Discovery of a Clinical Stage Multi-Kinase Inhibitor Sodium (E)-2-{2-Methoxy-5-[(2′,4′,6′-trimethoxystyrylsulfonyl)methyl]phenylamino}acetate (ON 01910.Na): Synthesis, Structure–Activity Relationship, and Biological Activity
Reddy, M. V. Ramana, Venkatapuram, Padmavathi, Mallireddigari, Muralidhar R, Pallela, Venkat R, Cosenza, Stephen C, Robell, Kimberly A, Akula, Balaiah, Hoffman, Benjamin S, Reddy, E. Premkumar
Published in Journal of medicinal chemistry (22.09.2011)
Published in Journal of medicinal chemistry (22.09.2011)
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Design, synthesis, and biological evaluation of 1-(4-sulfamylphenyl)-3-trifluoromethyl-5-indolyl pyrazolines as cyclooxygenase-2 (COX-2) and lipoxygenase (LOX) inhibitors
Reddy, M.V. Ramana, Billa, Vinay K., Pallela, Venkat R., Mallireddigari, Muralidhar R., Boominathan, Rengasamy, Gabriel, Jerome L., Reddy, E. Premkumar
Published in Bioorganic & medicinal chemistry (01.04.2008)
Published in Bioorganic & medicinal chemistry (01.04.2008)
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Discovery of 8‑Cyclopentyl-2-[4-(4-methyl-piperazin-1-yl)-phenylamino]-7-oxo-7,8-dihydro-pyrido[2,3‑d]pyrimidine-6-carbonitrile (7x) as a Potent Inhibitor of Cyclin-Dependent Kinase 4 (CDK4) and AMPK-Related Kinase 5 (ARK5)
Reddy, M. V. Ramana, Akula, Balireddy, Cosenza, Stephen C, Athuluridivakar, Saikrishna, Mallireddigari, Muralidhar R, Pallela, Venkat R, Billa, Vinay K, Subbaiah, D. R. C. Venkata, Bharathi, E. Vijaya, Vasquez-Del Carpio, Rodrigo, Padgaonkar, Amol, Baker, Stacey J, Reddy, E. Premkumar
Published in Journal of medicinal chemistry (13.02.2014)
Published in Journal of medicinal chemistry (13.02.2014)
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(Z)-1-Aryl-3-arylamino-2-propen-1-ones, Highly Active Stimulators of Tubulin Polymerization: Synthesis, Structure–Activity Relationship (SAR), Tubulin Polymerization, and Cell Growth Inhibition Studies
Reddy, M. V. Ramana, Akula, Balaiah, Cosenza, Stephen C, Lee, Clement M, Mallireddigari, Muralidhar R, Pallela, Venkat R, Subbaiah, D. R. C. Venkata, Udofa, Andrew, Reddy, E. Premkumar
Published in Journal of medicinal chemistry (14.06.2012)
Published in Journal of medicinal chemistry (14.06.2012)
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Discovery of 2-(1H-indol-5-ylamino)-6-(2,4-difluorophenylsulfonyl)-8-methylpyrido[2,3-d]pyrimidin-7(8H)-one (7ao) as a potent selective inhibitor of Polo like kinase 2 (PLK2)
Reddy, M.V. Ramana, Akula, Balireddy, Jatiani, Shashidhar, Vasquez-Del Carpio, Rodrigo, Billa, Vinay K., Mallireddigari, Muralidhar R., Cosenza, Stephen C., Venkata Subbaiah, D.R.C., Bharathi, E. Vijaya, Pallela, Venkat R., Ramkumar, Poornima, Jain, Rinku, Aggarwal, Aneel K., Reddy, E. Premkumar
Published in Bioorganic & medicinal chemistry (15.02.2016)
Published in Bioorganic & medicinal chemistry (15.02.2016)
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Design, Synthesis, and Biological Evaluation of (E)‑N‑Aryl-2-arylethenesulfonamide Analogues as Potent and Orally Bioavailable Microtubule-Targeted Anticancer Agents
Reddy, M. V. Ramana, Mallireddigari, Muralidhar R, Pallela, Venkat R, Cosenza, Stephen C, Billa, Vinay K, Akula, Balaiah, Subbaiah, D. R. C. Venkata, Bharathi, E. Vijaya, Padgaonkar, Amol, Lv, Hua, Gallo, James M, Reddy, E. Premkumar
Published in Journal of medicinal chemistry (11.07.2013)
Published in Journal of medicinal chemistry (11.07.2013)
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Hydrothiolation of benzyl mercaptan to arylacetylene: application to the synthesis of (E) and (Z)-isomers of ON 01910·Na (Rigosertib®), a phase III clinical stage anti-cancer agent
Pallela, Venkat R, Mallireddigari, Muralidhar R, Cosenza, Stephen C, Akula, Balaiah, Subbaiah, D R C Venkata, Reddy, E Premkumar, Reddy, M V Ramana
Published in Organic & biomolecular chemistry (28.03.2013)
Published in Organic & biomolecular chemistry (28.03.2013)
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Design, Synthesis, and Biological Evaluation of (E)-Styrylbenzylsulfones as Novel Anticancer Agents
Reddy, M. V. Ramana, Mallireddigari, Muralidhar R, Cosenza, Stephen C, Pallela, Venkat R, Iqbal, Nabisa M, Robell, Kimberly A, Kang, Anthony D, Reddy, E. Premkumar
Published in Journal of medicinal chemistry (10.01.2008)
Published in Journal of medicinal chemistry (10.01.2008)
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Design, synthesis and evaluation of ( E)-α-benzylthio chalcones as novel inhibitors of BCR-ABL kinase
Reddy, M.V. Ramana, Pallela, Venkat R., Cosenza, Stephen C., Mallireddigari, Muralidhar R., Patti, Revathi, Bonagura, Marie, Truongcao, May, Akula, Balaiah, Jatiani, Shashidhar S., Reddy, E. Premkumar
Published in Bioorganic & medicinal chemistry (15.03.2010)
Published in Bioorganic & medicinal chemistry (15.03.2010)
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Novel coumarin-3-( N-aryl)carboxamides arrest breast cancer cell growth by inhibiting ErbB-2 and ERK1
Reddy, Natala Srinivasa, Gumireddy, Kiranmai, Mallireddigari, Muralidhar R., Cosenza, Stephen C., Venkatapuram, Padmavathi, Bell, Stanley C., Reddy, E. Premkumar, Reddy, M.V. Ramana
Published in Bioorganic & medicinal chemistry (02.05.2005)
Published in Bioorganic & medicinal chemistry (02.05.2005)
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Journal Article
Hydrothiolation of benzyl mercaptan to arylacetylene: application to the synthesis of (E) and (Z)-isomers of ON 01910 center dot Na (Rigosertib (R)), a phase III clinical stage anti-cancer agent
Pallela, Venkat R., Mallireddigari, Muralidhar R., Cosenza, Stephen C., Akula, Balaiah, Subbaiah, D. R. C. Venkata, Reddy, E. Premkumar, Reddy, M. V. Ramana
Published in Organic & biomolecular chemistry (01.01.2013)
Published in Organic & biomolecular chemistry (01.01.2013)
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Discovery of 2-(1H-indol-5-ylamino)-6-(2,4-difluorophenylsulfonyl)-8-methylpyri d o[2,3-d]pyrimidin-7(8H)-one (7ao) as a potent selective inhibitor of Polo like kinase 2 (PLK2)
Reddy, MVRamana, Akula, Balireddy, Jatiani, Shashidhar, Carpio, Rodrigo Vasquez-Del, Billa, Vinay K, Mallireddigari, Muralidhar R, Cosenza, Stephen C, Subbaiah, DRCVenkata, Bharathi, EVijaya, Pallela, Venkat R, Ramkumar, Poornima, Jain, Rinku, Aggarwal, Aneel K, Reddy, EPremkumar
Published in Bioorganic & medicinal chemistry (15.02.2016)
Published in Bioorganic & medicinal chemistry (15.02.2016)
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Design, Synthesis and Biological Evaluation of (E)-N-Aryl-2-arylethene-sulfonamide Analogues as Potent and Orally Bioavailable Microtubule-targeted Anticancer Agents
Ramana Reddy, M. V., Mallireddigari, Muralidhar R., Pallela, Venkat R., Cosenza, Stephen C., Billa, Vinay K., Akula, Balaiah, Venkata Subbaiah, D. R. C., Bharathi, E. Vijaya, Padgaonkar, Amol, Lv, Hua, Gallo, James M., Reddy, E. Premkumar
Published in Journal of medicinal chemistry (25.06.2013)
Published in Journal of medicinal chemistry (25.06.2013)
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Hydrothiolation of benzyl mercaptan to arylacetylene: application to the synthesis of (E) and (Z)-isomers of ON 01910·Na (Rigosertib®), a phase III clinical stage anti-cancer agentElectronic supplementary information (ESI) available: 1H and 13C NMR spectra of all new compounds. See DOI: 10.1039/c3ob27220f
Pallela, Venkat R, Mallireddigari, Muralidhar R, Cosenza, Stephen C, Akula, Balaiah, Subbaiah, D. R. C. Venkata, Reddy, E. Premkumar, Reddy, M. V. Ramana
Year of Publication 27.02.2013
Year of Publication 27.02.2013
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