Putative ligand binding sites of two functionally characterized bark beetle odorant receptors
Yuvaraj, Jothi K, Roberts, Rebecca E, Sonntag, Yonathan, Hou, Xiao-Qing, Grosse-Wilde, Ewald, Machara, Aleš, Zhang, Dan-Dan, Hansson, Bill S, Johanson, Urban, Löfstedt, Christer, Andersson, Martin N
Published in BMC biology (26.01.2021)
Published in BMC biology (26.01.2021)
Get full text
Journal Article
Unraveling the anti-influenza effect of flavonoids: Experimental validation of luteolin and its congeners as potent influenza endonuclease inhibitors
Zima, Václav, Radilová, Kateřina, Kožíšek, Milan, Albiñana, Carlos Berenguer, Karlukova, Elena, Brynda, Jiří, Fanfrlík, Jindřich, Flieger, Miroslav, Hodek, Jan, Weber, Jan, Majer, Pavel, Konvalinka, Jan, Machara, Aleš
Published in European journal of medicinal chemistry (15.12.2020)
Published in European journal of medicinal chemistry (15.12.2020)
Get full text
Journal Article
Synthesis and In Vitro Evaluation of C-7 and C-8 Luteolin Derivatives as Influenza Endonuclease Inhibitors
Reiberger, Robert, Radilová, Kateřina, Kráľ, Michal, Zima, Václav, Majer, Pavel, Brynda, Jiří, Dračínský, Martin, Konvalinka, Jan, Kožíšek, Milan, Machara, Aleš
Published in International journal of molecular sciences (20.07.2021)
Published in International journal of molecular sciences (20.07.2021)
Get full text
Journal Article
Identification and Enantiodivergent Synthesis of (5Z,9S)‑Tetradec-5-en-9-olide, a Queen-Specific Volatile of the Termite Silvestritermes minutus
Machara, Aleš, Křivánek, Jan, Dolejšová, Klára, Havlíčková, Jana, Bednárová, Lucie, Hanus, Robert, Majer, Pavel, Kyjaková, Pavlína
Published in Journal of natural products (Washington, D.C.) (26.10.2018)
Published in Journal of natural products (Washington, D.C.) (26.10.2018)
Get full text
Journal Article
structural characterization of the interaction between the C-terminal domain of the influenza polymerase PA subunit and an optimized small peptide inhibitor
Hejdánek, Jakub, Radilová, Kateřina, Pachl, Petr, Hodek, Jan, Machara, Aleš, Weber, Jan, Řezáčová, Pavlína, Konvalinka, Jan, Kožíšek, Milan
Published in Antiviral research (01.01.2021)
Published in Antiviral research (01.01.2021)
Get full text
Journal Article
Specific Inhibitors of HIV Capsid Assembly Binding to the C‑Terminal Domain of the Capsid Protein: Evaluation of 2‑Arylquinazolines as Potential Antiviral Compounds
Machara, Aleš, Lux, Vanda, Kožíšek, Milan, Grantz Šašková, Klára, Štěpánek, Ondřej, Kotora, Martin, Parkan, Kamil, Pávová, Marcela, Glass, Bärbel, Sehr, Peter, Lewis, Joe, Müller, Barbara, Kräusslich, Hans-Georg, Konvalinka, Jan
Published in Journal of medicinal chemistry (28.01.2016)
Published in Journal of medicinal chemistry (28.01.2016)
Get full text
Journal Article
Characterization of Triacylglycerol Estolide Isomers Using High-Resolution Tandem Mass Spectrometry with Nanoelectrospray Ionization
Cudlman, Lukáš, Machara, Aleš, Vrkoslav, Vladimír, Polášek, Miroslav, Bosáková, Zuzana, Blanksby, Stephen J, Cvačka, Josef
Published in Biomolecules (Basel, Switzerland) (01.03.2023)
Published in Biomolecules (Basel, Switzerland) (01.03.2023)
Get full text
Journal Article
Kinetic, Thermodynamic, and Structural Analysis of Drug Resistance Mutations in Neuraminidase from the 2009 Pandemic Influenza Virus
Pokorná, Jana, Pachl, Petr, Karlukova, Elena, Hejdánek, Jakub, Řezáčová, Pavlína, Machara, Aleš, Hudlický, Jason, Konvalinka, Jan, Kožíšek, Milan
Published in Viruses (21.06.2018)
Published in Viruses (21.06.2018)
Get full text
Journal Article
DNA-linked inhibitor antibody assay (DIANA) as a new method for screening influenza neuraminidase inhibitors
Kožíšek, Milan, Navrátil, Václav, Rojíková, Kateřina, Pokorná, Jana, Berenguer Albiñana, Carlos, Pachl, Petr, Zemanová, Jitka, Machara, Aleš, Šácha, Pavel, Hudlický, Jason, Císařová, Ivana, Řezáčová, Pavlína, Konvalinka, Jan
Published in Biochemical journal (10.12.2018)
Published in Biochemical journal (10.12.2018)
Get more information
Journal Article
Understanding desaturation/hydroxylation activity of castor stearoyl Δ9-Desaturase through rational mutagenesis
Tupec, Michal, Culka, Martin, Machara, Aleš, Macháček, Stanislav, Bím, Daniel, Svatoš, Aleš, Rulíšek, Lubomír, Pichová, Iva
Published in Computational and structural biotechnology journal (01.01.2022)
Published in Computational and structural biotechnology journal (01.01.2022)
Get full text
Journal Article
Synthesis and evaluation of 2-pyridinylpyrimidines as inhibitors of HIV-1 structural protein assembly
Kožíšek, Milan, Štěpánek, Ondřej, Parkan, Kamil, Berenguer Albiñana, Carlos, Pávová, Marcela, Weber, Jan, Krӓusslich, Hans-Georg, Konvalinka, Jan, Machara, Aleš
Published in Bioorganic & medicinal chemistry letters (01.08.2016)
Published in Bioorganic & medicinal chemistry letters (01.08.2016)
Get full text
Journal Article
Evolution of Linoleic Acid Biosynthesis Paved the Way for Ecological Success of Termites
Macháček, Stanislav, Tupec, Michal, Horáček, Natan, Halmová, Martina, Roy, Amit, Machara, Aleš, Kyjaková, Pavlína, Lukšan, Ondřej, Pichová, Iva, Hanus, Robert
Published in Molecular biology and evolution (04.04.2023)
Published in Molecular biology and evolution (04.04.2023)
Get full text
Journal Article
Palladium(II) Complexes of Homologated Ferrocene Phosphanylether and Thioether Ligands
Zábranský, Martin, Machara, Aleš, Císařová, Ivana, Štěpnička, Petr
Published in European journal of inorganic chemistry (09.11.2017)
Published in European journal of inorganic chemistry (09.11.2017)
Get full text
Journal Article
Thermodynamic and structural characterization of an optimized peptide-based inhibitor of the influenza polymerase PA-PB1 subunit interaction
Radilová, Kateřina, Zima, Václav, Kráľ, Michal, Machara, Aleš, Majer, Pavel, Hodek, Jan, Weber, Jan, Brynda, Jiří, Strmeň, Timotej, Konvalinka, Jan, Kožíšek, Milan
Published in Antiviral research (01.12.2022)
Published in Antiviral research (01.12.2022)
Get full text
Journal Article
Female melon fruit flies, Zeugodacus cucurbitae, are attracted to a synthetic chemical blend based on male epicuticular components
Jacob, Vincent, Ramiaranjatovo, Gaëlle, Persyn, Emma, Machara, Aleš, Kyjaková, Pavlína, Atiama-Nurbel, Toulassi, Pompeiano, Antonio, Benelli, Giovanni, De Meyer, Marc, Vaníčková, Lucie
Published in Journal of pest science (01.06.2024)
Published in Journal of pest science (01.06.2024)
Get full text
Journal Article
Investigation of flexibility of neuraminidase 150-loop using tamiflu derivatives in influenza A viruses H1N1 and H5N1
Zima, Václav, Albiñana, Carlos Berenguer, Rojíková, Kateřina, Pokorná, Jana, Pachl, Petr, Řezáčová, Pavlína, Hudlicky, Jason, Navrátil, Václav, Majer, Pavel, Konvalinka, Jan, Kožíšek, Milan, Machara, Aleš
Published in Bioorganic & medicinal chemistry (01.07.2019)
Published in Bioorganic & medicinal chemistry (01.07.2019)
Get full text
Journal Article