Novel library synthesis of 3,4-disubstituted pyridin-2(1 H )-ones via cleavage of pyridine-2-oxy-7-azabenzotriazole ethers under ionic hydrogenation conditions at room temperature
Pierre, Romain, Brethon, Anne, Jacques, Sylvain A, Blond, Aurélie, Chambon, Sandrine, Talano, Sandrine, Raffin, Catherine, Musicki, Branislav, Bouix-Peter, Claire, Tomas, Loic, Ouvry, Gilles, Morgentin, Rémy, Hennequin, Laurent F, Harris, Craig S
Published in Beilstein journal of organic chemistry (2021)
Published in Beilstein journal of organic chemistry (2021)
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Synthesis and in vitro evaluation of novel highly potent coumarin inhibitors of gyrase B
Laurin, Patrick, Ferroud, Didier, Klich, Michel, Dupuis-Hamelin, Claudine, Mauvais, Pascale, Lassaigne, Patrice, Bonnefoy, Alain, Musicki, Branislav
Published in Bioorganic & medicinal chemistry letters (19.07.1999)
Published in Bioorganic & medicinal chemistry letters (19.07.1999)
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Journal Article
Discovery of phenoxyindazoles and phenylthioindazoles as RORγ inverse agonists
Ouvry, Gilles, Bouix-Peter, Claire, Ciesielski, Fabrice, Chantalat, Laurent, Christin, Olivier, Comino, Catherine, Duvert, Denis, Feret, Christophe, Harris, Craig S., Lamy, Laurent, Luzy, Anne-Pascale, Musicki, Branislav, Orfila, Danielle, Pascau, Jonathan, Parnet, Véronique, Perrin, Agnès, Pierre, Romain, Polge, Gaëlle, Raffin, Catherine, Rival, Yves, Taquet, Nathalie, Thoreau, Etienne, Hennequin, Laurent F.
Published in Bioorganic & medicinal chemistry letters (01.12.2016)
Published in Bioorganic & medicinal chemistry letters (01.12.2016)
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Journal Article
Route scouting and optimization of a potent sulfoximine-based inverse agonist of RORγt
Lafitte, Guillaume, Parnet, Veronique, Pierre, Romain, Raffin, Catherine, Vatinel, Rodolphe, Musicki, Branislav, Tomas, Loic, Bouix-Peter, Claire, Ouvry, Gilles, Daver, Sebastien, Arlabosse, Jean-Marie, Boiteau, Jean-Guy, Gerfaud, Thibaud, Harris, Craig S.
Published in Tetrahedron (04.10.2018)
Published in Tetrahedron (04.10.2018)
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Journal Article
Synthesis of the 4’-desmethoxy analogue of RU79115
Musicki, Branislav, Periers, Anne-Marie, Tessot, Nicole, Klich, Michel
Published in Journal of the Serbian Chemical Society (01.01.2004)
Published in Journal of the Serbian Chemical Society (01.01.2004)
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Journal Article
Sulfoximines as potent RORc inverse agonists
Ouvry, Gilles, Bihl, Franck, Bouix-Peter, Claire, Christin, Olivier, Defoin-Platel, Claire, Deret, Sophie, Feret, Christophe, Froude, David, Hacini-Rachinel, Feriel, Harris, Craig S., Hervouet, Catherine, Lafitte, Guillaume, Luzy, Anne-Pascale, Musicki, Branislav, Orfila, Danielle, Parnet, Veronique, Pascau, Coralie, Pascau, Jonathan, Pierre, Romain, Raffin, Catherine, Rossio, Patricia, Spiesse, Delphine, Taquet, Nathalie, Thoreau, Etienne, Vatinel, Rodolphe, Vial, Emmanuel, Hennequin, Laurent F.
Published in Bioorganic & medicinal chemistry letters (01.05.2018)
Published in Bioorganic & medicinal chemistry letters (01.05.2018)
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Journal Article
Early Development Scale-Up of a Novel CXCR Antagonist: Focus on Racemic and Stereoselective Routes of a Key Intermediate
Tabet, Samuel, Rodeville, Nicolas, Mathieu, Arnaud, Raffin, Catherine, Millois-Barbuis, Corinne, Musicki, Branislav, Muller, Franck, Gerfaud, Thibaud, Boiteau, Jean-Guy, Cardinaud, Isabelle
Published in Organic process research & development (15.12.2017)
Published in Organic process research & development (15.12.2017)
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Journal Article
Squaramides as novel class I and IIB histone deacetylase inhibitors for topical treatment of cutaneous t-cell lymphoma
Fournier, Jean-François, Bhurruth-Alcor, Yushma, Musicki, Branislav, Aubert, Jérome, Aurelly, Michèle, Bouix-Peter, Claire, Bouquet, Karinne, Chantalat, Laurent, Delorme, Marion, Drean, Bénédicte, Duvert, Gwenaelle, Fleury-Bregeot, Nicolas, Gauthier, Blanche, Grisendi, Karine, Harris, Craig S., Hennequin, Laurent F., Isabet, Tatiana, Joly, Florence, Lafitte, Guillaume, Millois, Corinne, Morgentin, Rémy, Pascau, Jonathan, Piwnica, David, Rival, Yves, Soulet, Catherine, Thoreau, Étienne, Tomas, Loïc
Published in Bioorganic & medicinal chemistry letters (15.09.2018)
Published in Bioorganic & medicinal chemistry letters (15.09.2018)
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Journal Article
Process Development and Good Manufacturing Practice Production of a Tyrosinase Inhibitor via Titanium-Mediated Coupling between Unprotected Resorcinols and Ketones
Gerfaud, Thibaud, Martin, Cédric, Bouquet, Karinne, Talano, Sandrine, Millois-Barbuis, Corinne, Musicki, Branislav, Boiteau, Jean-Guy, Cardinaud, Isabelle
Published in Organic process research & development (21.04.2017)
Published in Organic process research & development (21.04.2017)
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Journal Article
Sulfoximines as potent RORγ inverse agonists
Ouvry, Gilles, Bihl, Franck, Bouix-Peter, Claire, Christin, Olivier, Defoin-Platel, Claire, Deret, Sophie, Feret, Christophe, Froude, David, Hacini-Rachinel, Feriel, Harris, Craig S., Hervouet, Catherine, Lafitte, Guillaume, Luzy, Anne-Pascale, Musicki, Branislav, Orfila, Danielle, Parnet, Veronique, Pascau, Coralie, Pascau, Jonathan, Pierre, Romain, Raffin, Catherine, Rossio, Patricia, Spiesse, Delphine, Taquet, Nathalie, Thoreau, Etienne, Vatinel, Rodolphe, Vial, Emmanuel, Hennequin, Laurent F.
Published in Bioorganic & medicinal chemistry letters (01.05.2018)
Published in Bioorganic & medicinal chemistry letters (01.05.2018)
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Journal Article
A convenient one-pot synthesis of boroxoles from diboronic acid
Lafitte, Guillaume, Kunihiro, Kana, Bonneaud, Céline, Dréan, Bénédicte, Gaigne, Frédéric, Parnet, Véronique, Pierre, Romain, Raffin, Catherine, Vatinel, Rodolphe, Fournier, Jean-François, Musicki, Branislav, Ouvry, Gilles, Bouix-Peter, Claire, Tomas, Loic, Harris, Craig S.
Published in Tetrahedron letters (27.09.2017)
Published in Tetrahedron letters (27.09.2017)
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Journal Article
Discovery and Characterization of CD12681, a Potent ROR Inverse Agonist, Preclinical Candidate for the Topical Treatment of Psoriasis
Ouvry, Gilles, Atrux-Tallau, Nicolas, Bihl, Franck, Bondu, Aline, Bouix-Peter, Claire, Carlavan, Isabelle, Christin, Olivier, Cuadrado, Marie-Josee, Defoin-Platel, Claire, Deret, Sophie, Duvert, Denis, Feret, Christophe, Forissier, Mathieu, Fournier, Jean-Francois, Froude, David, Hacini-Rachinel, Feriel, Harris, Craig Steven, Hervouet, Catherine, Huguet, Helene, Lafitte, Guillaume, Luzy, Anne-Pascale, Musicki, Branislav, Orfila, Danielle, Ozello, Benjamin, Pascau, Coralie, Pascau, Jonathan, Parnet, Veronique, Peluchon, Guillaume, Pierre, Romain, Piwnica, David, Raffin, Catherine, Rossio, Patricia, Spiesse, Delphine, Taquet, Nathalie, Thoreau, Etienne, Vatinel, Rodolphe, Vial, Emmanuel, Hennequin, Laurent Francois
Published in ChemMedChem (20.02.2018)
Published in ChemMedChem (20.02.2018)
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Journal Article
Discovery and Characterization of CD12681, a Potent RORγ Inverse Agonist, Preclinical Candidate for the Topical Treatment of Psoriasis
Ouvry, Gilles, Atrux‐Tallau, Nicolas, Bihl, Franck, Bondu, Aline, Bouix‐Peter, Claire, Carlavan, Isabelle, Christin, Olivier, Cuadrado, Marie‐Josée, Defoin‐Platel, Claire, Deret, Sophie, Duvert, Denis, Feret, Christophe, Forissier, Mathieu, Fournier, Jean‐François, Froude, David, Hacini‐Rachinel, Fériel, Harris, Craig Steven, Hervouet, Catherine, Huguet, Hélène, Lafitte, Guillaume, Luzy, Anne‐Pascale, Musicki, Branislav, Orfila, Danielle, Ozello, Benjamin, Pascau, Coralie, Pascau, Jonathan, Parnet, Véronique, Peluchon, Guillaume, Pierre, Romain, Piwnica, David, Raffin, Catherine, Rossio, Patricia, Spiesse, Delphine, Taquet, Nathalie, Thoreau, Etienne, Vatinel, Rodolphe, Vial, Emmanuel, Hennequin, Laurent François
Published in ChemMedChem (20.02.2018)
Published in ChemMedChem (20.02.2018)
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Journal Article
Structure of the light emitter in krill (Euphausia pacifica) bioluminescence
Nakamura, Hideshi, Musicki, Branislav, Kishi, Yoshito, Shimomura, Osamu
Published in Journal of the American Chemical Society (01.04.1988)
Published in Journal of the American Chemical Society (01.04.1988)
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Journal Article
Improved antibacterial activities of coumarin antibiotics bearing 5′,5′-dialkylnoviose: biological activity of RU79115
Musicki, Branislav, Periers, Anne-Marie, Laurin, Patrick, Ferroud, Didier, Benedetti, Yannick, Lachaud, Sylvette, Chatreaux, Fabienne, Haesslein, Jean-Luc, Iltis, Alain, Pierre, Christine, Khider, Jean, Tessot, Nicole, Airault, Marlene, Demassey, Jacques, Dupuis-Hamelin, Claudine, Lassaigne, Patrice, Bonnefoy, Alain, Vicat, Pascale, Klich, Michel
Published in Bioorganic & medicinal chemistry letters (07.08.2000)
Published in Bioorganic & medicinal chemistry letters (07.08.2000)
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