AZD0284, a Potent, Selective, and Orally Bioavailable Inverse Agonist of Retinoic Acid Receptor-Related Orphan Receptor C2
Narjes, Frank, Llinas, Antonio, von Berg, Stefan, Jirholt, Johan, Lever, Sarah, Pehrson, Rikard, Collins, Mia, Malmberg, Anna, Svanberg, Petter, Xue, Yafeng, Olsson, Roine I, Malmberg, Jesper, Hughes, Glyn, Hossain, Nafizal, Grindebacke, Hanna, Leffler, Agnes, Krutrök, Nina, Bäck, Elisabeth, Ramnegård, Marie, Lepistö, Matti, Thunberg, Linda, Aagaard, Anna, McPheat, Jane, Hansson, Eva L, Chen, Rongfeng, Xiong, Yao, Hansson, Thomas G
Published in Journal of medicinal chemistry (23.09.2021)
Published in Journal of medicinal chemistry (23.09.2021)
Get full text
Journal Article
Discovery of the Oral Leukotriene C4 Synthase Inhibitor (1S,2S)‑2-({5-[(5-Chloro-2,4-difluorophenyl)(2-fluoro-2-methylpropyl)amino]-3-methoxypyrazin-2-yl}carbonyl)cyclopropanecarboxylic Acid (AZD9898) as a New Treatment for Asthma
Munck af Rosenschöld, Magnus, Johannesson, Petra, Nikitidis, Antonios, Tyrchan, Christian, Chang, Hui-Fang, Rönn, Robert, Chapman, Dave, Ullah, Victoria, Nikitidis, Grigorios, Glader, Pernilla, Käck, Helena, Bonn, Britta, Wågberg, Fredrik, Björkstrand, Eva, Andersson, Ulf, Swedin, Linda, Rohman, Mattias, Andreasson, Theresa, Bergström, Eva Lamm, Jiang, Fanyi, Zhou, Xiao-Hong, Lundqvist, Anders J, Malmberg, Anna, Ek, Margareta, Gordon, Euan, Pettersen, Anna, Ripa, Lena, Davis, Andrew M
Published in Journal of medicinal chemistry (12.09.2019)
Published in Journal of medicinal chemistry (12.09.2019)
Get full text
Journal Article