Search Results - "MacKenny, Malcolm" :: K.UTB vyhledávací portál | TBU Library Retrieval Portal

Design and synthesis of morpholine derivatives. SAR for dual serotonin & noradrenaline reuptake inhibition

Design and synthesis of morpholine derivatives. SAR for dual serotonin & noradrenaline reuptake inhibition

by Fish, Paul V., Deur, Christopher, Gan, Xinmin, Greene, Keri, Hoople, David, Mackenny, Malcolm, Para, Kimberly S., Reeves, Keith, Ryckmans, Thomas, Stiff, Cory, Stobie, Alan, Wakenhut, Florian, Whitlock, Gavin A.
Published in Bioorganic & medicinal chemistry (15.04.2008)

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Journal Article

Synthetic Studies on a Nonsteroidal Progesterone Metabolite: Regioselective N-Alkylation of an Activated Pyrazole

Synthetic Studies on a Nonsteroidal Progesterone Metabolite: Regioselective N-Alkylation of an Activated Pyrazole

by Bradley, Paul A., de Koning, Pieter D., Gibson, Karl R., Lecouturier, Yann C., MacKenny, Malcolm C., Morao, Inaki, Poinsard, Cedric, Underwood, Toby J.
Published in Synlett (01.04.2010)

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Journal Article

Serendipity in drug-discovery: A new series of 2-(benzyloxy)benzamides as TRPM8 antagonists

Serendipity in drug-discovery: A new series of 2-(benzyloxy)benzamides as TRPM8 antagonists

by Brown, Alan, Ellis, David, Favor, David A., Kirkup, Tony, Klute, Wolfgang, MacKenny, Malcolm, McMurray, Gordon, Stennett, Adam
Published in Bioorganic & medicinal chemistry letters (15.11.2013)

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Journal Article

Sulfonamides as selective oestrogen receptor β agonists

Sulfonamides as selective oestrogen receptor β agonists

by Roberts, Lee R., Armor, Duncan, Barker, Carolyn, Bent, Andrew, Bess, Kirstin, Brown, Alan, Favor, David A., Ellis, David, Irving, Stephen L., MacKenny, Malcolm, Phillips, Chris, Pullen, Nick, Stennett, Adam, Strand, Linda, Styles, Michelle
Published in Bioorganic & medicinal chemistry letters (01.10.2011)

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Journal Article

Design and optimization of selective serotonin re-uptake inhibitors with high synthetic accessibility Part 1

Design and optimization of selective serotonin re-uptake inhibitors with high synthetic accessibility Part 1

by Andrews, Mark, Brown, Alan, Chiva, Jean-Yves, Fradet, David, Gordon, David, Lansdell, Mark, MacKenny, Malcolm
Published in Bioorganic & medicinal chemistry letters (15.04.2009)

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Journal Article

Design and optimisation of selective serotonin re-uptake inhibitors with high synthetic accessibility: Part 2

Design and optimisation of selective serotonin re-uptake inhibitors with high synthetic accessibility: Part 2

by Andrews, Mark, Brown, Alan, Chiva, Jean-Yves, Fradet, David, Gordon, David, Lansdell, Mark, MacKenny, Malcolm
Published in Bioorganic & medicinal chemistry letters (15.10.2009)

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Journal Article

Sulfonamides as selective oestrogen receptor [beta] agonists

Sulfonamides as selective oestrogen receptor [beta] agonists

by Roberts, Lee R, Armor, Duncan, Barker, Carolyn, Bent, Andrew, Bess, Kirstin, Brown, Alan, Favor, David A, Ellis, David, Irving, Stephen L, MacKenny, Malcolm, Phillips, Chris, Pullen, Nick, Stennett, Adam, Strand, Linda, Styles, Michelle
Published in Bioorganic & medicinal chemistry letters (01.10.2011)

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Journal Article

Enantioselective synthesis of ( R)- and ( S)- N-Boc-morpholine-2-carboxylic acids by enzyme-catalyzed kinetic resolution: application to the synthesis of reboxetine analogs

Enantioselective synthesis of ( R)- and ( S)- N-Boc-morpholine-2-carboxylic acids by enzyme-catalyzed kinetic resolution: application to the synthesis of reboxetine analogs

by Fish, Paul V., Mackenny, Malcolm, Bish, Gerwyn, Buxton, Timothy, Cave, Russell, Drouard, David, Hoople, David, Jessiman, Alan, Miller, Duncan, Pasquinet, Christelle, Patel, Bhairavi, Reeves, Keith, Ryckmans, Thomas, Skerten, Melanie, Wakenhut, Florian
Published in Tetrahedron letters (28.01.2009)

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Journal Article

Designing rapid onset selective serotonin re-uptake inhibitors. Part 3: Site-directed metabolism as a strategy to avoid active circulating metabolites: Structure–activity relationships of (thioalkyl)phenoxy benzylamines

Designing rapid onset selective serotonin re-uptake inhibitors. Part 3: Site-directed metabolism as a strategy to avoid active circulating metabolites: Structure–activity relationships of (thioalkyl)phenoxy benzylamines

by Middleton, Donald S., Andrews, Mark, Glossop, Paul, Gymer, Geoffrey, Hepworth, David, Jessiman, Alan, Johnson, Patrick S., MacKenny, Malcolm, Stobie, Alan, Tang, Kim, Morgan, Paul, Jones, Barry
Published in Bioorganic & medicinal chemistry letters (01.10.2008)

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Journal Article

Designing rapid onset selective serotonin re-uptake inhibitors. 2: Structure–activity relationships of substituted (aryl)benzylamines

Designing rapid onset selective serotonin re-uptake inhibitors. 2: Structure–activity relationships of substituted (aryl)benzylamines

by Middleton, Donald S., Andrews, Mark, Glossop, Paul, Gymer, Geoffrey, Hepworth, David, Jessiman, Alan, Johnson, Patrick S., MacKenny, Malcolm, Pitcher, Michael J., Rooker, Tony, Stobie, Alan, Tang, Kim, Morgan, Paul
Published in Bioorganic & medicinal chemistry (15.07.2008)

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Journal Article

Designing rapid onset selective serotonin re-uptake inhibitors. Part 1: Structure–activity relationships of substituted (1 S,4 S)-4-(3,4-dichlorophenyl)- N-methyl-1,2,3,4-tetrahydro-1-naphthaleneamine

Designing rapid onset selective serotonin re-uptake inhibitors. Part 1: Structure–activity relationships of substituted (1 S,4 S)-4-(3,4-dichlorophenyl)- N-methyl-1,2,3,4-tetrahydro-1-naphthaleneamine

by Middleton, Donald S., Andrews, Mark, Glossop, Paul, Gymer, Geoffrey, Jessiman, Alan, Johnson, Patrick S., MacKenny, Malcolm, Pitcher, Michael J., Rooker, Tony, Stobie, Alan, Tang, Kim, Morgan, Paul
Published in Bioorganic & medicinal chemistry letters (01.03.2006)

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Journal Article

Facile decarboxylation of nitrobenzeneacetic acids as a convenient route to alkylnitrobenzenes

Facile decarboxylation of nitrobenzeneacetic acids as a convenient route to alkylnitrobenzenes

by Bull, DJ, Fray, MJ, Mackenny, MC, Malloy, KA
Published in Synlett (01.07.1996)

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Journal Article

Morpholine Compounds, Pharmaceutically Acceptable Salts Thereof, Pharmaceutical Compositions, and Methods Of Use Thereof

Morpholine Compounds, Pharmaceutically Acceptable Salts Thereof, Pharmaceutical Compositions, and Methods Of Use Thereof

by STOBIE ALAN, MACKENNY MALCOLM CHRISTIAN, WHITLOCK GAVIN ALISTAIR, FISH PAUL VINCENT, WAKENHUT FLORIAN
Year of Publication 03.06.2010

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Patent

MORPHOLINE COMPOUNDS

MORPHOLINE COMPOUNDS

by MACKENNY, MALCOLM CHRISTIAN, STOBIE, ALAN, WAKENHUT, FLORIAN, FISH, PAUL VINCENT, WHITLOCK, GAVIN ALISTAIR
Year of Publication 30.03.2010

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Patent

Morpholine compounds

Morpholine compounds

by MACKENNY, MALCOLM CHRISTIAN, STOBIE, ALAN, WAKENHUT, FLORIAN, FISH, PAUL VINCENT, WHITLOCK, GAVIN ALISTAIR
Year of Publication 27.11.2009

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Patent

MORPHOLINE COMPOUNDS

MORPHOLINE COMPOUNDS

by STOBIE ALAN, MACKENNY MALCOLM CHRISTIAN, WHITLOCK GAVIN ALISTAIR, FISH PAUL VINCENT, WAKENHUT FLORIAN
Year of Publication 10.06.2009

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Patent

MORPHOLINE COMPOUNDS

MORPHOLINE COMPOUNDS

by STOBIE ALAN, MACKENNY MALCOLM CHRISTIAN, WHITLOCK GAVIN ALISTAIR, FISH PAUL VINCENT, WAKENHUT FLORIAN
Year of Publication 15.01.2009

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Patent

MORPHOLINE COMPOUNDS

MORPHOLINE COMPOUNDS

by STOBIE ALAN, MACKENNY MALCOLM CHRISTIAN, WHITLOCK GAVIN ALISTAIR, FISH PAUL VINCENT, WAKENHUT FLORIAN
Year of Publication 15.01.2009

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Patent

MORPHOLINE COMPOUNDS

MORPHOLINE COMPOUNDS

by STOBIE ALAN, MACKENNY MALCOLM CHRISTIAN, WHITLOCK GAVIN ALISTAIR, FISH PAUL VINCENT, WAKENHUT FLORIAN
Year of Publication 15.01.2009

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Patent

MORPHOLINE COMPOUNDS

MORPHOLINE COMPOUNDS

by FISH, PAUL, VINCENT, WHITLOCK, GAVIN, ALISTAIR, STOBIE, ALAN, MACKENNY, MALCOLM, CHRISTIAN, WAKENHUT, FLORIAN
Year of Publication 25.11.2008

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Patent