Synthesis and biological evaluation of Doxorubicin-containing conjugate targeting PSMA
Ivanenkov, Yan A., Machulkin, Alexey E., Garanina, Anastasia S., Skvortsov, Dmitry A., Uspenskaya, Anastasia A., Deyneka, Ekaterina V., Trofimenko, Alexander V., Beloglazkina, Elena K., Zyk, Nikolay V., Koteliansky, Victor E, Bezrukov, Dmitry S., Aladinskaya, Anastasia V., Vorobyeva, Nataliya S., Puchinina, Maria M., Riabykh, Grigory K., Sofronova, Alina A., Malyshev, Alexander S., Majouga, Alexander G.
Published in Bioorganic & medicinal chemistry letters (15.05.2019)
Published in Bioorganic & medicinal chemistry letters (15.05.2019)
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Bifunctional Magnetite–Gold Nanoparticles for Magneto-Mechanical Actuation and Cancer Cell Destruction
Garanina, Anastasiia S, Efremova, Maria V, Machulkin, Alexey E, Lyubin, Evgeny V, Vorobyeva, Natalia S, Zhironkina, Oxana A, Strelkova, Olga S, Kireev, Igor I, Alieva, Irina B, Uzbekov, Rustem E, Agafonov, Viatcheslav N, Shchetinin, Igor V, Fedyanin, Andrey A, Erofeev, Alexander S, Gorelkin, Peter V, Korchev, Yuri E, Savchenko, Alexander G, Abakumov, Maxim A
Published in Magnetochemistry (01.12.2022)
Published in Magnetochemistry (01.12.2022)
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Large-scale High-throughput Screening Revealed 5'-(carbonylamino)-2,3'- bithiophene-4'-carboxylate as Novel Template for Antibacterial Agents
Ivanenkov, Yan A, Yamidanov, Renat S, Osterman, Ilya A, Sergiev, Petr V, Aladinskiy, Vladimir A, Aladinskaya, Anastasia V, Terentiev, Victor A, Veselov, Mark S, Ayginin, Andrey A, Skvortsov, Dmitry A, Komarova, Katerina S, Zagribelnyy, Bogdan A, Baimiev, Alexey Kh, Shvetc, Kseniya Yu, Baimiev, Andrey Kh, Sofronova, Alina A, Machulkin, Alexey E, Petrov, Rostislav A, Zainullina, Liana F, Maximova, Marina A, Zileeva, Zulfiya R, Vakhitova, Yulia V, Bezrukov, Dmitry S, Puchinina, Maria M, Dontsova, Olga A
Published in Current drug discovery technologies (2020)
Published in Current drug discovery technologies (2020)
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Synthesis and biological evaluation of PSMA-targeting paclitaxel conjugates
Machulkin, Alexey E., Skvortsov, Dmitry A., Ivanenkov, Yan A., Ber, Anton P., Kavalchuk, Mikhail V., Aladinskaya, Anastasia V., Uspenskaya, Anastasia A., Shafikov, Radik R., Plotnikova, Ekaterina A., Yakubovskaya, Raisa I., Nimenko, Ekaterina A., Zyk, Nikolay U., Beloglazkina, Elena K., Zyk, Nikolay V., Koteliansky, Victor E, Majouga, Alexander G.
Published in Bioorganic & medicinal chemistry letters (15.08.2019)
Published in Bioorganic & medicinal chemistry letters (15.08.2019)
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Small-molecule PSMA ligands. Current state, SAR and perspectives
Machulkin, Alexey E., Ivanenkov, Yan A., Aladinskaya, Anastasia V., Veselov, Mark S., Aladinskiy, Vladimir A., Beloglazkina, Elena K., Koteliansky, Victor E., Shakhbazyan, Artem G., Sandulenko, Yuri B., Majouga, Alexander G.
Published in Journal of drug targeting (13.09.2016)
Published in Journal of drug targeting (13.09.2016)
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Design, synthesis and biological evaluation of novel potent MDM2/p53 small-molecule inhibitors
Ivanenkov, Yan A., Vasilevski, Sergei V., Beloglazkina, Elena K., Kukushkin, Maksim E., Machulkin, Alexey E., Veselov, Mark S., Chufarova, Nina V., Chernyaginab, Elizaveta S., Vanzcool, Anton S., Zyk, Nikolay V., Skvortsov, Dmitry A., Khutornenko, Anastasia A., Rusanov, Alexander L., Tonevitsky, Alexander G., Dontsova, Olga A., Majouga, Alexander G.
Published in Bioorganic & medicinal chemistry letters (15.01.2015)
Published in Bioorganic & medicinal chemistry letters (15.01.2015)
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Journal Article
Corrigendum to ‘Synthesis and biological evaluation of Doxorubicin-containing conjugate targeting PSMA’ [Bioor. Med. Chem. Lett. 29/10 (2019) 1246–1255]
Ivanenkov, Yan A., Machulkin, Alexey E., Garanina, Anastasia S., Skvortsov, Dmitry A., Uspenskaya, Anastasia A., Deyneka, Ekaterina V., Trofimenko, Alexander V., Beloglazkina, Elena K., Zyk, Nikolay V., Koteliansky, Victor E., Bezrukov, Dmitry S., Aladinskaya, Anastasia V., Vorobyeva, Nataliya S., Puchinina, Maria M., Ryabykh, Grigory K., Sofronova, Alina A., Malyshev, Alexander S., Majouga, Alexander G.
Published in Bioorganic & medicinal chemistry letters (01.07.2019)
Published in Bioorganic & medicinal chemistry letters (01.07.2019)
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Journal Article
2-Pyrazol-1-yl-thiazole derivatives as novel highly potent antibacterials
Ivanenkov, Yan A, Yamidanov, Renat S, Osterman, Ilya A, Sergiev, Petr V, Aladinskiy, Vladimir A, Aladinskaya, Anastasia V, Terentiev, Victor A, Veselov, Mark S, Ayginin, Andrey A, Skvortsov, Dmitry A, Komarova, Katerina S, Sadovnikov, Sergey V, Matniyazov, Rustam, Sofronova, Alina A, Malyshev, Alexander S, Machulkin, Alexey E, Petrov, Rostislav A, Lukianov, Dmitrii, Iarovenko, Svetlana, Bezrukov, Dmitry S, Baymiev, Andrey Kh, Dontsova, Olga A
Published in Journal of antibiotics (01.11.2019)
Published in Journal of antibiotics (01.11.2019)
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Identification of pyrrolo-pyridine derivatives as novel class of antibacterials
Veselov, Mark S., Ivanenkov, Yan A., Yamidanov, Renat S., Osterman, Ilya A., Sergiev, Petr V., Aladinskiy, Vladimir A., Aladinskaya, Anastasia V., Terentiev, Victor A., Ayginin, Andrey A., Skvortsov, Dmitry A., Komarova, Katerina S., Chemeris, Alexey V., Baimiev, Alexey Kh, Sofronova, Alina A., Machulkin, Alexey E., Petrov, Rostislav A., Maklakova, Svetlana Yu, Bezrukov, Dmitry S., Filkov, Gleb I., Zainullina, Liana F., Maximova, Marina A., Zileeva, Zulfiya R., Kartsev, Victor G., Vakhitova, Yulia V., Dontsova, Olga A.
Published in Molecular diversity (01.02.2020)
Published in Molecular diversity (01.02.2020)
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Journal Article
Identification of N-Substituted Triazolo-azetidines as Novel Antibacterials using pDualrep2 HTS Platform
Ivanenkov, Yan A, Yamidanov, Renat S, Osterman, Ilya A, Sergiev, Petr V, Aladinskiy, Vladimir A, Aladinskaya, Anastasia V, Terentiev, Victor A, Veselov, Mark S, Ayginin, Andrey A, Skvortsov, Dmitry A, Komarova, Katerina S, Chemeris, Alexey V, Baimiev, Alexey Kh, Sofronova, Alina A, Malyshev, Alexander S, Machulkin, Alexey E, Petrov, Rostislav A, Bezrukov, Dmitry S, Filkov, Gleb I, Puchinina, Maria M, Zainullina, Liana F, Maximova, Marina A, Zileeva, Zulfiya R, Vakhitova, Yulia V, Dontsova, Olga A
Published in Combinatorial chemistry & high throughput screening (08.08.2019)
Published in Combinatorial chemistry & high throughput screening (08.08.2019)
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Journal Article
Substituted Furanocoumarins as Novel Class of Antibacterial Translation Inhibitors
Ivanenkov, Yan A, Yamidanov, Renat S, Osterman, Ilya A, Sergiev, Petr V, Ayginin, Andrey A, Aladinskiy, Vladimir A, Aladinskaya, Anastasia V, Terentiev, Victor A, Veselov, Mark S, Skvortsov, Dmitry A, Komarova, Katerina S, Chemeris, Alexey V, Zainullina, Liana F, Maximova, Marina A, Zileeva, Zulfiya R, Vakhitova, Yulia V, Baymiev, Alexey Kh, Baymiev, Andrey Kh, Sofronova, Alina A, Machulkin, Alexey E, Petrov, Rostislav A, Bezrukov, Dmitry S, Puchinina, Maria M, Lukianov, Dmitrii A, Dontsova, Olga A
Published in Combinatorial chemistry & high throughput screening (01.01.2019)
Published in Combinatorial chemistry & high throughput screening (01.01.2019)
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Journal Article
Influence of the dipeptide linker configuration on the activity of PSMA ligands
Uspenskaya, Anastasiya A., Machulkin, Alexey E., Nimenko, Ekaterina A., Shafikov, Radik R., Petrov, Stanislav A., Skvortsov, Dmitry A., Beloglazkina, Elena K., Majouga, Alexander G.
Published in Mendeleev communications (01.11.2020)
Published in Mendeleev communications (01.11.2020)
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