Synthesis and anti-cancer screening of novel heterocyclic-(2H)-1,2,3-triazoles as potential anti-cancer agents
Penthala, Narsimha Reddy, Madhukuri, Leena, Thakkar, Shraddha, Madadi, Nikhil Reddy, Lamture, Gauri, Eoff, Robert L, Crooks, Peter A
Published in MedChemComm (01.08.2015)
Published in MedChemComm (01.08.2015)
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Journal Article
Synthesis and in vitro evaluation of N-alkyl-3-hydroxy-3-(2-imino-3-methyl-5-oxoimidazolidin-4-yl)indolin-2-one analogs as potential anticancer agents
Penthala, Narsimha Reddy, Yerramreddy, Thirupathi Reddy, Madadi, Nikhil Reddy, Crooks, Peter A.
Published in Bioorganic & medicinal chemistry letters (01.08.2010)
Published in Bioorganic & medicinal chemistry letters (01.08.2010)
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Journal Article
Comparison of crystal structures of 4-(benzo[b]thio-phen-2-yl)-5-(3,4,5-tri-meth-oxy-phen-yl)-2H-1,2,3-triazole and 4-(benzo[b]thio-phen-2-yl)-2-methyl-5-(3,4,5-tri-meth-oxy-phen-yl)-2H-1,2,3-triazole
Penthala, Narsimha Reddy, Madadi, Nikhil Reddy, Bommagani, Shobanbabu, Parkin, Sean, Crooks, Peter A
Published in Acta crystallographica. Section E, Structure reports online (01.11.2014)
Published in Acta crystallographica. Section E, Structure reports online (01.11.2014)
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Journal Article
Crystal structure of 4,5-bis-(3,4,5-tri-meth-oxy-phen-yl)-2H-1,2,3-triazole methanol monosolvate
Madadi, Nikhil Reddy, Penthala, Narsimha Reddy, Bommagani, Shobanbabu, Parkin, Sean, Crooks, Peter A
Published in Acta crystallographica. Section E, Structure reports online (01.10.2014)
Published in Acta crystallographica. Section E, Structure reports online (01.10.2014)
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Journal Article
Monosuccinate ester of melampomagnolide B
Janganati, Venumadhav, Penthala, Narsimha Reddy, Madadi, Nikhil Reddy, Parkin, Sean, Crooks, Peter A
Published in Acta crystallographica. Section E, Structure reports online (01.03.2014)
Published in Acta crystallographica. Section E, Structure reports online (01.03.2014)
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Journal Article
Synthesis and anti-proliferative activity of aromatic substituted 5-((1-benzyl-1H-indol-3-yl)methylene)-1,3-dimethylpyrimidine-2,4,6(1H,3H,5H)-trione analogs against human tumor cell lines
Madadi, Nikhil Reddy, Penthala, Narsimha Reddy, Janganati, Venumadhav, Crooks, Peter A.
Published in Bioorganic & medicinal chemistry letters (15.01.2014)
Published in Bioorganic & medicinal chemistry letters (15.01.2014)
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Journal Article
Synthesis, anticancer activity and molecular docking studies on a series of heterocyclic trans-cyanocombretastatin analogues as antitubulin agents
Penthala, Narsimha Reddy, Zong, Hongliang, Ketkar, Amit, Madadi, Nikhil Reddy, Janganati, Venumadav, Eoff, Robert L., Guzman, Monica L., Crooks, Peter A.
Published in European journal of medicinal chemistry (06.03.2015)
Published in European journal of medicinal chemistry (06.03.2015)
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Journal Article
L-Proline catalyzed one-step synthesis of 4,5-diaryl-2 H -1,2,3-triazoles from heteroaryl cyanostilbenes via [3+2] cycloaddition of azide
Penthala, Narsimha Reddy, Madadi, Nikhil Reddy, Janganati, Venumadhav, Crooks, Peter A
Published in Tetrahedron letters (01.10.2014)
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Published in Tetrahedron letters (01.10.2014)
Journal Article
Evaluation of (Z)-2-((1-benzyl-1H-indol-3-yl)methylene)-quinuclidin-3-one analogues as novel, high affinity ligands for CB1 and CB2 cannabinoid receptors
Madadi, Nikhil Reddy, Penthala, Narsimha Reddy, Brents, Lisa K., Ford, Benjamin M., Prather, Paul L., Crooks, Peter A.
Published in Bioorganic & medicinal chemistry letters (01.04.2013)
Published in Bioorganic & medicinal chemistry letters (01.04.2013)
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Journal Article
( Z )-2-Amino-5-[2,4-dimethoxy-6-(4-methoxystyryl)benzylidene]-1,3-thiazol-4(5 H )-one methanol solvate
Madadi, Nikhil Reddy, Reddy, Thirupathi Reddy Yerram, Penthala, Narsimha Reddy, Parkin, Sean, Crooks, Peter A.
Published in Acta crystallographica. Section E, Structure reports online (01.07.2010)
Published in Acta crystallographica. Section E, Structure reports online (01.07.2010)
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Journal Article
Synthesis and in vitro evaluation of N-alkyl-3-hydroxy-3-(2-imino-3-methyl-5-oxoimidazolidin-4-yl)in dolin-2-one analogs as potential anticancer agents
Penthala, Narsimha Reddy, Yerramreddy, Thirupathi Reddy, Madadi, Nikhil Reddy, Crooks, Peter A
Published in Bioorganic & medicinal chemistry letters (01.08.2010)
Published in Bioorganic & medicinal chemistry letters (01.08.2010)
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Journal Article
Comparison of crystal structures of 4-(benzo[ b ]thiophen-2-yl)-5-(3,4,5-trimethoxyphenyl)-2 H -1,2,3-triazole and 4-(benzo[ b ]thiophen-2-yl)-2-methyl-5-(3,4,5-trimethoxyphenyl)-2 H -1,2,3-triazole
Penthala, Narsimha Reddy, Madadi, Nikhil Reddy, Bommagani, Shobanbabu, Parkin, Sean, Crooks, Peter A.
Published in Acta crystallographica. Section E, Structure reports online (01.11.2014)
Published in Acta crystallographica. Section E, Structure reports online (01.11.2014)
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Journal Article
Crystal structure of 4,5-bis(3,4,5-trimethoxyphenyl)-2 H -1,2,3-triazole methanol monosolvate
Madadi, Nikhil Reddy, Penthala, Narsimha Reddy, Bommagani, Shobanbabu, Parkin, Sean, Crooks, Peter A.
Published in Acta crystallographica. Section E, Structure reports online (01.10.2014)
Published in Acta crystallographica. Section E, Structure reports online (01.10.2014)
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Journal Article
Disubstituted triazole analogs
Penthala, Narsimha Reddy, Maddukuri, Leena, Madadi, Nikhil Reddy, Crooks, Peter, Eoff, Robert
Year of Publication 26.03.2019
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Year of Publication 26.03.2019
Patent
ChemInform Abstract: L-Proline Catalyzed One-Step Synthesis of 4,5-Diaryl-2H-1,2,3-triazoles from Heteroaryl Cyanostilbenes via [3 + 2]Cycloaddition of Azide
Penthala, Narsimha Reddy, Madadi, Nikhil Reddy, Janganati, Venumadhav, Crooks, Peter A.
Published in ChemInform (01.03.2015)
Published in ChemInform (01.03.2015)
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Journal Article
DISUBSTITUTED TRIAZOLE ANALOGS
Penthala, Narsimha Reddy, Maddukuri, Leena, Madadi, Nikhil Reddy, Crooks, Peter, Eoff, Robert
Year of Publication 05.07.2018
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Year of Publication 05.07.2018
Patent