Total Synthesis of Unsymmetrically Oxidized Nuphar Thioalkaloids via Copper-Catalyzed Thiolane Assembly
Lacharity, Jacob J, Fournier, Jeremy, Lu, Ping, Mailyan, Artur K, Herrmann, Aaron T, Zakarian, Armen
Published in Journal of the American Chemical Society (27.09.2017)
Published in Journal of the American Chemical Society (27.09.2017)
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Journal Article
Total Synthesis of (+)-Guadinomic Acid via Hydroxyl-Directed Guanidylation
Reid, Bradley T, Mailyan, Artur K, Zakarian, Armen
Published in Journal of organic chemistry (17.08.2018)
Published in Journal of organic chemistry (17.08.2018)
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Journal Article
Scalable Total Synthesis, IP3R Inhibitory Activity of Desmethylxestospongin B, and Effect on Mitochondrial Function and Cancer Cell Survival
Podunavac, Maša, Mailyan, Artur K., Jackson, Jeffrey J., Lovy, Alenka, Farias, Paula, Huerta, Hernan, Molgó, Jordi, Cardenas, Cesar, Zakarian, Armen
Published in Angewandte Chemie International Edition (10.05.2021)
Published in Angewandte Chemie International Edition (10.05.2021)
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Journal Article
Stereoselective Synthesis of Cyclic Guanidines by Directed Diamination of Unactivated Alkenes
Mailyan, Artur K, Young, Kyle, Chen, Joanna L, Reid, Bradley T, Zakarian, Armen
Published in Organic letters (04.11.2016)
Published in Organic letters (04.11.2016)
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Journal Article
Discovery of Potent and Selective PI3Kγ Inhibitors
Drew, Samuel L, Thomas-Tran, Rhiannon, Beatty, Joel W, Fournier, Jeremy, Lawson, Kenneth V, Miles, Dillon H, Mata, Guillaume, Sharif, Ehesan U, Yan, Xuelei, Mailyan, Artur K, Ginn, Elaine, Chen, Jie, Wong, Kent, Soni, Divyank, Dhanota, Puja, Chen, Pei-Yu, Shaqfeh, Stefan G, Meleza, Cesar, Pham, Amber T, Chen, Ada, Zhao, Xiaoning, Banuelos, Jesus, Jin, Lixia, Schindler, Ulrike, Walters, Matthew J, Young, Stephen W, Walker, Nigel P, Leleti, Manmohan Reddy, Powers, Jay P, Jeffrey, Jenna L
Published in Journal of medicinal chemistry (08.10.2020)
Published in Journal of medicinal chemistry (08.10.2020)
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Journal Article
Design, Synthesis, and Structure-Activity Relationship Optimization of Pyrazolopyrimidine Amide Inhibitors of Phosphoinositide 3-Kinase γ (PI3Kγ)
Mata, Guillaume, Miles, Dillon H, Drew, Samuel L, Fournier, Jeremy, Lawson, Kenneth V, Mailyan, Artur K, Sharif, Ehesan U, Yan, Xuelei, Beatty, Joel W, Banuelos, Jesus, Chen, Jie, Ginn, Elaine, Chen, Ada, Gerrick, Kimberline Y, Pham, Amber T, Wong, Kent, Soni, Divyank, Dhanota, Puja, Shaqfeh, Stefan G, Meleza, Cesar, Narasappa, Nell, Singh, Hema, Zhao, Xiaoning, Jin, Lixia, Schindler, Ulrike, Walters, Matthew J, Young, Stephen W, Walker, Nigel P, Leleti, Manmohan Reddy, Powers, Jay P, Jeffrey, Jenna L
Published in Journal of medicinal chemistry (27.01.2022)
Published in Journal of medicinal chemistry (27.01.2022)
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Journal Article
Total Synthesis of Covalent Cysteine Protease Inhibitor N‑Desmethyl Thalassospiramide C and Crystallographic Evidence for Its Mode of Action
Fournier, Jeremy, Chen, Karen, Mailyan, Artur K, Jackson, Jeffrey J, Buckman, Brad O, Emayan, Kumar, Yuan, Shendong, Rajagopalan, Ravi, Misialek, Shawn, Adler, Marc, Blaesse, Michael, Griessner, Andreas, Zakarian, Armen
Published in Organic letters (18.01.2019)
Published in Organic letters (18.01.2019)
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Journal Article
Fluorinated Unsymmetrical N,N′‐Diaryl Imidazolium Salts—New Functionalized NHC‐Ligand Precursors
Topchiy, Maxim A., Zotova, Maria A., Masoud, Salekh M., Mailyan, Artur K., Ananyev, Ivan V., Nefedov, Sergey E., Asachenko, Andrey F., Osipov, Sergey N.
Published in Chemistry : a European journal (11.05.2017)
Published in Chemistry : a European journal (11.05.2017)
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Journal Article
Metathesis Catalysts with Fluorinated Unsymmetrical NHC Ligands
Masoud, Salekh M, Mailyan, Artur K, Dorcet, Vincent, Roisnel, Thierry, Dixneuf, Pierre H, Bruneau, Christian, Osipov, Sergey N
Published in Organometallics (08.06.2015)
Published in Organometallics (08.06.2015)
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Journal Article
Short Total Synthesis of [ 15 N 5 ]-Cylindrospermopsins from 15 NH 4 Cl Enables Precise Quantification of Freshwater Cyanobacterial Contamination
Mailyan, Artur K, Chen, Joanna L, Li, Weiwei, Keller, Arturo A, Sternisha, Shawn M, Miller, Brian G, Zakarian, Armen
Published in Journal of the American Chemical Society (09.05.2018)
Published in Journal of the American Chemical Society (09.05.2018)
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Journal Article
Short Total Synthesis of [15N5]‑Cylindrospermopsins from 15NH4Cl Enables Precise Quantification of Freshwater Cyanobacterial Contamination
Mailyan, Artur K, Chen, Joanna L, Li, Weiwei, Keller, Arturo A, Sternisha, Shawn M, Miller, Brian G, Zakarian, Armen
Published in Journal of the American Chemical Society (09.05.2018)
Published in Journal of the American Chemical Society (09.05.2018)
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Journal Article
Access to Cyclic -CF3-Substituted -Amino Acid Derivatives by Ring-Closing Metathesis of Functionalized 1,7-Enynes
Mailyan, Artur K., Krylov, Ivan M., Bruneau, Christian, Dixneuf, Pierre H., Osipov, Sergey N.
Published in European journal of organic chemistry (01.08.2013)
Published in European journal of organic chemistry (01.08.2013)
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Journal Article
Cyclobutene Ring-Opening of Bicyclo[4.2.0]octa-1,6-dienes: Access to CF3‑Substituted 5,6,7,8-Tetrahydro-1,7-naphthyridines
Mailyan, Artur K, Peregudov, Alexander S, Dixneuf, Pierre H, Bruneau, Christian, Osipov, Sergey N
Published in Journal of organic chemistry (05.10.2012)
Published in Journal of organic chemistry (05.10.2012)
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Journal Article
Concise Synthesis of (+)‐[13C4]‐Anatoxin‐a by Dynamic Kinetic Resolution of a Cyclic Iminium Ion
Lacharity, Jacob J., Mailyan, Artur K., Chen, Karen Y., Zakarian, Armen
Published in Angewandte Chemie (06.07.2020)
Published in Angewandte Chemie (06.07.2020)
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Journal Article
Scalable Total Synthesis, IP3R Inhibitory Activity of Desmethylxestospongin B, and Effect on Mitochondrial Function and Cancer Cell Survival
Podunavac, Maša, Mailyan, Artur K., Jackson, Jeffrey J., Lovy, Alenka, Farias, Paula, Huerta, Hernan, Molgó, Jordi, Cardenas, Cesar, Zakarian, Armen
Published in Angewandte Chemie (10.05.2021)
Published in Angewandte Chemie (10.05.2021)
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Journal Article
Synthesis of functionalized CF3-containing heterocycles via [2,3]-sigmatropic rearrangement and sequential catalytic carbocyclization
Vorobyeva, Daria V., Mailyan, Artur K., Peregudov, Alexander S., Karimova, Natalia M., Vasilyeva, Tamara P., Bushmarinov, Ivan S., Bruneau, Christian, Dixneuf, Pierre H., Osipov, Sergey N.
Published in Tetrahedron (13.05.2011)
Published in Tetrahedron (13.05.2011)
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Journal Article
Preparation, X-ray Structure, and Oxidative Reactivity of N-(2-Iodylphenyl)tosylamides and 2-Iodylphenyl Tosylate: Iodylarenes Stabilized by Ortho-Substitution with a Sulfonyl Group
Mailyan, Artur K, Geraskin, Ivan M, Nemykin, Victor N, Zhdankin, Viktor V
Published in Journal of organic chemistry (06.11.2009)
Published in Journal of organic chemistry (06.11.2009)
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Journal Article
Convenient synthesis of diarylpropargyl alcohols
Shirinian, Valerii Z., Shimkin, Aleksei A., Mailyan, Artur K., Leonova, Evgeniya S., Krayushkin, Mikhail M.
Published in Mendeleev communications (01.11.2011)
Published in Mendeleev communications (01.11.2011)
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Journal Article