Identification of Novel Pathways of Osimertinib Disposition and Potential Implications for the Outcome of Lung Cancer Therapy
MacLeod, A Kenneth, Lin, De, Huang, Jeffrey T-J, McLaughlin, Lesley A, Henderson, Colin J, Wolf, C Roland
Published in Clinical cancer research (01.05.2018)
Published in Clinical cancer research (01.05.2018)
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Aldo-keto reductases are biomarkers of NRF2 activity and are co-ordinately overexpressed in non-small cell lung cancer
MacLeod, A Kenneth, Acosta-Jimenez, Lourdes, Coates, Philip J, McMahon, Michael, Carey, Frank A, Honda, Tadashi, Henderson, Colin J, Wolf, C Roland
Published in British journal of cancer (06.12.2016)
Published in British journal of cancer (06.12.2016)
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Journal Article
Supine posture changes lung volumes and increases ventilation heterogeneity in cystic fibrosis
Smith, Laurie J, Macleod, Kenneth A, Collier, Guilhem J, Horn, Felix C, Sheridan, Helen, Aldag, Ina, Taylor, Chris J, Cunningham, Steve, Wild, Jim M, Horsley, Alex
Published in PloS one (27.11.2017)
Published in PloS one (27.11.2017)
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Biologicals in childhood severe asthma: the European PERMEABLE survey on the status quo
Santos-Valente, Elisangela, Buntrock-Döpke, Heike, Abou Taam, Rola, Arasi, Stefania, Bakirtas, Arzu, Lozano Blasco, Jaime, Bønnelykke, Klaus, Craiu, Mihai, Cutrera, Renato, Deschildre, Antoine, Elnazir, Basil, Fleming, Louise, Frey, Urs, Gappa, Monika, Nieto García, Antonio, Skamstrup Hansen, Kirsten, Hanssens, Laurence, Jahnz-Rozyk, Karina, Jesenak, Milos, Kerzel, Sebastian, Kopp, Matthias V., Koppelman, Gerard H., Krivec, Uros, MacLeod, Kenneth A., Mäkelä, Mika, Melén, Erik, Mezei, Györgyi, Moeller, Alexander, Moreira, Andre, Pohunek, Petr, Minić, Predrag, Rutjes, Niels W.P., Sammut, Patrick, Schwerk, Nicolaus, Szépfalusi, Zsolt, Turkalj, Mirjana, Tzotcheva, Iren, Ulmeanu, Alexandru, Verhulst, Stijn, Xepapadaki, Paraskevi, Niggel, Jakob, Vijverberg, Susanne, Maitland-van der Zee, Anke H., Potočnik, Uroš, Reinartz, Susanne M., van Drunen, Cornelis M., Kabesch, Michael
Published in ERJ open research (01.07.2021)
Published in ERJ open research (01.07.2021)
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A Targeted in Vivo SILAC Approach for Quantification of Drug Metabolism Enzymes: Regulation by the Constitutive Androstane Receptor
MacLeod, A. Kenneth, Zang, Tuo, Riches, Zoe, Henderson, Colin J, Wolf, C. Roland, Huang, Jeffrey T.-J
Published in Journal of proteome research (07.02.2014)
Published in Journal of proteome research (07.02.2014)
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Lung clearance index (LCI2.5) changes after initiation of Elexacaftor/Tezacaftor/Ivacaftor in children with cystic fibrosis aged between 6 and 11 years: The “real‐world” differs from trial data
Urquhart, Don S., Dowle, Heather, Moffat, Kellie, Forster, Jody, Cunningham, Steve, Macleod, Kenneth A.
Published in Pediatric pulmonology (01.05.2024)
Published in Pediatric pulmonology (01.05.2024)
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Characterization of the cancer chemopreventive NRF2-dependent gene battery in human keratinocytes: demonstration that the KEAP1–NRF2 pathway, and not the BACH1–NRF2 pathway, controls cytoprotection against electrophiles as well as redox-cycling compounds
MacLeod, A.Kenneth, McMahon, Michael, Plummer, Simon M., Higgins, Larry G., Penning, Trevor M., Igarashi, Kazuhiko, Hayes, John D.
Published in Carcinogenesis (New York) (01.09.2009)
Published in Carcinogenesis (New York) (01.09.2009)
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Journal Article
Acceleration of infectious disease drug discovery and development using a humanized model of drug metabolism
MacLeod, A Kenneth, Coquelin, Kevin-Sebastien, Huertas, Leticia, Simeons, Frederick R C, Riley, Jennifer, Casado, Patricia, Guijarro, Laura, Casanueva, Ruth, Frame, Laura, Pinto, Erika G, Ferguson, Liam, Duncan, Christina, Mutter, Nicole, Shishikura, Yoko, Henderson, Colin J, Cebrian, David, Wolf, C Roland, Read, Kevin D
Published in Proceedings of the National Academy of Sciences - PNAS (13.02.2024)
Published in Proceedings of the National Academy of Sciences - PNAS (13.02.2024)
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Journal Article
Expression and Localization of Rat Aldo-Keto Reductases and Induction of the 1B13 and 1D2 Isoforms by Phenolic Antioxidants
MACLEOD, A. Kenneth, KELLY, Vincent P, HIGGINS, Larry G, KELLEHER, Michael O, PRICE, Sally A, BIGLEY, Alison L, BETTON, Graham R, HAYES, John D
Published in Drug metabolism and disposition (01.02.2010)
Published in Drug metabolism and disposition (01.02.2010)
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Journal Article
Metabolism of deltamethrin and cis- and trans-permethrin by human expressed cytochrome P450 and carboxylesterase enzymes
Hedges, Laura, Brown, Susan, MacLeod, A Kenneth, Vardy, Audrey, Doyle, Edward, Song, Gina, Moreau, Marjory, Yoon, Miyoung, Osimitz, Thomas G, Lake, Brian G
Published in Xenobiotica (04.05.2019)
Published in Xenobiotica (04.05.2019)
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Metabolism of bifenthrin, β-cyfluthrin, λ-cyhalothrin, cyphenothrin and esfenvalerate by rat and human cytochrome P450 and carboxylesterase enzymes
Hedges, Laura, Brown, Susan, MacLeod, A. Kenneth, Moreau, Marjory, Yoon, Miyoung, Creek, Moire R., Osimitz, Thomas G., Lake, Brian G.
Published in Xenobiotica (01.12.2020)
Published in Xenobiotica (01.12.2020)
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Journal Article
Changes in physiological, functional and structural markers of cystic fibrosis lung disease with treatment of a pulmonary exacerbation
Horsley, Alex R, Davies, Jane C, Gray, Robert D, Macleod, Kenneth A, Donovan, Jackie, Aziz, Zelena A, Bell, Nicholas J, Rainer, Margaret, Mt-Isa, Shahrul, Voase, Nia, Dewar, Maria H, Saunders, Clare, Gibson, James S, Parra-Leiton, Javier, Larsen, Mia D, Jeswiet, Sarah, Soussi, Samia, Bakar, Yusura, Meister, Mark G, Tyler, Philippa, Doherty, Ann, Hansell, David M, Ashby, Deborah, Hyde, Stephen C, Gill, Deborah R, Greening, Andrew P, Porteous, David J, Innes, J Alastair, Boyd, A Christopher, Griesenbach, Uta, Cunningham, Steve, Alton, Eric WFW
Published in Thorax (01.06.2013)
Published in Thorax (01.06.2013)
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Differential lymphatic versus portal vein uptake of the synthetic pyrethroids deltamethrin and cis-permethrin in rats
Higgins, Larry G., Chatham, Lynsey R., Tomczynski, Sara L., MacLeod, A. Kenneth, Moreau, Marjory, Clewell, Harvey J., Yoon, Miyoung, Creek, Moire R., Osimitz, Thomas G., Lake, Brian G.
Published in Toxicology (Amsterdam) (01.10.2020)
Published in Toxicology (Amsterdam) (01.10.2020)
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Journal Article
Aldo-keto reductases are biomarkers of NRF2 activity and are co-ordinately overexpressed in non-small cell lung cancer
MacLeod, A Kenneth, Acosta-Jimenez, Lourdes, Coates, Philip J, McMahon, Michael, Carey, Frank A, Honda, Tadashi, Hayes, John D, Henderson, Colin J, Wolf, C Roland
Published in British journal of cancer (22.08.2017)
Published in British journal of cancer (22.08.2017)
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Journal Article
Xenobiotic CAR Activators Induce Dlk1-Dio3 Locus Noncoding RNA Expression in Mouse Liver
Pouché, Lucie, Vitobello, Antonio, Römer, Michael, Glogovac, Milica, MacLeod, A Kenneth, Ellinger-Ziegelbauer, Heidrun, Westphal, Magdalena, Dubost, Valérie, Stiehl, Daniel Philipp, Dumotier, Bérengère, Fekete, Alexander, Moulin, Pierre, Zell, Andreas, Schwarz, Michael, Moreno, Rita, Huang, Jeffrey T J, Elcombe, Cliff R, Henderson, Colin J, Roland Wolf, C, Moggs, Jonathan G, Terranova, Rémi
Published in Toxicological sciences (01.08.2017)
Published in Toxicological sciences (01.08.2017)
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