Characterising covalent warhead reactivity
Martin, James S., MacKenzie, Claire J., Fletcher, Daniel, Gilbert, Ian H.
Published in Bioorganic & medicinal chemistry (15.05.2019)
Published in Bioorganic & medicinal chemistry (15.05.2019)
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Synthesis of a Series of Diaminoindoles
Martin, James S, Mackenzie, Claire J, Gilbert, Ian H
Published in Journal of organic chemistry (03.09.2021)
Published in Journal of organic chemistry (03.09.2021)
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Respiratory flexibility in response to inhibition of cytochrome C oxidase in Mycobacterium tuberculosis
Arora, Kriti, Ochoa-Montaño, Bernardo, Tsang, Patricia S, Blundell, Tom L, Dawes, Stephanie S, Mizrahi, Valerie, Bayliss, Tracy, Mackenzie, Claire J, Cleghorn, Laura A T, Ray, Peter C, Wyatt, Paul G, Uh, Eugene, Lee, Jinwoo, Barry, 3rd, Clifton E, Boshoff, Helena I
Published in Antimicrobial agents and chemotherapy (01.11.2014)
Published in Antimicrobial agents and chemotherapy (01.11.2014)
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Application of an NMR/Crystallography Fragment Screening Platform for the Assessment and Rapid Discovery of New HIV‐CA Binding Fragments
Lang, Stuart, Fletcher, Daniel A., Petit, Alain‐Pierre, Luise, Nicola, Fyfe, Paul, Zuccotto, Fabio, Porter, David, Hope, Anthony, Bellany, Fiona, Kerr, Catrina, Mackenzie, Claire J., Wyatt, Paul G., Gray, David W.
Published in ChemMedChem (02.07.2024)
Published in ChemMedChem (02.07.2024)
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Design and Synthesis of Covalent Inhibitors of FabA
Martin, James S., Mackenzie, Claire J., Lin, De, Homeyer, Nadine, Gray, David W., Zuccotto, Fabio, Gilbert, Ian H.
Published in ACS omega (11.04.2023)
Published in ACS omega (11.04.2023)
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Correction for Arora et al., "Respiratory Flexibility in Response to Inhibition of Cytochrome c Oxidase in Mycobacterium tuberculosis "
Arora, Kriti, Ochoa-Montaño, Bernardo, Tsang, Patricia S, Blundell, Tom L, Dawes, Stephanie S, Mizrahi, Valerie, Bayliss, Tracy, Mackenzie, Claire J, Cleghorn, Laura A T, Ray, Peter C, Wyatt, Paul G, Uh, Eugene, Lee, Jinwoo, Barry, 3rd, Clifton E, Boshoff, Helena I
Published in Antimicrobial agents and chemotherapy (01.09.2017)
Published in Antimicrobial agents and chemotherapy (01.09.2017)
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Discovery of an Allosteric Binding Site in Kinetoplastid Methionyl-tRNA Synthetase
Torrie, Leah S, Robinson, David A, Thomas, Michael G, Hobrath, Judith V, Shepherd, Sharon M, Post, John M, Ko, Eun-Jung, Ferreira, Rafael Alves, Mackenzie, Claire J, Wrobel, Karolina, Edwards, Darren P, Gilbert, Ian H, Gray, David W, Fairlamb, Alan H, De Rycker, Manu
Published in ACS infectious diseases (08.05.2020)
Published in ACS infectious diseases (08.05.2020)
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Identification of 6-amino-1H-pyrazolo[3,4-d]pyrimidines with in vivo efficacy against visceral leishmaniasis
Thomas, Michael G, De Rycker, Manu, Ajakane, Myriam, Crouch, Sabrinia D, Campbell, Lorna, Daugan, Alain, Fra, Gloria, Guerrero, César, Mackenzie, Claire J, MacLean, Lorna, Manthri, Sujatha, Martin, Franck, Norval, Suzanne, Osuna-Cabello, Maria, Riley, Jennifer, Shishikura, Yoko, Miguel-Siles, Juan, Simeons, Frederick R C, Stojanovski, Laste, Thomas, John, Thompson, Stephen, Velasco, Raul F, Fiandor, Jose M, Wyatt, Paul G, Read, Kevin D, Gilbert, Ian H, Miles, Timothy J
Published in MedChemComm (01.10.2020)
Published in MedChemComm (01.10.2020)
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Identification of 6-amino-1 H -pyrazolo[3,4- d ]pyrimidines with in vivo efficacy against visceral leishmaniasis
Thomas, Michael G, De Rycker, Manu, Ajakane, Myriam, Crouch, Sabrinia D, Campbell, Lorna, Daugan, Alain, Fra, Gloria, Guerrero, César, Mackenzie, Claire J, MacLean, Lorna, Manthri, Sujatha, Martin, Franck, Norval, Suzanne, Osuna-Cabello, Maria, Riley, Jennifer, Shishikura, Yoko, Miguel-Siles, Juan, Simeons, Frederick R C, Stojanovski, Laste, Thomas, John, Thompson, Stephen, Velasco, Raul F, Fiandor, Jose M, Wyatt, Paul G, Read, Kevin D, Gilbert, Ian H, Miles, Timothy J
Published in RSC medicinal chemistry (01.10.2020)
Published in RSC medicinal chemistry (01.10.2020)
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Identification of GSK3186899/DDD853651 as a Preclinical Development Candidate for the Treatment of Visceral Leishmaniasis
Thomas, Michael G, De Rycker, Manu, Ajakane, Myriam, Albrecht, Sébastian, Álvarez-Pedraglio, Ana Isabel, Boesche, Markus, Brand, Stephen, Campbell, Lorna, Cantizani-Perez, Juan, Cleghorn, Laura A.T, Copley, Royston C.B, Crouch, Sabrinia D, Daugan, Alain, Drewes, Gerard, Ferrer, Santiago, Ghidelli-Disse, Sonja, Gonzalez, Silvia, Gresham, Stephanie L, Hill, Alan P, Hindley, Sean J, Lowe, Rhiannon M, MacKenzie, Claire J, MacLean, Lorna, Manthri, Sujatha, Martin, Franck, Miguel-Siles, Juan, Nguyen, Van Loc, Norval, Suzanne, Osuna-Cabello, Maria, Woodland, Andrew, Patterson, Stephen, Pena, Imanol, Quesada-Campos, Maria Teresa, Reid, Iain H, Revill, Charlotte, Riley, Jennifer, Ruiz-Gomez, Jose Ramon, Shishikura, Yoko, Simeons, Frederick R.C, Smith, Alasdair, Smith, Victoria C, Spinks, Daniel, Stojanovski, Laste, Thomas, John, Thompson, Stephen, Underwood, Tim, Gray, David W, Fiandor, Jose M, Gilbert, Ian H, Wyatt, Paul G, Read, Kevin D, Miles, Timothy J
Published in Journal of medicinal chemistry (14.02.2019)
Published in Journal of medicinal chemistry (14.02.2019)
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Essential but Not Vulnerable: Indazole Sulfonamides Targeting Inosine Monophosphate Dehydrogenase as Potential Leads against Mycobacterium tuberculosis
Park, Yumi, Pacitto, Angela, Bayliss, Tracy, Cleghorn, Laura A. T, Wang, Zhe, Hartman, Travis, Arora, Kriti, Ioerger, Thomas R, Sacchettini, Jim, Rizzi, Menico, Donini, Stefano, Blundell, Tom L, Ascher, David B, Rhee, Kyu, Breda, Ardala, Zhou, Nian, Dartois, Veronique, Jonnala, Surendranadha Reddy, Via, Laura E, Mizrahi, Valerie, Epemolu, Ola, Stojanovski, Laste, Simeons, Fred, Osuna-Cabello, Maria, Ellis, Lucy, MacKenzie, Claire J, Smith, Alasdair R. C, Davis, Susan H, Murugesan, Dinakaran, Buchanan, Kirsteen I, Turner, Penelope A, Huggett, Margaret, Zuccotto, Fabio, Rebollo-Lopez, Maria Jose, Lafuente-Monasterio, Maria Jose, Sanz, Olalla, Diaz, Gracia Santos, Lelièvre, Joël, Ballell, Lluis, Selenski, Carolyn, Axtman, Matthew, Ghidelli-Disse, Sonja, Pflaumer, Hannah, Bösche, Markus, Drewes, Gerard, Freiberg, Gail M, Kurnick, Matthew D, Srikumaran, Myron, Kempf, Dale J, Green, Simon R, Ray, Peter C, Read, Kevin, Wyatt, Paul, Barry, Clifton E, Boshoff, Helena I
Published in ACS infectious diseases (13.01.2017)
Published in ACS infectious diseases (13.01.2017)
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Journal Article
Identification of 6-amino-1-pyrazolo[3,4-]pyrimidines with efficacy against visceral leishmaniasis
Thomas, Michael G, De Rycker, Manu, Ajakane, Myriam, Crouch, Sabrinia D, Campbell, Lorna, Daugan, Alain, Fra, Gloria, Guerrero, César, Mackenzie, Claire J, MacLean, Lorna, Manthri, Sujatha, Martin, Franck, Norval, Suzanne, Osuna-Cabello, Maria, Riley, Jennifer, Shishikura, Yoko, Miguel-Siles, Juan, Simeons, Frederick R. C, Stojanovski, Laste, Thomas, John, Thompson, Stephen, Velasco, Raul F, Fiandor, Jose M, Wyatt, Paul G, Read, Kevin D, Gilbert, Ian H, Miles, Timothy J
Published in RSC medicinal chemistry (21.10.2020)
Published in RSC medicinal chemistry (21.10.2020)
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Identification of 6-amino-1H-pyrazolo[3,4-d]pyrimidines with in vivo efficacy against visceral leishmaniasis† †Electronic supplementary information (ESI) available. See DOI: 10.1039/d0md00203h
Thomas, Michael G., De Rycker, Manu, Ajakane, Myriam, Crouch, Sabrinia D., Campbell, Lorna, Daugan, Alain, Fra, Gloria, Guerrero, César, Mackenzie, Claire J., MacLean, Lorna, Manthri, Sujatha, Martin, Franck, Norval, Suzanne, Osuna-Cabello, Maria, Riley, Jennifer, Shishikura, Yoko, Miguel-Siles, Juan, Simeons, Frederick R. C., Stojanovski, Laste, Thomas, John, Thompson, Stephen, Velasco, Raul F., Fiandor, Jose M., Wyatt, Paul G., Read, Kevin D., Gilbert, Ian H., Miles, Timothy J.
Published in RSC medicinal chemistry (06.08.2020)
Published in RSC medicinal chemistry (06.08.2020)
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Application of an NMR/crystallography fragment screening platform for the assessment and rapid discovery of new HIV-CA binding fragments
Lang, Stuart, Fletcher, Dan A, Alain-Pierre Petit, Luise, Nicola, Fyfe, Paul K, Zuccotto, Fabio, Porter, David, Hope, Anthony, Bellany, Fiona, Kerr, Catrina, Mackenzie, Claire J, Wyatt, Paul G, Gray, David W
Published in bioRxiv (15.12.2023)
Published in bioRxiv (15.12.2023)
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