Ligands for Glutamate Receptors: Design and Therapeutic Prospects
Bräuner-Osborne, Hans, Egebjerg, Jan, Nielsen, Elsebet Ø, Madsen, Ulf, Krogsgaard-Larsen, Povl
Published in Journal of medicinal chemistry (13.07.2000)
Published in Journal of medicinal chemistry (13.07.2000)
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Inhibitors of AMPA and Kainate Receptors
Madsen, U., Stensbol, T., Krogsgaard-Larsen, P.
Published in Current medicinal chemistry (01.09.2001)
Published in Current medicinal chemistry (01.09.2001)
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Novel 1-Hydroxyazole Bioisosteres of Glutamic Acid. Synthesis, Protolytic Properties, and Pharmacology
Stensbøl, Tine B, Uhlmann, Peter, Morel, Sandrine, Eriksen, Birgitte L, Felding, Jakob, Kromann, Hasse, Hermit, Mette B, Greenwood, Jeremy R, Braüner-Osborne, Hans, Madsen, Ulf, Junager, Finn, Krogsgaard-Larsen, Povl, Begtrup, Mikael, Vedsø, Per
Published in Journal of medicinal chemistry (03.01.2002)
Published in Journal of medicinal chemistry (03.01.2002)
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Structural Determinants of AMPA Agonist Activity in Analogues of 2-Amino-3-(3-carboxy-5-methyl-4-isoxazolyl)propionic Acid: Synthesis and Pharmacology
Bang-Andersen, Benny, Ahmadian, Haleh, Lenz, Sibylle M, Stensbøl, Tine B, Madsen, Ulf, Bøgesø, Klaus P, Krogsgaard-Larsen, Povl
Published in Journal of medicinal chemistry (14.12.2000)
Published in Journal of medicinal chemistry (14.12.2000)
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Agonist discrimination between AMPA receptor subtypes
Coquelle, T, Christensen, J K, Banke, T G, Madsen, U, Schousboe, A, Pickering, D S
Published in Neuroreport (21.08.2000)
Published in Neuroreport (21.08.2000)
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(S)-Homo-AMPA, a Specific Agonist at the mGlu6 Subtype of Metabotropic Glutamic Acid Receptors
Ahmadian, Haleh, Nielsen, Birgitte, Bräuner-Osborne, Hans, Johansen, Tommy N, Stensbøl, Tine B, Sløk, Frank A, Sekiyama, Naohiro, Nakanishi, Shigetada, Krogsgaard-Larsen, Povl, Madsen, Ulf
Published in Journal of medicinal chemistry (24.10.1997)
Published in Journal of medicinal chemistry (24.10.1997)
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Synthesis and Pharmacology of 3-Isoxazolol Amino Acids as Selective Antagonists at Group I Metabotropic Glutamic Acid Receptors
Madsen, Ulf, Bräuner-Osborne, Hans, Frydenvang, Karla, Hvene, Lise, Johansen, Tommy N, Nielsen, Birgitte, Sánchez, Connie, Stensbøl, Tine B, Bischoff, Francois, Krogsgaard-Larsen, Povl
Published in Journal of medicinal chemistry (29.03.2001)
Published in Journal of medicinal chemistry (29.03.2001)
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Pharmacology and toxicology of ATOA, an AMPA receptor antagonist and a partial agonist at GluR5 receptors
Wahl, P, Frandsen, A, Madsen, U, Schousboe, A, Krogsgaard-Larsen, P
Published in Neuropharmacology (01.10.1998)
Published in Neuropharmacology (01.10.1998)
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Design of excitatory amino acid receptor agonists, partial agonists and antagonists: ibotenic acid as a key lead structure
Krogsgaard-Larsen, P, Ebert, B, Lund, TM, Bräuner-Osborne, H, Sløk, FA, Johansen, TN, Brehm, L, Madsen, U
Published in European journal of medicinal chemistry (1996)
Published in European journal of medicinal chemistry (1996)
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Excitatory amino-acid receptor agonists. Synthesis and pharmacology of analogues of 2-amino-3-(3-hydroxy-5-methylisoxazol-4-yl)propionic acid
Sløk, F.A., Ebert, B, Lang, Y, Krogsgaard-Larsen, P, Lenz, S.M., Madsen, U
Published in European journal of medicinal chemistry (1997)
Published in European journal of medicinal chemistry (1997)
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Synthesis and Pharmacology of a New AMPA−Kainate Receptor Agonist with Potent Convulsant Activity
Conti, Paola, De Amici, Marco, De Sarro, Giovambattista, Stensbøl, Tine Bryan, Bräuner-Osborne, Hans, Madsen, Ulf, De Micheli, Carlo
Published in Journal of medicinal chemistry (24.09.1998)
Published in Journal of medicinal chemistry (24.09.1998)
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Excitatory amino acid receptor ligands: Asymmetric synthesis, absolute stereochemistry and pharmacology of ( R)- and ( S)-homoibotenic acid
Bischoff, F., Johansen, T.N., Ebert, B., Krogsgaard-Larsen, P., Madsen, U.
Published in Bioorganic & medicinal chemistry (01.05.1995)
Published in Bioorganic & medicinal chemistry (01.05.1995)
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Differentiation of in vivo effects of AMPA and NMDA receptor ligands using drug discrimination methods and convulsant/anticonvulsant activity
Arnt, Jørn, Sánchez, Connie, Lenz, Sibylle Moltzen, Madsen, Ulf, Krogsgaard-Larsen, Povl
Published in European journal of pharmacology (24.10.1995)
Published in European journal of pharmacology (24.10.1995)
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Studies of the antagonist actions of (RS)‐2‐amino‐3‐[5‐tert‐butyl‐3‐(phosphonomethoxy)‐4‐isoxazolyl]propionic acid (ATPO) on non‐NMDA receptors in cultured rat neurones
Dai, W‐M, Ebert, B, Madsen, U, Lambert, J D C
Published in British journal of pharmacology (01.12.1998)
Published in British journal of pharmacology (01.12.1998)
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