MicroRNA-21 promotes fibrosis of the kidney by silencing metabolic pathways
Chau, B Nelson, Xin, Cuiyan, Hartner, Jochen, Ren, Shuyu, Castano, Ana P, Linn, Geoffrey, Li, Jian, Tran, Phong T, Kaimal, Vivek, Huang, Xinqiang, Chang, Aaron N, Li, Shenyang, Kalra, Aarti, Grafals, Monica, Portilla, Didier, MacKenna, Deidre A, Orkin, Stuart H, Duffield, Jeremy S
Published in Science translational medicine (15.02.2012)
Published in Science translational medicine (15.02.2012)
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Identification of 4‑(Aminomethyl)-6-(trifluoromethyl)-2-(phenoxy)pyridine Derivatives as Potent, Selective, and Orally Efficacious Inhibitors of the Copper-Dependent Amine Oxidase, Lysyl Oxidase-Like 2 (LOXL2)
Rowbottom, Martin W, Bain, Gretchen, Calderon, Imelda, Lasof, Taylor, Lonergan, David, Lai, Andiliy, Huang, Fei, Darlington, Janice, Prodanovich, Patricia, Santini, Angelina M, King, Christopher D, Goulet, Lance, Shannon, Kristen E, Ma, Gina L, Nguyen, Katherine, MacKenna, Deidre A, Evans, Jilly F, Hutchinson, John H
Published in Journal of medicinal chemistry (25.05.2017)
Published in Journal of medicinal chemistry (25.05.2017)
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Let-7 Coordinately Suppresses Components of the Amino Acid Sensing Pathway to Repress mTORC1 and Induce Autophagy
Dubinsky, Amy N., Dastidar, Somasish Ghosh, Hsu, Cynthia L., Zahra, Rabaab, Djakovic, Stevan N., Duarte, Sonia, Esau, Christine C., Spencer, Brian, Ashe, Travis D., Fischer, Kimberlee M., MacKenna, Deidre A., Sopher, Bryce L., Masliah, Eliezer, Gaasterland, Terry, Chau, B. Nelson, Pereira de Almeida, Luis, Morrison, Bradley E., La Spada, Albert R.
Published in Cell metabolism (07.10.2014)
Published in Cell metabolism (07.10.2014)
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Polysome shift assay for direct measurement of miRNA inhibition by anti-miRNA drugs
Androsavich, John R, Sobczynski, Daniel J, Liu, Xueqing, Pandya, Shweta, Kaimal, Vivek, Owen, Tate, Liu, Kai, MacKenna, Deidre A, Chau, B Nelson
Published in Nucleic acids research (29.01.2016)
Published in Nucleic acids research (29.01.2016)
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Liver-Targeted Drug Delivery Using HepDirect Prodrugs
Erion, Mark D, van Poelje, Paul D, Mackenna, Deidre A, Colby, Timothy J, Montag, Annika C, Fujitaki, James M, Linemeyer, David L, Bullough, David A
Published in The Journal of pharmacology and experimental therapeutics (01.02.2005)
Published in The Journal of pharmacology and experimental therapeutics (01.02.2005)
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Anti-microRNA-21 oligonucleotides prevent Alport nephropathy progression by stimulating metabolic pathways
Gomez, Ivan G, MacKenna, Deidre A, Johnson, Bryce G, Kaimal, Vivek, Roach, Allie M, Ren, Shuyu, Nakagawa, Naoki, Xin, Cuiyan, Newitt, Rick, Pandya, Shweta, Xia, Tai-He, Liu, Xueqing, Borza, Dorin-Bogdan, Grafals, Monica, Shankland, Stuart J, Himmelfarb, Jonathan, Portilla, Didier, Liu, Shiguang, Chau, B Nelson, Duffield, Jeremy S
Published in The Journal of clinical investigation (01.01.2015)
Published in The Journal of clinical investigation (01.01.2015)
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Lysyl oxidase like-2 contributes to renal fibrosis in Col4α3/Alport mice
Cosgrove, Dominic, Dufek, Brianna, Meehan, Daniel T., Delimont, Duane, Hartnett, Michael, Samuelson, Gina, Gratton, Michael Anne, Phillips, Grady, MacKenna, Deidre A., Bain, Gretchen
Published in Kidney international (01.08.2018)
Published in Kidney international (01.08.2018)
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A Potent and Selective AMPK Activator That Inhibits de Novo Lipogenesis
Gómez-Galeno, Jorge E, Dang, Qun, Nguyen, Thanh H, Boyer, Serge H, Grote, Matthew P, Sun, Zhili, Chen, Mingwei, Craigo, William A, van Poelje, Paul D, MacKenna, Deidre A, Cable, Edward E, Rolzin, Paul A, Finn, Patricia D, Chi, Bert, Linemeyer, David L, Hecker, Scott J, Erion, Mark D
Published in ACS medicinal chemistry letters (09.12.2010)
Published in ACS medicinal chemistry letters (09.12.2010)
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Synthesis and Characterization of a Novel Liver-Targeted Prodrug of Cytosine-1-β-d-arabinofuranoside Monophosphate for the Treatment of Hepatocellular Carcinoma
Boyer, Serge H, Sun, Zhili, Jiang, Hongjian, Esterbrook, Julie, Gómez-Galeno, Jorge E, Craigo, William, Reddy, K. Raja, Ugarkar, Bheemarao G, MacKenna, Deidre A, Erion, Mark D
Published in Journal of medicinal chemistry (28.12.2006)
Published in Journal of medicinal chemistry (28.12.2006)
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2 USES OF A LYSYL OXIDASE-LIKE 2 INHIBITOR
BAIN GRETCHEN, HUTCHINSON JOHN HOWARD, EVANS JILLIAN FRANCES, MACKENNA DEIDRE A
Year of Publication 29.11.2023
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Year of Publication 29.11.2023
Patent
Delivery of high levels of anti-proliferative nucleoside triphosphates to CYP3A-expressing cells as a potential treatment for hepatocellular carcinoma
MacKenna, Deidre A, Montag, Annika, Boyer, Serge H, Linemeyer, David L, Erion, Mark D
Published in Cancer chemotherapy and pharmacology (01.10.2009)
Published in Cancer chemotherapy and pharmacology (01.10.2009)
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Therapeutic modulation of microRNAs
Chau, B. Nelson, Esau, Christine C, MacKenna, Deidre A, Neben, Steve, Gibson, Neil W
Published in Drug discovery today. Therapeutic strategies (2013)
Published in Drug discovery today. Therapeutic strategies (2013)
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리실 옥시다제 유사 2 억제제의 용도
BAIN GRETCHEN, HUTCHINSON JOHN HOWARD, EVANS JILLIAN FRANCES, MACKENNA DEIDRE A
Year of Publication 11.06.2019
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Year of Publication 11.06.2019
Patent
Measurement of strain and analysis of stress in resting rat left ventricular myocardium
Omens, Jeffrey H., MacKenna, Deidre A., McCulloch, Andrew D.
Published in Journal of biomechanics (01.06.1993)
Published in Journal of biomechanics (01.06.1993)
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Journal Article
Lysyl oxidase like-2 contributes to renal fibrosis in Col4a3/Alport Mice
Cosgrove, Dominic, Dufek, Brianna, Meehan, Daniel T., Delimont, Duane, Hartnett, Michael, Samuelson, Gina, Gratton, Michael Anne, Phillips, Grady, MacKenna, Deidre A., Bain, Gretchen
Published in Kidney international (16.05.2018)
Published in Kidney international (16.05.2018)
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