HT2C receptor agonists
ADAMS, David R, BENTLEY, Jonathan M, MALCOLM, Craig S, MANSELL, Howard L, MISRA, Anil, QUIRK, Kathleen, ROFFEY, Jonathan R. A, VICKERS, Steven P, BENWELL, Karen R, BICKERDIKE, Michael J, BODKIN, Corinna D, CLIFFE, Ian A, DOURISH, Colin T, GEORGE, Ashley R, KENNETT, Guy A, KNIGHT, Antony R
Published in Bioorganic & medicinal chemistry letters (01.02.2006)
Published in Bioorganic & medicinal chemistry letters (01.02.2006)
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WAY100135 : a novel, selective antagonist at presynaptic and postsynaptic 5-HT1A receptors
FLETCHER, A, BILL, D. J, BILL, S. J, CLIFFE, I. A, DOVER, G. M, FORSTER, E. A, HASKINS, J. T, JONES, D, MANSELL, H. L, REILLY, Y
Published in European journal of pharmacology (24.06.1993)
Published in European journal of pharmacology (24.06.1993)
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Targeting conserved water molecules: Design of 4-aryl-5-cyanopyrrolo[2,3-d]pyrimidine Hsp90 inhibitors using fragment-based screening and structure-based optimization
Davies, Nicholas G.M., Browne, Helen, Davis, Ben, Drysdale, Martin J., Foloppe, Nicolas, Geoffrey, Stephanie, Gibbons, Ben, Hart, Terance, Hubbard, Roderick, Jensen, Michael Rugaard, Mansell, Howard, Massey, Andrew, Matassova, Natalia, Moore, Jonathan D., Murray, James, Pratt, Robert, Ray, Stuart, Robertson, Alan, Roughley, Stephen D., Schoepfer, Joseph, Scriven, Kirsten, Simmonite, Heather, Stokes, Stephen, Surgenor, Allan, Webb, Paul, Wood, Mike, Wright, Lisa, Brough, Paul
Published in Bioorganic & medicinal chemistry (15.11.2012)
Published in Bioorganic & medicinal chemistry (15.11.2012)
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Fatty acid amide hydrolase inhibitors. Surprising selectivity of chiral azetidine ureas
Hart, Terance, Macias, Alba T., Benwell, Karen, Brooks, Teresa, D’Alessandro, Jalanie, Dokurno, Pawel, Francis, Geraint, Gibbons, Ben, Haymes, Timothy, Kennett, Guy, Lightowler, Sean, Mansell, Howard, Matassova, Natalia, Misra, Anil, Padfield, Anthony, Parsons, Rachel, Pratt, Robert, Robertson, Alan, Walls, Steven, Wong, Melanie, Roughley, Stephen
Published in Bioorganic & medicinal chemistry letters (01.08.2009)
Published in Bioorganic & medicinal chemistry letters (01.08.2009)
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Fatty acid amide hydrolase inhibitors. 3: Tetra-substituted azetidine ureas with in vivo activity
Roughley, Stephen D., Browne, Helen, Macias, Alba T., Benwell, Karen, Brooks, Teresa, D’Alessandro, Jalanie, Daniels, Zoe, Dugdale, Sarah, Francis, Geraint, Gibbons, Ben, Hart, Terance, Haymes, Timothy, Kennett, Guy, Lightowler, Sean, Matassova, Natalia, Mansell, Howard, Merrett, Angela, Misra, Anil, Padfield, Anthony, Parsons, Rachel, Pratt, Robert, Robertson, Alan, Simmonite, Heather, Tan, Kiri, Walls, Steven B., Wong, Melanie
Published in Bioorganic & medicinal chemistry letters (15.01.2012)
Published in Bioorganic & medicinal chemistry letters (15.01.2012)
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Oral hypoglycemic agents. Pyrimido[1,2-a]indoles and related compounds
Cliffe, Ian A, Lien, Eric L, Mansell, Howard L, Steiner, Kurt E, Todd, Richard S, White, Alan C, Black, Robin M
Published in Journal of medicinal chemistry (01.04.1992)
Published in Journal of medicinal chemistry (01.04.1992)
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(S)-N-tert-Butyl-3-(4-(2-methoxyphenyl)piperazin-1-yl)-2-phenylpropanamide [(S)-WAY-100135]: a selective antagonist at presynaptic and postsynaptic 5-HT1A receptors
Cliffe, Ian A, Brightwell, Christopher I, Fletcher, Allan, Forster, Elaine A, Mansell, Howard L, Reilly, Yvonne, Routledge, Carol, White, Alan C
Published in Journal of medicinal chemistry (01.05.1993)
Published in Journal of medicinal chemistry (01.05.1993)
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Journal Article
Antagonists of the human A 2A receptor. Part 5: Highly bio-available pyrimidine-4-carboxamides
Gillespie, Roger J., Bamford, Samantha J., Gaur, Suneel, Jordan, Allan M., Lerpiniere, Joanne, Mansell, Howard L., Stratton, Gemma C.
Published in Bioorganic & medicinal chemistry letters (2009)
Published in Bioorganic & medicinal chemistry letters (2009)
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Journal Article
Antagonists of the human A sub(2A) receptor. Part 6: Further optimization of pyrimidine-4-carboxamides
Gillespie, Roger J, Bamford, Samantha J, Clay, Alex, Gaur, Suneel, Haymes, Tim, Jackson, Philip S, Jordan, Allan M, Klenke, Burkhard, Leonardi, Stefania, Liu, Jeanette, Mansell, Howard L, Ng, Sean, Saadi, Mona, Simmonite, Heather, Stratton, Gemma C, Todd, Richard S, Williamson, Douglas S, Yule, Ian A
Published in Bioorganic & medicinal chemistry (01.09.2009)
Published in Bioorganic & medicinal chemistry (01.09.2009)
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Journal Article
Antagonists of the human A 2A receptor. Part 6: Further optimization of pyrimidine-4-carboxamides
Gillespie, Roger J., Bamford, Samantha J., Clay, Alex, Gaur, Suneel, Haymes, Tim, Jackson, Philip S., Jordan, Allan M., Klenke, Burkhard, Leonardi, Stefania, Liu, Jeanette, Mansell, Howard L., Ng, Sean, Saadi, Mona, Simmonite, Heather, Stratton, Gemma C., Todd, Richard S., Williamson, Douglas S., Yule, Ian A.
Published in Bioorganic & medicinal chemistry (2009)
Published in Bioorganic & medicinal chemistry (2009)
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Journal Article
Pyrrolo(iso)quinoline derivatives as 5-HT(2C) receptor agonists
Adams, David R, Bentley, Jonathan M, Benwell, Karen R, Bickerdike, Michael J, Bodkin, Corinna D, Cliffe, Ian A, Dourish, Colin T, George, Ashley R, Kennett, Guy A, Knight, Antony R, Malcolm, Craig S, Mansell, Howard L, Misra, Anil, Quirk, Kathleen, Roffey, Jonathan R A, Vickers, Steven P
Published in Bioorganic & medicinal chemistry letters (01.02.2006)
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Published in Bioorganic & medicinal chemistry letters (01.02.2006)
Journal Article
Pyrrolo(iso)quinoline derivatives as 5-HT 2C receptor agonists
Adams, David R., Bentley, Jonathan M., Benwell, Karen R., Bickerdike, Michael J., Bodkin, Corinna D., Cliffe, Ian A., Dourish, Colin T., George, Ashley R., Kennett, Guy A., Knight, Antony R., Malcolm, Craig S., Mansell, Howard L., Misra, Anil, Quirk, Kathleen, Roffey, Jonathan R.A., Vickers, Steven P.
Published in Bioorganic & medicinal chemistry letters (2006)
Published in Bioorganic & medicinal chemistry letters (2006)
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Journal Article