The Discovery of Two Novel Classes of 5,5-Bicyclic Nucleoside-Derived PRMT5 Inhibitors for the Treatment of Cancer
Quiroz, Ryan V, Reutershan, Michael H, Schneider, Sebastian E, Sloman, David, Lacey, Brian M, Swalm, Brooke M, Yeung, Charles S, Gibeau, Craig, Spellman, Daniel S, Rankic, Danica A, Chen, Dapeng, Witter, David, Linn, Doug, Munsell, Erik, Feng, Guo, Xu, Haiyan, Hughes, Jonathan M. E, Lim, Jongwon, Saurí, Josep, Geddes, Kristin, Wan, Murray, Mansueto, My Sam, Follmer, Nicole E, Fier, Patrick S, Siliphaivanh, Phieng, Daublain, Pierre, Palte, Rachel L, Hayes, Robert P, Lee, Sandra, Kawamura, Shuhei, Silverman, Steven, Sanyal, Sulagna, Henderson, Timothy J, Ye, Yingchun, Gao, Yuanwei, Nicholson, Benjamin, Machacek, Michelle R
Published in Journal of medicinal chemistry (08.04.2021)
Published in Journal of medicinal chemistry (08.04.2021)
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Journal Article
PRMT5 INHIBITORS
HUANG, Chunhui, MACHACEK, Michelle, SCHNEIDER, Sebastian, KAWAMURA, Shuhei, WITTER, David, WAN, Murray
Year of Publication 11.05.2022
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Year of Publication 11.05.2022
Patent
PRMT5 INHIBITORS
Machacek, Michelle, Wan, Murray, Schneider, Sebastian, Kawamura, Shuhei, Witter, David, Huang, Chunhui
Year of Publication 07.10.2021
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Year of Publication 07.10.2021
Patent
PRMT5 INHIBITORS
HUANG, Chunhui, MACHACEK, Michelle, SCHNEIDER, Sebastian, KAWAMURA, Shuhei, WITTER, David, WAN, Murray
Year of Publication 16.06.2021
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Year of Publication 16.06.2021
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MACROCYCLIC PEPTIDES TARGETING KRAS
HUANG, Chunhui, PALANI, Anandan, ZHU, Yuping, BISWAS, Kaustav, TOMIYAMA, Tatsuya, KURASAKI, Haruaki, DING, Fa-Xiang, SUN, Zhongxiang, JOHNSTON, Jennifer Marie, LIN, Songnian, JOSIEN, Hubert, REID, Patrick C, WAN, Murray
Year of Publication 25.01.2024
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Year of Publication 25.01.2024
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CYCLIC PEPTIDES FOR INHIBITING TNF RECEPTOR 1 ACTIVITY
Zultanski, Susan L, Mapelli, Claudio, Kekec, Ahmet, Boyer, Nicolas C, Biswas, Kaustav, Frost, John R, Chau, Ryan, Sindhikara, Daniel J, Ding, Fa-Xiang, Siu, Tony, Pasquini, Nicolo Maria, Haidle, Andrew M, Rao, Ashwin U, Gambini, Luca, Wan, Murray, Lee, Hu-Jung Julie, Jewell, James P, Zhu, Yuping, Wuo, Michael, Tozzi, Roberta, Cash, Brandon D, Garrigou, Michael B, Lin, Songnian, Proietti, Giordano, Orvieto, Federica, Abate, Luigi
Year of Publication 29.08.2024
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Year of Publication 29.08.2024
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CYCLIC PEPTIDES FOR INHIBITING TNF RECEPTOR 1 ACTIVITY
HAIDLE, Andrew M, ZHU, Yuping, WUO, Michael, ZULTANSKI, Susan L, FROST, John R, JEWELL, James P, DING, Fa-Xiang, GARRIGOU, Michael B, LIN, Songnian, ORVIETO, Federica, GAMBINI, Luca, SIU, Tony, LEE, Hu-Jung Julie, BOYER, Nicolas C, BISWAS, Kaustav, TOZZI, Roberta, KEKEC, Ahmet, ABATE, Luigi, RAO, Ashwin U, PASQUINI, Nicolo Maria, CHAU, Ryan, CASH, Brandon D, SINDHIKARA, Daniel J, MAPELLI, Claudio, PROIETTI, Giordano, WAN, Murray
Year of Publication 08.08.2024
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Year of Publication 08.08.2024
Patent
PRMT5 INHIBITORS
HUANG, Chunhui, MACHACEK, Michelle, SCHNEIDER, Sebastian, KAWAMURA, Shuhei, WITTER, David, WAN, Murray
Year of Publication 13.02.2020
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Year of Publication 13.02.2020
Patent
PRMT5 INHIBITORS
Reutershan, Michael H, Machacek, Michelle, Wan, Murray, Quiroz, Ryan, Schneider, Sebastian, Paparin, Jean-Laurent, Fier, Patrick S, Gibeau, Craig, Kawamura, Shuhei, Candito, David A, Huang, Chunhui, Ye, Yingchun, Henderson, Timothy J, Silverman, Steven M, Sanyal, Sulagna, Sloman, David L, Yeung, Charles S, Siliphaivanh, Phieng, Hughes, Jonathan M. E, Witter, David, Rahali, Houcine
Year of Publication 17.11.2022
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Year of Publication 17.11.2022
Patent
INHIBITEURS DE PRMT5
YE, Yingchun, FIER, Patrick, S, REUTERSHAN, Michael, H, HUANG, Chunhui, YEUNG, Charles, S, MACHACEK, Michelle, SCHNEIDER, Sebastian, CANDITO, David, A, WITTER, David, SILIPHAIVANH, Phieng, SLOMAN, David, L, QUIROZ, Ryan, PAPARIN, Jean-Laurent, SANYAL, Sulagna, HUGHES, Jonathan, M., E, HENDERSON, Timothy, J, GIBEAU, Craig, KAWAMURA, Shuhei, SILVERMAN, Steven, M, RAHALI, Houcine, WAN, Murray
Year of Publication 11.05.2022
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Year of Publication 11.05.2022
Patent
PRMT5 INHIBITORS
YE, Yingchun, REUTERSHAN, Michael, H, FIER, Patrick, S, HUANG, Chunhui, YEUNG, Charles, S, MACHACEK, Michelle, SCHNEIDER, Sebastian, CANDITO, David, A, WITTER, David, SLOMAN, David, L, SILIPHAIVANH, Phieng, QUIROZ, Ryan, PAPARIN, Jean-Laurent, SANYAL, Sulagna, HUGHES, Jonathan, M., E, HENDERSON, Timothy, J, GIBEAU, Craig, KAWAMURA, Shuhei, SILVERMAN, Steven, M, RAHALI, Houcine, WAN, Murray
Year of Publication 11.05.2022
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Year of Publication 11.05.2022
Patent
PRMT5 INHIBITORS
YE, Yingchun, REUTERSHAN, Michael, H, FIER, Patrick, S, HUANG, Chunhui, YEUNG, Charles, S, MACHACEK, Michelle, SCHNEIDER, Sebastian, CANDITO, David, A, WITTER, David, SLOMAN, David, L, SILIPHAIVANH, Phieng, QUIROZ, Ryan, PAPARIN, Jean-Laurent, SANYAL, Sulagna, HUGHES, Jonathan, M., E, HENDERSON, Timothy, J, GIBEAU, Craig, KAWAMURA, Shuhei, SILVERMAN, Steven, M, RAHALI, Houcine, WAN, Murray
Year of Publication 16.06.2021
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Year of Publication 16.06.2021
Patent
PRMT5 inhibitors
Reutershan, Michael H, Machacek, Michelle, Wan, Murray, Quiroz, Ryan, Schneider, Sebastian, Fier, Patrick S, Gibeau, Craig, Kawamura, Shuhei, Candito, David A, Huang, Chunhui, Ye, Yingchun, Henderson, Timothy J, PAPARIN, Jean-Laurent, Silverman, Steven M, Sanyal, Sulagna, SLOMAN, David L, Yeung, Charles S, Hughes, Jonathan M, Siliphaivanh, Phieng, Witter, David, Rahali, Houcine
Year of Publication 25.02.2021
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Year of Publication 25.02.2021
Patent
PRMT5 INHIBITORS
PAPARIN, JEAN-LAURENT, RAHALI, HOUCINE, SILIPHAIVANH, PHIENG, QUIROZ, RYAN, FIER, PATRICK S, HENDERSON, TIMOTHY J, SCHNEIDER, SEBASTIAN, SANYAL, SULAGNA, GIBEAU, CRAIG, SILVERMAN, STEVEN M, KAWAMURA, SHUHEI, MACHACEK, MICHELLE, SLOMAN, DAVID L, WAN, MURRAY, WITTER, DAVID, HUANG, CHUNHUI, CANDITO, DAVID A, YE, YINGCHUN, REUTERSHAN, MICHAEL H, HUGHES, JONATHAN M. E, YEUNG, CHARLES S
Year of Publication 13.02.2020
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Year of Publication 13.02.2020
Patent
PRMT5 INHIBITORS
SILVERMAN, Steven, YE, Yingchun, HUANG, Chunhui, MACHACEK, Michelle, SCHNEIDER, Sebastian, HUGHES, Jonathan, FIER, Patrick, WITTER, David, SILIPHAIVANH, Phieng, QUIROZ, Ryan, PAPARIN, Jean-Laurent, SANYAL, Sulagna, CANDITO, David, REUTERSHAN, Michael, SLOMAN, David, GIBEAU, Craig, KAWAMURA, Shuhei, HENDERSON, Timothy, RAHALI, Houcine, WAN, Murray, YEUNG, Charles
Year of Publication 13.02.2020
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Year of Publication 13.02.2020
Patent
INIBIDORES DE PRMT5
DAVID L. SLOMAN, SULAGNA SANYAL, DAVID A. CANDITO, MICHAEL H. REUTERSHAN, JONATHAN M. E. HUGHES, CRAIG GIBEAU, MICHELLE MACHACEK, SEBASTIAN SCHNEIDER, STEVEN M. SILVERMAN, PATRICK S. FIER, PHIENG SILIPHAIVANH, JEAN-LAURENT PAPARIN, RYAN QUIROZ, TIMOTHY J. HENDERSON, HOUCINE RAHALI, DAVID WITTER, CHARLES S. YEUNG, CHUNHUI HUANG, MURRAY WAN, SHUHEI KAWAMURA, YINGCHUN YE
Year of Publication 07.02.2023
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Year of Publication 07.02.2023
Patent
PRMT5 INHIBITORS
HUGHES Jonathan, M., E, REUTERSHAN Michael, H, YE Yingchun, FIER Patrick, S, SLOMAN David, L, SILIPHAIVANH Phieng, PAPARIN Jean-laurent, SANYAL Sulagna, CANDITO David, A, MACHACEK Michelle, SCHNEIDER Sebastian, HUANG Chunhui, WITTER David, WAN Murray, HENDERSON Timothy, J, QUIROZ Ryan, GIBEAU Craig, KAWAMURA Shuhei, RAHALI Houcine, YEUNG Charles, S, SILVERMAN Steven, M
Year of Publication 15.07.2021
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Year of Publication 15.07.2021
Patent
PRMT5 INHIBITORS
CANDITO DAVID A, QUIROZ RYAN, WITTER DAVID, PAPARIN JEAN-LAURENT, HUGHES JONATHAN M E, HUANG CHUNHUI, SILIPHAIVANH PHIENG, HENDERSON TIMOTHY J, YE YINGCHUN, SCHNEIDER SEBASTIAN, KAWAMURA SHUHEI, YEUNG CHARLES S, FIER PATRICK S, WAN MURRAY, REUTERSHAN MICHAEL H, RAHALI HOUCINE, SANYAL SULAGNA, GIBEAU CRAIG, SILVERMAN STEVEN M, MACHACEK MICHELLE, SLOMAN DAVID L
Year of Publication 14.05.2021
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Year of Publication 14.05.2021
Patent
inibidores de prmt5
DAVID L. SLOMAN, DAVID A. CANDITO, SULAGNA SANYAL, MICHAEL H. REUTERSHAN, JONATHAN M. E. HUGHES, CRAIG GIBEAU, MICHELLE MACHACEK, SEBASTIAN SCHNEIDER, PATRICK S. FIER, STEVEN M. SILVERMAN, PHIENG SILIPHAIVANH, JEAN-LAURENT PAPARIN, HOUCINE RAHALI, RYAN QUIROZ, TIMOTHY J. HENDERSON, CHARLES S. YEUNG, DAVID WITTER, CHUNHUI HUANG, MURRAY WAN, SHUHEI KAWAMURA, YINGCHUN YE
Year of Publication 04.05.2021
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Year of Publication 04.05.2021
Patent