Discovery of an MLLT1/3 YEATS Domain Chemical Probe
Moustakim, Moses, Christott, Thomas, Monteiro, Octovia P., Bennett, James, Giroud, Charline, Ward, Jennifer, Rogers, Catherine M., Smith, Paul, Panagakou, Ioanna, Díaz‐Sáez, Laura, Felce, Suet Ling, Gamble, Vicki, Gileadi, Carina, Halidi, Nadia, Heidenreich, David, Chaikuad, Apirat, Knapp, Stefan, Huber, Kilian V. M., Farnie, Gillian, Heer, Jag, Manevski, Nenad, Poda, Gennady, Al‐awar, Rima, Dixon, Darren J., Brennan, Paul E., Fedorov, Oleg
Published in Angewandte Chemie International Edition (10.12.2018)
Published in Angewandte Chemie International Edition (10.12.2018)
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Journal Article
Albumin stimulates the activity of the human UDP-glucuronosyltransferases 1A7, 1A8, 1A10, 2A1 and 2B15, but the effects are enzyme and substrate dependent
Manevski, Nenad, Troberg, Johanna, Svaluto-Moreolo, Paolo, Dziedzic, Klaudyna, Yli-Kauhaluoma, Jari, Finel, Moshe
Published in PloS one (23.01.2013)
Published in PloS one (23.01.2013)
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P38 - Exploring species differences in aldehyde oxidase activity
Shah, Pranav, Siramshetty, Vishal, Tawa, Gregory, Nguyen, Dac-Trung, Zakharov, Alexey, Southall, Noel, Isin, Emre M., Obach, R. Scott, Xu, Xin, Manevski, Nenad
Published in Drug metabolism and pharmacokinetics (2020)
Published in Drug metabolism and pharmacokinetics (2020)
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Journal Article
Aldehyde oxidase dependent metabolite profiling methodologies in early drug discovery projects
King, Lloyd M., Claessens, Jehan, Derwa, Christelle, Jones, Liz, Foley, Anne, Isin, Emre M., Manevski, Nenad, Mackenzie, Harold
Published in Drug metabolism and pharmacokinetics (01.01.2018)
Published in Drug metabolism and pharmacokinetics (01.01.2018)
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Journal Article
Glucocorticoids promote breast cancer metastasis
Obradović, Milan M S, Hamelin, Baptiste, Manevski, Nenad, Couto, Joana Pinto, Sethi, Atul, Coissieux, Marie-May, Münst, Simone, Okamoto, Ryoko, Kohler, Hubertus, Schmidt, Alexander, Bentires-Alj, Mohamed
Published in Nature (London) (01.03.2019)
Published in Nature (London) (01.03.2019)
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Evaluation of In Vitro Models for Assessment of Human Intestinal Metabolism in Drug Discovery
Davies, Mari, Peramuhendige, Prabha, King, Lloyd, Golding, Melanie, Kotian, Apoorva, Penney, Mark, Shah, Syeda, Manevski, Nenad
Published in Drug metabolism and disposition (01.11.2020)
Published in Drug metabolism and disposition (01.11.2020)
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Journal Article
Can We Predict Clinical Pharmacokinetics of Highly Lipophilic Compounds by Integration of Machine Learning or In Vitro Data into Physiologically Based Models? A Feasibility Study Based on 12 Development Compounds
Parrott, Neil, Manevski, Nenad, Olivares-Morales, Andrés
Published in Molecular pharmaceutics (07.11.2022)
Published in Molecular pharmaceutics (07.11.2022)
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Journal Article
Computational Predictions of Nonclinical Pharmacokinetics at the Drug Design Stage
Stoyanova, Raya, Katzberger, Paul Maximilian, Komissarov, Leonid, Khadhraoui, Aous, Sach-Peltason, Lisa, Groebke Zbinden, Katrin, Schindler, Torsten, Manevski, Nenad
Published in Journal of chemical information and modeling (23.01.2023)
Published in Journal of chemical information and modeling (23.01.2023)
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Journal Article
UDP-glucuronic acid binds first and the aglycone substrate binds second to form a ternary complex in UGT1A9-catalyzed reactions, in both the presence and absence of bovine serum albumin
Manevski, Nenad, Yli-Kauhaluoma, Jari, Finel, Moshe
Published in Drug metabolism and disposition (01.11.2012)
Published in Drug metabolism and disposition (01.11.2012)
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Journal Article
Functional assessment of rat pulmonary flavin-containing monooxygenase activity
Yilmaz, Yildiz, Williams, Gareth, Manevski, Nenad, Walles, Markus, Krähenbühl, Stephan, Camenisch, Gian
Published in Xenobiotica (04.05.2019)
Published in Xenobiotica (04.05.2019)
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Journal Article
Discovery of Orally Available and Brain Penetrant AEP Inhibitors
Krummenacher, Daniela, He, Weiping, Kuhn, Bernd, Schnider, Christian, Beurier, Angélica, Brom, Virginie, Sivasothy, Thulase, Marty, Christine, Tosstorff, Andreas, Hewings, David S., Mesch, Stefanie, Pinard, Emmanuel, Brändlin, Mathis, Hochstrasser, Remo, Westwood, Paul, Rothe, Judith, Kronenberger, Alexandra, Morandi, Federica, Gutbier, Simon, Schuler, Angelika, Heer, Dominik, Gloria, Ludivine Esteves, Joedicke, Lisa, Rudolph, Markus G., Müller, Lutz, Grüninger, Fiona, Baumann, Karlheinz, Kaniyappan, Senthilvelrajan, Manevski, Nenad, Bartels, Björn
Published in Journal of medicinal chemistry (28.12.2023)
Published in Journal of medicinal chemistry (28.12.2023)
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