The Role of Heme and the Mitochondrion in the Chemical and Molecular Mechanisms of Mammalian Cell Death Induced by the Artemisinin Antimalarials
Mercer, Amy E., Copple, Ian M., Maggs, James L., O'Neill, Paul M., Park, B. Kevin
Published in The Journal of biological chemistry (14.01.2011)
Published in The Journal of biological chemistry (14.01.2011)
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Journal Article
Evaluation of clinical and genetic factors in the population pharmacokinetics of carbamazepine
Yip, Vincent L.M., Pertinez, Henry, Meng, Xiaoli, Maggs, James L., Carr, Daniel F., Park, B. Kevin, Marson, Anthony G., Pirmohamed, Munir
Published in British journal of clinical pharmacology (01.06.2021)
Published in British journal of clinical pharmacology (01.06.2021)
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Journal Article
The role of metabolic activation in drug-induced hepatotoxicity
PARK, B. Kevin, KITTERINGHAM, Neil R, MAGGS, James L, PIRMOHAMED, Munir, WILLIAMS, Dominic P
Published in Annual review of pharmacology and toxicology (01.01.2005)
Published in Annual review of pharmacology and toxicology (01.01.2005)
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Journal Article
Evidence for the Involvement of Carbon-centered Radicals in the Induction of Apoptotic Cell Death by Artemisinin Compounds
Mercer, Amy E., Maggs, James L., Sun, Xiao-Ming, Cohen, Gerald M., Chadwick, James, O'Neill, Paul M., Park, B. Kevin
Published in The Journal of biological chemistry (30.03.2007)
Published in The Journal of biological chemistry (30.03.2007)
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Journal Article
Acyl glucuronides: the good, the bad and the ugly
Regan, Sophie L., Maggs, James L., Hammond, Thomas G., Lambert, Craig, Williams, Dominic P., Park, B. Kevin
Published in Biopharmaceutics & drug disposition (01.10.2010)
Published in Biopharmaceutics & drug disposition (01.10.2010)
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Journal Article
Mass Spectrometric Characterization of Circulating Covalent Protein Adducts Derived from Epoxide Metabolites of Carbamazepine in Patients
Yip, Vincent L. M, Meng, Xiaoli, Maggs, James L, Jenkins, Rosalind E, Marlot, Philippe T, Marson, Anthony G, Park, B. Kevin, Pirmohamed, Munir
Published in Chemical research in toxicology (17.07.2017)
Published in Chemical research in toxicology (17.07.2017)
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Journal Article
Comparison of the Reactivity of Antimalarial 1,2,4,5-Tetraoxanes with 1,2,4-Trioxolanes in the Presence of Ferrous Iron Salts, Heme, and Ferrous Iron Salts/Phosphatidylcholine
Bousejra-El Garah, Fatima, Wong, Michael He-Long, Amewu, Richard K, Muangnoicharoen, Sant, Maggs, James L, Stigliani, Jean-Luc, Park, B. Kevin, Chadwick, James, Ward, Stephen A, O’Neill, Paul M
Published in Journal of medicinal chemistry (13.10.2011)
Published in Journal of medicinal chemistry (13.10.2011)
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Journal Article
Direct evidence for the formation of diastereoisomeric benzylpenicilloyl haptens from benzylpenicillin and benzylpenicillenic acid in patients
Meng, Xiaoli, Jenkins, Rosalind E, Berry, Neil G, Maggs, James L, Farrell, John, Lane, Catherine S, Stachulski, Andrew V, French, Neil S, Naisbitt, Dean J, Pirmohamed, Munir, Park, B Kevin
Published in The Journal of pharmacology and experimental therapeutics (01.09.2011)
Published in The Journal of pharmacology and experimental therapeutics (01.09.2011)
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Journal Article
Mass spectrometric characterization of circulating covalent protein adducts derived from a drug acyl glucuronide metabolite: multiple albumin adductions in diclofenac patients
Hammond, Thomas G, Meng, Xiaoli, Jenkins, Rosalind E, Maggs, James L, Castelazo, Anahi Santoyo, Regan, Sophie L, Bennett, Stuart N L, Earnshaw, Caroline J, Aithal, Guruprasad P, Pande, Ira, Kenna, J Gerry, Stachulski, Andrew V, Park, B Kevin, Williams, Dominic P
Published in The Journal of pharmacology and experimental therapeutics (01.08.2014)
Published in The Journal of pharmacology and experimental therapeutics (01.08.2014)
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Journal Article
Characterisation of the NRF2 transcriptional network and its response to chemical insult in primary human hepatocytes: implications for prediction of drug-induced liver injury
Copple, Ian M., den Hollander, Wouter, Callegaro, Giulia, Mutter, Fiona E., Maggs, James L., Schofield, Amy L., Rainbow, Lucille, Fang, Yongxiang, Sutherland, Jeffrey J., Ellis, Ewa C., Ingelman-Sundberg, Magnus, Fenwick, Stephen W., Goldring, Christopher E., van de Water, Bob, Stevens, James L., Park, B. Kevin
Published in Archives of toxicology (01.02.2019)
Published in Archives of toxicology (01.02.2019)
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Journal Article
Characterization of Peroxidases Expressed in Human Antigen Presenting Cells and Analysis of the Covalent Binding of Nitroso Sulfamethoxazole to Myeloperoxidase
Ogese, Monday O, Jenkins, Rosalind E, Maggs, James L, Meng, Xiaoli, Whitaker, Paul, Peckham, Daniel, Faulkner, Lee, Park, B. Kevin, Naisbitt, Dean J
Published in Chemical research in toxicology (20.01.2015)
Published in Chemical research in toxicology (20.01.2015)
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Journal Article
Acyl Glucuronides: Biological Activity, Chemical Reactivity, and Chemical Synthesis
Stachulski, Andrew V, Harding, John R, Lindon, John C, Maggs, James L, Park, B. Kevin, Wilson, Ian D
Published in Journal of medicinal chemistry (30.11.2006)
Published in Journal of medicinal chemistry (30.11.2006)
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Journal Article
Dapsone and Nitroso Dapsone Activation of Naı̈ve T‑Cells from Healthy Donors
Alzahrani, Abdulaziz, Ogese, Monday, Meng, Xiaoli, Waddington, James C, Tailor, Arun, Farrell, John, Maggs, James L, Betts, Catherine, Park, B. Kevin, Naisbitt, Dean
Published in Chemical research in toxicology (18.12.2017)
Published in Chemical research in toxicology (18.12.2017)
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Journal Article
Quantifying the Metabolic Activation of Nevirapine in Patients by Integrated Applications of NMR and Mass Spectrometries
SRIVASTAVA, Abhishek, LIAN, Lu-Yun, MAGGS, James L, CHAPONDA, Masautso, PIRMOHAMED, Munir, WILLIAMS, Dominic P, KEVIN PARK, B
Published in Drug metabolism and disposition (01.01.2010)
Published in Drug metabolism and disposition (01.01.2010)
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Journal Article
Multiple Adduction Reactions of Nitroso Sulfamethoxazole with Cysteinyl Residues of Peptides and Proteins: Implications for Hapten Formation
Callan, Hayley E, Jenkins, Rosalind E, Maggs, James L, Lavergne, Sidonie N, Clarke, Stephen E, Naisbitt, Dean J, Park, B. Kevin
Published in Chemical research in toxicology (18.05.2009)
Published in Chemical research in toxicology (18.05.2009)
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Journal Article
Abacavir Forms Novel Cross-Linking Abacavir Protein Adducts in Patients
Meng, Xiaoli, Lawrenson, Alexandre S, Berry, Neil G, Maggs, James L, French, Neil S, Back, David J, Khoo, Saye H, Naisbitt, Dean J, Park, B. Kevin
Published in Chemical research in toxicology (21.04.2014)
Published in Chemical research in toxicology (21.04.2014)
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Journal Article
Convenient Syntheses of Benzo-Fluorinated Dibenz[b,f]azepines: Rearrangements of Isatins, Acridines, and Indoles
Elliott, Emma-Claire, Bowkett, Elizabeth R, Maggs, James L, Bacsa, John, Park, B. Kevin, Regan, Sophie L, O’Neill, Paul M, Stachulski, Andrew V
Published in Organic letters (21.10.2011)
Published in Organic letters (21.10.2011)
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Journal Article
Haloarene Derivatives of Carbamazepine with Reduced Bioactivation Liabilities: 2‑Monohalo and 2,8-Dihalo Derivatives
Elliott, Emma-Claire, Regan, Sophie L, Maggs, James L, Bowkett, Elizabeth R, Parry, Laura J, Williams, Dominic P, Park, B. Kevin, Stachulski, Andrew V
Published in Journal of medicinal chemistry (26.11.2012)
Published in Journal of medicinal chemistry (26.11.2012)
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Journal Article