K858, a Novel Inhibitor of Mitotic Kinesin Eg5 and Antitumor Agent, Induces Cell Death in Cancer Cells
NAKAI, Ryuichiro, IIDA, Shin-Ichi, AKINAGA, Shiro, MURAKATA, Chikara, HONDA, Shinobu, NITTA, Masayuki, SAYA, Hideyuki, YAMASHITA, Yoshinori, TAKAHASHI, Takeshi, TSUJITA, Tetsuya, OKAMOTO, Seiho, TAKADA, Chie, AKASAKA, Kazuhito, ICHIKAWA, Shunji, ISHIDA, Hiroyuki, KUSAKA, Hideaki
Published in Cancer research (Chicago, Ill.) (01.05.2009)
Published in Cancer research (Chicago, Ill.) (01.05.2009)
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Rescue of hearing, auditory hair cells, and neurons by CEP-1347/KT7515, an inhibitor of c-Jun N-terminal kinase activation
Pirvola, U, Xing-Qun, L, Virkkala, J, Saarma, M, Murakata, C, Camoratto, A M, Walton, K M, Ylikoski, J
Published in The Journal of neuroscience (01.01.2000)
Published in The Journal of neuroscience (01.01.2000)
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A novel steroidal selective steroid sulfatase inhibitor KW-2581 inhibits sulfated-estrogen dependent growth of breast cancer cells in vitro and in animal models
ISHIDA, Hiroyuki, NAKATA, Taisuke, LI, Pui-Kai, KUWABARA, Takashi, AKINAGA, Shiro, SUZUKI, Masayo, SHIOTSU, Yukimasa, TANAKA, Hideyuki, SATO, Natsuko, TERASAKI, Yoko, TAKEBAYASHI, Miho, ANAZAWA, Hideharu, MURAKATA, Chikara
Published in Breast cancer research and treatment (01.12.2007)
Published in Breast cancer research and treatment (01.12.2007)
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Synthesis and Antitumor Activity of Novel O-Carbamoylmethyloxime Derivatives of Radicicol
Ikuina, Yoji, Amishiro, Nobuyoshi, Miyata, Mayumi, Narumi, Hiroaki, Ogawa, Harumi, Akiyama, Tadakazu, Shiotsu, Yukimasa, Akinaga, Shiro, Murakata, Chikara
Published in Journal of medicinal chemistry (05.06.2003)
Published in Journal of medicinal chemistry (05.06.2003)
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Role of steroid sulfatase in local formation of estrogen in post-menopausal breast cancer patients
Nakata, Taisuke, Takashima, Shigemitsu, Shiotsu, Yukimasa, Murakata, Chikara, Ishida, Hiroyuki, Akinaga, Shiro, Li, Pui-Ki, Sasano, Hironobu, Suzuki, Takashi, Saeki, Toshiaki
Published in Journal of steroid biochemistry and molecular biology (01.09.2003)
Published in Journal of steroid biochemistry and molecular biology (01.09.2003)
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Conference Proceeding
Neurotrophic 3,9-Bis[(alkylthio)methyl]- and -Bis(alkoxymethyl)-K-252a Derivatives
Kaneko, Masami, Saito, Yutaka, Saito, Hiromitsu, Matsumoto, Tadashi, Matsuda, Yuzuru, Vaught, Jeffry L, Dionne, Craig A, Angeles, Thelma S, Glicksman, Marcie A, Neff, Nicola T, Rotella, David P, Kauer, James C, Mallamo, John P, Hudkins, Robert L, Murakata, Chikara
Published in Journal of medicinal chemistry (06.06.1997)
Published in Journal of medicinal chemistry (06.06.1997)
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K-252 compounds, novel and potent inhibitors of protein kinase C and cyclic nucleotide-dependent protein kinases
Kase, Hiroshi, Iwahashi, Kazuyuki, Nakanishi, Satoshi, Matsuda, Yuzuru, Yamada, Koji, Takahashi, Mitsuru, Murakata, Chikara, Sato, Akira, Kaneko, Masami
Published in Biochemical and biophysical research communications (30.01.1987)
Published in Biochemical and biophysical research communications (30.01.1987)
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A Novel Eg5 Inhibitor (LY2523355) Causes Mitotic Arrest and Apoptosis in Cancer Cells and Shows Potent Antitumor Activity in Xenograft Tumor Models
Ye, Xiang S, Fan, Li, Van Horn, Robert D, Nakai, Ryuichiro, Ohta, Yoshihisa, Akinaga, Shiro, Murakata, Chikara, Yamashita, Yoshinori, Yin, Tinggui, Credille, Kelly M, Donoho, Gregory P, Merzoug, Farhana F, Li, Heng, Aggarwal, Amit, Blanchard, Kerry, Westin, Eric H
Published in Molecular cancer therapeutics (01.11.2015)
Published in Molecular cancer therapeutics (01.11.2015)
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CEP-751 inhibits trk receptor tyrosine kinase activityin vitro and exhibits anti-tumor activity
Camoratto, Anna Marie, Jani, Jitesh P., Angeles, Thelma S., Maroney, Anna C., Sanders, Christa Y., Murakata, Chikara, Neff, Nicola T., Vaught, Jeffry L., Isaacs, John T., Dionne, Craig A.
Published in International journal of cancer (07.08.1997)
Published in International journal of cancer (07.08.1997)
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KF25706, a novel oxime derivative of radicicol, exhibits in vivo antitumor activity via selective depletion of Hsp90 binding signaling molecules
SOGA, S, NECKERS, L. M, AKINAGA, S, SCHULTE, T. W, SHIOTSU, Y, AKASAKA, K, NARUMI, H, AGATSUMA, T, IKUINA, Y, MURAKATA, C, TAMAOKI, T
Published in Cancer research (Chicago, Ill.) (15.06.1999)
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Published in Cancer research (Chicago, Ill.) (15.06.1999)
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Glycolipids with nonreducing end α‐mannosyl residues that have the potential to activate invariant Vα19 NKT cells
Shimamura, Michio, Huang, Yi‐Ying, Okamoto, Naoki, Watanabe, Yutaka, Murakami, Yoshiko, Kinoshita, Taroh, Hirabayashi, Yoshio, Murakata, Chikara, Ito, Yukishige, Ogawa, Tomoya
Published in The FEBS journal (01.06.2007)
Published in The FEBS journal (01.06.2007)
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Glycolipids with nonreducing end alpha -mannosyl residues that have the potential to activate invariant V alpha 19 NKT cells
Shimamura, Michio, Huang, Yi-Ying, Okamoto, Naoki, Watanabe, Yutaka, Murakami, Yoshiko, Kinoshita, Taroh, Hirabayashi, Yoshio, Murakata, Chikara, Ito, Yukishige, Ogawa, Tomoya
Published in The FEBS journal (01.06.2007)
Published in The FEBS journal (01.06.2007)
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Novel oxime derivatives of radicicol induce erythroid differentiation associated with preferential G1 phase accumulation against chronic myelogenous leukemia cells through destabilization of Bcr-Abl with Hsp90 complex
Shiotsu, Yukimasa, Neckers, Leonard M., Wortman, Ivo, An, Won G., Schulte, Theodor W., Soga, Shiro, Murakata, Chikara, Tamaoki, Tatsuya, Akinaga, Shiro
Published in Blood (15.09.2000)
Published in Blood (15.09.2000)
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Sustained in vivo regression of Dunning H rat prostate cancers treated with combinations of androgen ablation and Trk tyrosine kinase inhibitors, CEP-751 (KT-6587) or CEP-701 (KT-5555)
GEORGE, D. J, DIONNE, C. A, JANI, J, ANGELES, T, MURAKATA, C, LAMB, J, ISAACS, J. T
Published in Cancer research (Chicago, Ill.) (15.05.1999)
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Published in Cancer research (Chicago, Ill.) (15.05.1999)
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Abstract A62: A novel Eg5 inhibitor that causes mitotic arrest leading to rapid cancer cell death shows broad-spectrum antitumor activity in preclinical xenograft tumor models
Ye, Xiang S., Fan, Li, Van Horn, Robert, Yin, Tinggui, Nakai, Ryuichiro, Ohta, Yoshihisa, Credille, Kelly, Donoho, Gregory, Akinaga, Shiro, Murakata, Chikara, Perkins, Everett, Ocheltree, Scott, Yamashita, Yoshinori, Blanchard, Kerry, Westin, Eric
Published in Molecular cancer therapeutics (10.12.2009)
Published in Molecular cancer therapeutics (10.12.2009)
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Mixed lineage kinase activity of indolocarbazole analogues
Murakata, Chikara, Kaneko, Masami, Gessner, George, Angeles, Thelma S, Ator, Mark A, O'Kane, Teresa M, McKenna, Beth Ann W, Thomas, Beth Ann, Mathiasen, Joanne R, Saporito, Michael S, Bozyczko-Coyne, Donna, Hudkins, Robert L
Published in Bioorganic & medicinal chemistry letters (21.01.2002)
Published in Bioorganic & medicinal chemistry letters (21.01.2002)
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Glycolipids with nonreducing end [alpha]-mannosyl residues that have the potential to activate invariant V[alpha]19 NKT cells
Shimamura, Michio, Yi-Ying, Huang, Okamoto, Naoki, Watanabe, Yutaka, Murakami, Yoshiko, Kinoshita, Taroh, Hirabayashi, Yoshio, Murakata, Chikara, Ito, Yukishige, Ogawa, Tomoya
Published in The FEBS journal (01.06.2007)
Published in The FEBS journal (01.06.2007)
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