Lipolysis of Triglyceride-Rich Lipoproteins Generates PPAR Ligands: Evidence for an Antiinflammatory Role for Lipoprotein Lipase
Ziouzenkova, Ouliana, Perrey, Stephane, Asatryan, Liana, Hwang, Juliana, MacNaul, Karen L., Moller, David E., Rader, Daniel J., Sevanian, Alex, Zechner, Rudolf, Hoefler, Gerald, Plutzky, Jorge
Published in Proceedings of the National Academy of Sciences - PNAS (04.03.2003)
Published in Proceedings of the National Academy of Sciences - PNAS (04.03.2003)
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Journal Article
A Potent Synthetic LXR Agonist Is More Effective than Cholesterol Loading at Inducing ABCA1 mRNA and Stimulating Cholesterol Efflux
Sparrow, Carl P., Baffic, Joanne, Lam, My-Hanh, Lund, Erik G., Adams, Alan D., Fu, Xuan, Hayes, Nancy, Jones, A. Brian, Macnaul, Karen L., Ondeyka, John, Singh, Sheo, Wang, Jianhua, Zhou, Gaochao, Moller, David E., Wright, Samuel D., Menke, John G.
Published in The Journal of biological chemistry (22.03.2002)
Published in The Journal of biological chemistry (22.03.2002)
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Journal Article
27-Hydroxycholesterol Is an Endogenous Ligand for Liver X Receptor in Cholesterol-loaded Cells
Fu, Xuan, Menke, John G., Chen, Yuli, Zhou, Gaochao, MacNaul, Karen L., Wright, Samuel D., Sparrow, Carl P., Lund, Erik G.
Published in The Journal of biological chemistry (19.10.2001)
Published in The Journal of biological chemistry (19.10.2001)
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Journal Article
Distinct Properties and Advantages of a Novel Peroxisome Proliferator-Activated Protein γ Selective Modulator
Berger, Joel P, Petro, Ann E, Macnaul, Karen L, Kelly, Linda J, Zhang, Bei B, Richards, Karen, Elbrecht, Alex, Johnson, Bruce A, Zhou, Gaochao, Doebber, Thomas W, Biswas, Chhabi, Parikh, Mona, Sharma, Neelam, Tanen, Michael R, Thompson, G. Marie, Ventre, John, Adams, Alan D, Mosley, Ralph, Surwit, Richard S, Moller, David E
Published in Molecular endocrinology (Baltimore, Md.) (01.04.2003)
Published in Molecular endocrinology (Baltimore, Md.) (01.04.2003)
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Journal Article
PPAR-gamma activation mediates adipose depot-specific effects on gene expression and lipoprotein lipase activity: mechanisms for modulation of postprandial lipemia and differential adipose accretion
Laplante, Mathieu, Sell, Henrike, MacNaul, Karen L, Richard, Denis, Berger, Joel P, Deshaies, Yves
Published in Diabetes (New York, N.Y.) (01.02.2003)
Published in Diabetes (New York, N.Y.) (01.02.2003)
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Journal Article
Benzoyl 2-methyl indoles as selective PPARγ modulators
Acton, John J., Black, Regina M., Jones, A. Brian, Moller, David E., Colwell, Lawrence, Doebber, Thomas W., MacNaul, Karen L., Berger, Joel, Wood, Harold B.
Published in Bioorganic & medicinal chemistry letters (17.01.2005)
Published in Bioorganic & medicinal chemistry letters (17.01.2005)
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Journal Article
Novel 2,3-Dihydrobenzofuran-2-carboxylic Acids: Highly Potent and Subtype-Selective PPARα Agonists with Potent Hypolipidemic Activity
Shi, Guo Q, Dropinski, James F, Zhang, Yong, Santini, Conrad, Sahoo, Soumya P, Berger, Joel P, MacNaul, Karen L, Zhou, Gaochao, Agrawal, Arun, Alvaro, Raul, Cai, Tian-quan, Hernandez, Melba, Wright, Samuel D, Moller, David E, Heck, James V, Meinke, Peter T
Published in Journal of medicinal chemistry (25.08.2005)
Published in Journal of medicinal chemistry (25.08.2005)
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Journal Article
Design and Synthesis of α-Aryloxyphenylacetic Acid Derivatives: A Novel Class of PPARα/γ Dual Agonists with Potent Antihyperglycemic and Lipid Modulating Activity
Shi, Guo Q, Dropinski, James F, McKeever, Brian M, Xu, Shihua, Becker, Joseph W, Berger, Joel P, MacNaul, Karen L, Elbrecht, Alex, Zhou, Gaochao, Doebber, Thomas W, Wang, Peiran, Chao, Yu-Sheng, Forrest, Mike, Heck, James V, Moller, David E, Jones, A. Brian
Published in Journal of medicinal chemistry (30.06.2005)
Published in Journal of medicinal chemistry (30.06.2005)
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Journal Article
A Novel Liver X Receptor Agonist Establishes Species Differences in the Regulation of Cholesterol 7α-Hydroxylase (CYP7a)
Menke, John G, Macnaul, Karen L, Hayes, Nancy S, Baffic, Joanne, Chao, Yu-Sheng, Elbrecht, Alex, Kelly, Linda J, Lam, My-Hanh, Schmidt, Azriel, Sahoo, Soumya, Wang, Jianhua, Wright, Samuel D, Xin, Patrick, Zhou, Gaochao, Moller, David E, Sparrow, Carl P
Published in Endocrinology (Philadelphia) (01.07.2002)
Published in Endocrinology (Philadelphia) (01.07.2002)
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Journal Article
Selective PPARγ modulators with improved pharmacological profiles
Liu, Kun, Black, Regina M., Acton, John J., Mosley, Ralph, Debenham, Sheryl, Abola, Ramon, Yang, Meng, Tschirret-Guth, Richard, Colwell, Lawrence, Liu, Cherrie, Wu, Margaret, Wang, Chuanlin F., MacNaul, Karen L., McCann, Margaret E., Moller, David E., Berger, Joel P., Meinke, Peter T., Jones, A. Brian, Wood, Harold B.
Published in Bioorganic & medicinal chemistry letters (16.05.2005)
Published in Bioorganic & medicinal chemistry letters (16.05.2005)
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Journal Article
Discovery of a Novel Series of Peroxisome Proliferator-Activated Receptor α/γ Dual Agonists for the Treatment of Type 2 Diabetes and Dyslipidemia
Liu, Kun, Xu, Libo, Berger, Joel P, MacNaul, Karen L, Zhou, Gauchao, Doebber, Thomas W, Forrest, Michael J, Moller, David E, Jones, A. Brian
Published in Journal of medicinal chemistry (07.04.2005)
Published in Journal of medicinal chemistry (07.04.2005)
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Journal Article
5-Aryl thiazolidine-2,4-diones: discovery of PPAR dual α/γ agonists as antidiabetic agents
Desai, Ranjit C., Han, Wei, Metzger, Edward J., Bergman, Jeffrey P., Gratale, Dominick F., MacNaul, Karen L., Berger, Joel P., Doebber, Thomas W., Leung, Kwan, Moller, David E., Heck, James V., Sahoo, Soumya P.
Published in Bioorganic & medicinal chemistry letters (18.08.2003)
Published in Bioorganic & medicinal chemistry letters (18.08.2003)
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Journal Article
(2R)-2-Ethylchromane-2-carboxylic Acids: Discovery of Novel PPARα/γ Dual Agonists as Antihyperglycemic and Hypolipidemic Agents
Koyama, Hiroo, Miller, Daniel J, Boueres, Julia K, Desai, Ranjit C, Jones, A. Brian, Berger, Joel P, MacNaul, Karen L, Kelly, Linda J, Doebber, Thomas W, Wu, Margaret S, Zhou, Gaochao, Wang, Pei-ran, Ippolito, Marc C, Chao, Yu-Sheng, Agrawal, Arun K, Franklin, Ronald, Heck, James V, Wright, Samuel D, Moller, David E, Sahoo, Soumya P
Published in Journal of medicinal chemistry (03.06.2004)
Published in Journal of medicinal chemistry (03.06.2004)
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Journal Article
Amphipathic 3-Phenyl-7-propylbenzisoxazoles; human pPaR γ, δ and α agonists
Adams, Alan D, Yuen, Winston, Hu, Zao, Santini, Conrad, Jones, A.Brian, MacNaul, Karen L, Berger, Joel P, Doebber, Thomas W, Moller, David E
Published in Bioorganic & medicinal chemistry letters (10.03.2003)
Published in Bioorganic & medicinal chemistry letters (10.03.2003)
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Journal Article
A Novel Peroxisome Proliferator-Activated Receptor α/γ Dual Agonist Demonstrates Favorable Effects on Lipid Homeostasis
Guo, Qiu, Sahoo, Soumya P, Wang, Pei-Ran, Milot, Denise P, Ippolito, Marc C, Wu, Margaret S, Baffic, Joanne, Biswas, Chhabi, Hernandez, Melba, Lam, My-Hanh, Sharma, Neelam, Han, Wei, Kelly, Linda J, MacNaul, Karen L, Zhou, Gaochao, Desai, Ranjit, Heck, James V, Doebber, Thomas W, Berger, Joel P, Moller, David E, Sparrow, Carl P, Chao, Yu-sheng, Wright, Samuel D
Published in Endocrinology (Philadelphia) (01.04.2004)
Published in Endocrinology (Philadelphia) (01.04.2004)
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Journal Article
Design and synthesis of potent and subtype-selective PPARα agonists
Desai, Ranjit C., Metzger, Edward, Santini, Conrad, Meinke, Peter T., Heck, James V., Berger, Joel P., MacNaul, Karen L., Cai, Tian-quan, Wright, Samuel D., Agrawal, Arun, Moller, David E., Sahoo, Soumya P.
Published in Bioorganic & medicinal chemistry letters (15.03.2006)
Published in Bioorganic & medicinal chemistry letters (15.03.2006)
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Journal Article
(2 R)-2-Methylchromane-2-carboxylic acids: Discovery of selective PPARα agonists as hypolipidemic agents
Koyama, Hiroo, Boueres, Julia K., Miller, Daniel J., Berger, Joel P., MacNaul, Karen L., Wang, Pei-ran, Ippolito, Marc C., Wright, Samuel D., Agrawal, Arun K., Moller, David E., Sahoo, Soumya P.
Published in Bioorganic & medicinal chemistry letters (15.07.2005)
Published in Bioorganic & medicinal chemistry letters (15.07.2005)
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Journal Article
Aryloxazolidinediones: Identification of potent orally active PPAR dual α/γ agonists
DESAI, Ranjit C, GRATALE, Dominick F, FRANKLIN, Ronald, MOLLER, David E, HECK, James V, SAHOO, Soumya P, WEI HAN, KOYAMA, Hiroo, METZGER, Edward, LOMBARDO, Victoria K, MACNAUL, Karen L, DOEBBER, Thomas W, BERGER, Joel P, LEUNG, Kwan
Published in Bioorganic & medicinal chemistry letters (20.10.2003)
Published in Bioorganic & medicinal chemistry letters (20.10.2003)
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Journal Article
O-Arylmandelic acids as highly selective human PPAR α/γ agonists
Adams, Alan D, Hu, Zao, von Langen, Derek, Dadiz, Adonis, Elbrecht, Alex, MacNaul, Karen L, Berger, Joel P, Zhou, Gaochao, Doebber, Thomas W, Meurer, Roger, Forrest, Michael J, Moller, David E, Brian Jones, A
Published in Bioorganic & medicinal chemistry letters (06.10.2003)
Published in Bioorganic & medicinal chemistry letters (06.10.2003)
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Journal Article
5-Aryl thiazolidine-2,4-diones as selective PPARγ agonists
Koyama, Hiroo, Boueres, Julia K, Han, Wei, Metzger, Edward J, Bergman, Jeffrey P, Gratale, Dominick F, Miller, Daniel J, Tolman, Richard L, MacNaul, Karen L, Berger, Joel P, Doebber, Thomas W, Leung, Kwan, Moller, David E, Heck, James V, Sahoo, Soumya P
Published in Bioorganic & medicinal chemistry letters (19.05.2003)
Published in Bioorganic & medicinal chemistry letters (19.05.2003)
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Journal Article