Ligand Efficiency Driven Design of New Inhibitors of Mycobacterium tuberculosis Transcriptional Repressor EthR Using Fragment Growing, Merging, and Linking Approaches
Villemagne, Baptiste, Flipo, Marion, Blondiaux, Nicolas, Crauste, Céline, Malaquin, Sandra, Leroux, Florence, Piveteau, Catherine, Villeret, Vincent, Brodin, Priscille, Villoutreix, Bruno O, Sperandio, Olivier, Soror, Sameh H, Wohlkönig, Alexandre, Wintjens, René, Deprez, Benoit, Baulard, Alain R, Willand, Nicolas
Published in Journal of medicinal chemistry (12.06.2014)
Published in Journal of medicinal chemistry (12.06.2014)
Get full text
Journal Article
Synthesis of five- and six-membered lactams via solvent-free microwave Ugi reaction
Jida, Mouhamad, Malaquin, Sandra, Deprez-Poulain, Rebecca, Laconde, Guillaume, Deprez, Benoit
Published in Tetrahedron letters (29.09.2010)
Published in Tetrahedron letters (29.09.2010)
Get full text
Journal Article
Ugi reaction for the synthesis of 4-aminopiperidine-4-carboxylic acid derivatives. Application to the synthesis of carfentanil and remifentanil
Malaquin, Sandra, Jida, Mouhamad, Gesquiere, Jean-Claude, Deprez-Poulain, Rebecca, Deprez, Benoit, Laconde, Guillaume
Published in Tetrahedron letters (02.06.2010)
Published in Tetrahedron letters (02.06.2010)
Get full text
Journal Article
Solvent-free microwave-assisted Meyers' lactamization
JIDA, Mouhamad, DEPREZ-POULAIN, Rebecca, MALAQUIN, Sandra, ROUSSEL, Pascal, AGBOSSOU-NIEDERCORN, Francine, DEPREZ, Benoit, LACONDE, Guillaume
Published in Green chemistry : an international journal and green chemistry resource : GC (01.01.2010)
Published in Green chemistry : an international journal and green chemistry resource : GC (01.01.2010)
Get full text
Journal Article
Solvent-free microwave-assisted Meyers' lactamizationElectronic supplementary information (ESI) available: Compound characterization and NMR spectra. CCDC reference numbers 749287 and 749288. For ESI and crystallographic data in CIF or other electronic format see DOI: 10.1039/b924111f
Jida, Mouhamad, Deprez-Poulain, Rebecca, Malaquin, Sandra, Roussel, Pascal, Agbossou-Niedercorn, Francine, Deprez, Benoit, Laconde, Guillaume
Year of Publication 08.06.2010
Year of Publication 08.06.2010
Get full text
Journal Article