Enlarging the NSAIDs family: ether, ester and acid derivatives of the 1,5-diarylpyrrole scaffold as novel anti-inflammatory and analgesic agents
Biava, M, Porretta, G C, Poce, G, Battilocchio, C, Botta, M, Manetti, F, Rovini, M, Cappelli, A, Sautebin, L, Rossi, A, Pergola, C, Ghelardini, C, Galeotti, N, Makovec, F, Giordani, A, Anzellotti, P, Tacconelli, S, Patrignani, P, Anzini, M
Published in Current medicinal chemistry (01.04.2011)
Published in Current medicinal chemistry (01.04.2011)
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Pharmacokinetic study of a new angiotensin-AT1 antagonist by HPLC
RIZZO, M, VENTRICE, D, CASALE, F, CASELLI, G. F, MAKOVEC, F
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Published in Journal of pharmaceutical and biomedical analysis (29.09.2008)
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Development and validation of a bioanalytical method for the determination of the cholecystokinin type-1 (CCK 1) receptor antagonist dexloxiglumide in human plasma
Brodie, R, Peard, A, Roth, A, Persiani, S, Makovec, F, D’Amato, M
Published in Journal of chromatography. B, Analytical technologies in the biomedical and life sciences (25.01.2003)
Published in Journal of chromatography. B, Analytical technologies in the biomedical and life sciences (25.01.2003)
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Sensitive SPE-HPLC method to determine a novel angiotensin-AT1 antagonist in biological samples
RIZZO, M, VENTRICE, D, MONFORTE, F, PROCOPIO, S, DE SARRO, G, ANZINI, M, CAPPELLI, A, MAKOVEC, F
Published in Journal of pharmaceutical and biomedical analysis (16.04.2004)
Published in Journal of pharmaceutical and biomedical analysis (16.04.2004)
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Conference Proceeding
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N-terminal anthranoyl-phenylalanine derivatives as CCK1 receptor antagonists: the final approach
Varnavas, A, Lassiani, L, Valenta, V, Ciogli, A, Gasparrini, F, Mennuni, L, Makovec, F
Published in Medicinal chemistry (Shp-sariqah, United Arab Emirates) (01.09.2005)
Published in Medicinal chemistry (Shp-sariqah, United Arab Emirates) (01.09.2005)
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Pharmacokinetics and metabolism of the cholecystokinin antagonist dexloxiglumide in male human subjects
Webber, C., Roth, A., Persiani, S., Peard, A. J., Makovec, F., Kapil, R. P., John, B. A., Holding, J. D., D'amato, M., Cybulski, Z. R., Chasseaud, L. F., Rovati, L. C.
Published in Xenobiotica (01.06.2003)
Published in Xenobiotica (01.06.2003)
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Pharmacokinetics of dexloxiglumide after administration of single and repeat oral escalating doses in healthy young males
Persiani, S, D'Amato, M, Makovec, F, Tavares, I A, Bishai, P M, Rovati, L C
Published in International journal of clinical pharmacology and therapeutics (01.05.2002)
Published in International journal of clinical pharmacology and therapeutics (01.05.2002)
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Effect of three nonpeptide cholecystokinin antagonists on human isolated gallbladder
MASELLI, M. A, PIEPOLI, A. L, PEZZOLLA, F, GUERRA, V, CARUSO, M. L, MENNUNI, L, LORUSSO, D, MAKOVEC, F
Published in Digestive diseases and sciences (01.12.2001)
Published in Digestive diseases and sciences (01.12.2001)
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Absorption, distribution, metabolism and excretion of the cholecystokinin-1 antagonist dexloxiglumide in the dog
WEBBER, C, STOKES, C. A, PERSIANI, S, MAKOVEC, F, MCBURNEY, A, KAPIL, R. P, JOHN, B. A, D'AMATO, M, CHASSEAUD, L. F
Published in European journal of drug metabolism and pharmacokinetics (01.01.2004)
Published in European journal of drug metabolism and pharmacokinetics (01.01.2004)
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Determination of a novel angiotensin-AT1 antagonist CR 3210 in biological samples by HPLC
RIZZO, M, ANZINI, M, CAPPELLI, A, VOMERO, S, VENTRICE, D, DE SARRO, G, PROCOPIO, S, COSTA, N, MAKOVEC, F
Published in Farmaco (Società chimica italiana : 1989) (01.09.2003)
Published in Farmaco (Società chimica italiana : 1989) (01.09.2003)
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Absorption, distribution, metabolism and excretion of the cholecystokinin-1 antagonist dexloxiglumide in the rat
WEBBER, C, STOKES, C. A, PERSIANI, S, MAKOVEC, F, MCBURNEY, A, KAPIL, R. P, JOHN, B. A, HOUCHEN, T. L, D'AMATO, M, CHASSEAUD, L. F
Published in European journal of drug metabolism and pharmacokinetics (01.07.2003)
Published in European journal of drug metabolism and pharmacokinetics (01.07.2003)
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Protective effect of CR 1409 (cholecystokinin antagonist) on experimental pancreatitis in rats and mice
Makovec, F., Bani, M., Cereda, R., Chistè, R., Revel, L., Rovati, L.C., Setnikar, I., Rovati, L.A.
Published in Peptides (New York, N.Y. : 1980) (01.11.1986)
Published in Peptides (New York, N.Y. : 1980) (01.11.1986)
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Further studies on the interaction of the 5-hydroxytryptamine(3) (5-HT3) receptor with arylpiperazine ligands. Development of a new 5-HT3 receptor ligand showing potent acetylcholinesterase inhibitory properties
Cappelli, A, Gallelli, A, Manini, M, Anzini, M, Mennuni, L, Makovec, F, Menziani, MC, Alcaro, S, Ortuso, F, Vomero, S
Published in Journal of medicinal chemistry (19.05.2005)
Published in Journal of medicinal chemistry (19.05.2005)
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Discovery of new CCK2 receptor antagonists. A review of pharmacological studies. Part I: Development of potential therapeutic tools for gastrin-related gastrointestinal diseases
Revel, L, Makovec, F
Published in Methods and findings in experimental and clinical pharmacology (01.06.1999)
Published in Methods and findings in experimental and clinical pharmacology (01.06.1999)
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